NO20091107L - 2-amido-4-isoksazolyltiazolforbindelser som oppviser ATP-utnyttende enzyminhibitoraktivitet, og preparater og anvendelser derav - Google Patents
2-amido-4-isoksazolyltiazolforbindelser som oppviser ATP-utnyttende enzyminhibitoraktivitet, og preparater og anvendelser deravInfo
- Publication number
- NO20091107L NO20091107L NO20091107A NO20091107A NO20091107L NO 20091107 L NO20091107 L NO 20091107L NO 20091107 A NO20091107 A NO 20091107A NO 20091107 A NO20091107 A NO 20091107A NO 20091107 L NO20091107 L NO 20091107L
- Authority
- NO
- Norway
- Prior art keywords
- isoxazolylthiazole
- amido
- enzyme inhibitor
- utilizing enzyme
- inhibitor activity
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 230000000694 effects Effects 0.000 title abstract 3
- 229940125532 enzyme inhibitor Drugs 0.000 title abstract 3
- 239000002532 enzyme inhibitor Substances 0.000 title abstract 3
- 238000002360 preparation method Methods 0.000 title 1
- 230000001747 exhibiting effect Effects 0.000 abstract 3
- 102000004190 Enzymes Human genes 0.000 abstract 1
- 108090000790 Enzymes Proteins 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US83824306P | 2006-08-16 | 2006-08-16 | |
| PCT/US2007/075648 WO2008022002A2 (en) | 2006-08-16 | 2007-08-09 | 2-amido-4-isoxazolyl thiazole compounds exhibiting atp-utilizing enzyme inhibitory activity, and compositions, and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20091107L true NO20091107L (no) | 2009-05-15 |
Family
ID=38982868
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20091107A NO20091107L (no) | 2006-08-16 | 2009-03-13 | 2-amido-4-isoksazolyltiazolforbindelser som oppviser ATP-utnyttende enzyminhibitoraktivitet, og preparater og anvendelser derav |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20080242709A1 (ja) |
| EP (1) | EP2057157A2 (ja) |
| JP (1) | JP2010500998A (ja) |
| KR (1) | KR20090038905A (ja) |
| CN (1) | CN101522675A (ja) |
| AU (1) | AU2007286111A1 (ja) |
| BR (1) | BRPI0714535A2 (ja) |
| CA (1) | CA2659276A1 (ja) |
| CR (1) | CR10616A (ja) |
| IL (1) | IL196717A0 (ja) |
| MA (1) | MA30708B1 (ja) |
| MX (1) | MX2009001625A (ja) |
| NO (1) | NO20091107L (ja) |
| RU (1) | RU2009109205A (ja) |
| WO (1) | WO2008022002A2 (ja) |
| ZA (1) | ZA200900605B (ja) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG155222A1 (en) * | 2004-08-13 | 2009-09-30 | Genentech Inc | Thiazole based inhibitors of atp-utilizing enzymes |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG155222A1 (en) * | 2004-08-13 | 2009-09-30 | Genentech Inc | Thiazole based inhibitors of atp-utilizing enzymes |
-
2007
- 2007-08-09 EP EP07800075A patent/EP2057157A2/en not_active Withdrawn
- 2007-08-09 AU AU2007286111A patent/AU2007286111A1/en not_active Abandoned
- 2007-08-09 WO PCT/US2007/075648 patent/WO2008022002A2/en not_active Ceased
- 2007-08-09 CN CNA2007800367521A patent/CN101522675A/zh active Pending
- 2007-08-09 RU RU2009109205/04A patent/RU2009109205A/ru not_active Application Discontinuation
- 2007-08-09 CA CA002659276A patent/CA2659276A1/en not_active Abandoned
- 2007-08-09 MX MX2009001625A patent/MX2009001625A/es unknown
- 2007-08-09 KR KR1020097003005A patent/KR20090038905A/ko not_active Withdrawn
- 2007-08-09 ZA ZA200900605A patent/ZA200900605B/xx unknown
- 2007-08-09 JP JP2009524744A patent/JP2010500998A/ja active Pending
- 2007-08-09 US US11/836,528 patent/US20080242709A1/en not_active Abandoned
- 2007-08-09 BR BRPI0714535-7A patent/BRPI0714535A2/pt not_active Application Discontinuation
-
2009
- 2009-01-26 IL IL196717A patent/IL196717A0/en unknown
- 2009-02-13 CR CR10616A patent/CR10616A/es unknown
- 2009-03-09 MA MA31702A patent/MA30708B1/fr unknown
- 2009-03-13 NO NO20091107A patent/NO20091107L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US20080242709A1 (en) | 2008-10-02 |
| JP2010500998A (ja) | 2010-01-14 |
| BRPI0714535A2 (pt) | 2013-07-02 |
| MX2009001625A (es) | 2009-02-23 |
| IL196717A0 (en) | 2009-11-18 |
| MA30708B1 (fr) | 2009-09-01 |
| EP2057157A2 (en) | 2009-05-13 |
| ZA200900605B (en) | 2010-04-28 |
| RU2009109205A (ru) | 2010-09-27 |
| WO2008022002A2 (en) | 2008-02-21 |
| AU2007286111A1 (en) | 2008-02-21 |
| CR10616A (es) | 2009-05-25 |
| CA2659276A1 (en) | 2008-02-21 |
| KR20090038905A (ko) | 2009-04-21 |
| WO2008022002A3 (en) | 2008-10-09 |
| CN101522675A (zh) | 2009-09-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |