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NO20084328L - Nye forbindelser - Google Patents

Nye forbindelser

Info

Publication number
NO20084328L
NO20084328L NO20084328A NO20084328A NO20084328L NO 20084328 L NO20084328 L NO 20084328L NO 20084328 A NO20084328 A NO 20084328A NO 20084328 A NO20084328 A NO 20084328A NO 20084328 L NO20084328 L NO 20084328L
Authority
NO
Norway
Prior art keywords
new connections
compounds
inflammation
medicament
manufacture
Prior art date
Application number
NO20084328A
Other languages
English (en)
Inventor
Keith Biggadike
Anthony William James Cooper
David House
Iain Mcfarlane Mclay
Grahame Robert Woollam
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0607840A external-priority patent/GB0607840D0/en
Priority claimed from GB0620382A external-priority patent/GB0620382D0/en
Priority claimed from GB0706516A external-priority patent/GB0706516D0/en
Priority claimed from GB0706515A external-priority patent/GB0706515D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20084328L publication Critical patent/NO20084328L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4409—Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 4, e.g. isoniazid, iproniazid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Foreliggende oppfinnelse tilveiebringer forbindelser med formel (I): farmasøytiske preparater omfattende forbindelsene, og anvendelse av forbindelsene for fremstilling av et medikament, spesielt for behandling av inflammasjon og/eller allergiske lidelser.
NO20084328A 2006-04-20 2008-10-16 Nye forbindelser NO20084328L (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0607840A GB0607840D0 (en) 2006-04-20 2006-04-20 Novel compounds
GB0620382A GB0620382D0 (en) 2006-10-13 2006-10-13 Novel compounds
GB0706516A GB0706516D0 (en) 2007-04-03 2007-04-03 Novel compounds
GB0706515A GB0706515D0 (en) 2007-04-03 2007-04-03 Novel compounds
PCT/EP2007/053795 WO2007122165A1 (en) 2006-04-20 2007-04-18 Novel compounds

Publications (1)

Publication Number Publication Date
NO20084328L true NO20084328L (no) 2008-11-18

Family

ID=38093410

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20084328A NO20084328L (no) 2006-04-20 2008-10-16 Nye forbindelser

Country Status (17)

Country Link
US (2) US7943651B2 (no)
EP (1) EP2013185B1 (no)
JP (1) JP5298008B2 (no)
KR (1) KR20090003349A (no)
AR (1) AR060536A1 (no)
AU (1) AU2007242851A1 (no)
BR (1) BRPI0710240A2 (no)
CA (1) CA2649509A1 (no)
CR (1) CR10353A (no)
EA (1) EA200801997A1 (no)
ES (1) ES2388351T3 (no)
MA (1) MA30406B1 (no)
MX (1) MX2008013411A (no)
NO (1) NO20084328L (no)
PE (1) PE20071227A1 (no)
TW (1) TW200811111A (no)
WO (1) WO2007122165A1 (no)

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EA201691068A1 (ru) * 2013-11-22 2016-09-30 Тева Брэндид Фармасьютикал Продактс Ар Энд Ди, Инк. Ингалируемое лекарственное средство
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US10626106B2 (en) * 2017-12-18 2020-04-21 Gruenenthal Gmbh Substituted pyrrolidine amides I
TW201927769A (zh) 2017-12-18 2019-07-16 德商歌林達有限公司 經取代之吡咯啶醯胺ｉｉ
JP7446316B2 (ja) 2019-01-11 2024-03-08 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング 置換ピロリジンアミドｉｉｉ
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EP3986886A2 (en) 2019-06-19 2022-04-27 Grünenthal GmbH Substituted pyrrolidine amides v
CN116194114A (zh) 2020-03-26 2023-05-30 葛兰素史密斯克莱知识产权发展有限公司 用于防止或治疗病毒感染的组织蛋白酶抑制剂
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PE20071227A1 (es) 2008-02-18
KR20090003349A (ko) 2009-01-09
JP2009534353A (ja) 2009-09-24
BRPI0710240A2 (pt) 2011-08-09
WO2007122165A1 (en) 2007-11-01
US7943651B2 (en) 2011-05-17
CA2649509A1 (en) 2007-11-01
AR060536A1 (es) 2008-06-25
US20070265326A1 (en) 2007-11-15
US8178573B2 (en) 2012-05-15
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TW200811111A (en) 2008-03-01
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CR10353A (es) 2009-01-09
AU2007242851A1 (en) 2007-11-01
MX2008013411A (es) 2008-11-04
ES2388351T3 (es) 2012-10-11

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