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NO20082125L - Substituerte benzokondenserte derivater og deres anvendelse som vanilloidreseptorligander - Google Patents

Substituerte benzokondenserte derivater og deres anvendelse som vanilloidreseptorligander

Info

Publication number
NO20082125L
NO20082125L NO20082125A NO20082125A NO20082125L NO 20082125 L NO20082125 L NO 20082125L NO 20082125 A NO20082125 A NO 20082125A NO 20082125 A NO20082125 A NO 20082125A NO 20082125 L NO20082125 L NO 20082125L
Authority
NO
Norway
Prior art keywords
receptor ligands
substituted benzo
fused derivatives
vanilloid receptor
methods
Prior art date
Application number
NO20082125A
Other languages
English (en)
Norwegian (no)
Inventor
Laxmikant Altmaram Gharat
Uday Mukund Joshi
Neelima Khairatkar Joshi
Original Assignee
Glenmark Pharmaceuticals Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37603267&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20082125(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glenmark Pharmaceuticals Sa filed Critical Glenmark Pharmaceuticals Sa
Publication of NO20082125L publication Critical patent/NO20082125L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Otolaryngology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
NO20082125A 2005-10-07 2008-05-06 Substituerte benzokondenserte derivater og deres anvendelse som vanilloidreseptorligander NO20082125L (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN1269MU2005 2005-10-07
US73066005P 2005-10-26 2005-10-26
IN996MU2006 2006-06-26
US80720506P 2006-07-13 2006-07-13
PCT/IB2006/002814 WO2007042906A1 (fr) 2005-10-07 2006-10-09 Dérivés benzofusionnés substitués et leur utilisation en tant que ligands des récepteurs vanilloïdes

Publications (1)

Publication Number Publication Date
NO20082125L true NO20082125L (no) 2008-07-07

Family

ID=37603267

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20082125A NO20082125L (no) 2005-10-07 2008-05-06 Substituerte benzokondenserte derivater og deres anvendelse som vanilloidreseptorligander

Country Status (12)

Country Link
US (4) US7842703B2 (fr)
EP (1) EP1931681B1 (fr)
JP (1) JP2009511465A (fr)
KR (1) KR20080064972A (fr)
AP (1) AP2008004432A0 (fr)
AR (1) AR057543A1 (fr)
CA (1) CA2624307C (fr)
EA (1) EA200801013A1 (fr)
IL (1) IL190587A0 (fr)
NO (1) NO20082125L (fr)
TW (1) TW200801013A (fr)
WO (1) WO2007042906A1 (fr)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
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JP2009511465A (ja) * 2005-10-07 2009-03-19 グレンマーク・ファーマシューティカルズ・エスエー 置換ベンゾ縮合誘導体およびバニロイド受容体リガンドとしてのその使用
CN101426498A (zh) * 2006-04-18 2009-05-06 艾博特公司 香草素受体亚型1（vr1）的拮抗剂及其用途
EP2032585B1 (fr) 2006-05-24 2014-07-23 Boehringer Ingelheim International GmbH Pteridines substituteés comme agents therapeutiques
WO2008110863A1 (fr) * 2007-03-15 2008-09-18 Glenmark Pharmaceuticals S.A. Dérivés d'indazole et leur utilisation comme ligands des récepteurs vanilloïdes
KR101518525B1 (ko) 2007-10-16 2015-05-15 산텐 세이야꾸 가부시키가이샤 Ｔｒｐｖ1 매개성 질환 치료제
AU2008344922A1 (en) * 2007-12-18 2012-01-19 Glenmark Pharmaceuticals, S.A. Chromane derivatives as TRPV3 modulators
WO2009081219A1 (fr) * 2007-12-20 2009-07-02 Glenmark Pharmaceuticals, S.A. Dérivés quinazoline utiles en tant que modulateurs d'un récepteur vanilloïde
US8349846B2 (en) * 2008-01-11 2013-01-08 Glenmark Pharmaceuticals, S.A. Fused pyrimidine derivatives as TRPV3 modulators
US8557872B2 (en) 2008-01-28 2013-10-15 Amorepacific Corporation Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same
WO2009095726A1 (fr) * 2008-01-29 2009-08-06 Glenmark Pharmaceuticals, S.A. Dérivés d'acrylamide en tant que modulateurs du récepteur vanilloïde de type 1
CA2728405A1 (fr) 2008-06-17 2010-01-14 Glenmark Pharmaceuticals, S.A. Derives du chromane comme modulateurs de trpv3
KR101621444B1 (ko) 2008-07-02 2016-05-19 (주)아모레퍼시픽 바닐로이드 수용체 길항제로 작용하는 신규 화합물, 이의 이성질체 또는 이의 약제학적으로 허용 가능한 염, 및 이를 포함하는 약학 조성물
WO2010023512A1 (fr) * 2008-08-28 2010-03-04 Matrix Laboratories Ltd. Nouveaux modulateurs de récepteur vanilloïde, procédé pour leur préparation et compositions pharmaceutiques contenant ceux-ci
TW201020236A (en) * 2008-10-17 2010-06-01 Abbott Lab TRPV1 antagonists
EP2352727A1 (fr) * 2008-10-17 2011-08-10 Abbott Laboratories Antagonistes de trpv1
US8318928B2 (en) 2008-12-15 2012-11-27 Glenmark Pharmaceuticals, S.A. Fused imidazole carboxamides as TRPV3 modulators
MX2011006821A (es) 2008-12-26 2012-01-03 Glenmark Pharmaceuticals Sa Derivados de imidazol fusionados como antagonistas de trpv3.
US8349852B2 (en) 2009-01-13 2013-01-08 Novartis Ag Quinazolinone derivatives useful as vanilloid antagonists
EP2531510B1 (fr) 2010-02-01 2014-07-23 Novartis AG Dérivés de pyrazolo[5,1-b]utilisés en tant qu'antagonistes du récepteur de crf-1
AR080056A1 (es) 2010-02-01 2012-03-07 Novartis Ag Derivados de ciclohexil-amida como antagonistas de los receptores de crf
US8835444B2 (en) 2010-02-02 2014-09-16 Novartis Ag Cyclohexyl amide derivatives as CRF receptor antagonists
WO2012049555A1 (fr) 2010-10-13 2012-04-19 Lupin Limited Composés spirocycliques en tant que modulateurs de canaux sodiques dépendants du voltage
EP2635281B1 (fr) * 2010-11-03 2018-03-14 University Of Hawaii Procédés et compositions pour la prévention et le traitement de l'hypertrophie cardiaque
UY33966A (es) 2011-03-25 2012-10-31 Abbott Lab Antagonistas del receptor transitorio potencial de vanilloides 1 (trpv1)
WO2013096223A1 (fr) 2011-12-19 2013-06-27 Abbvie Inc. Antagonistes de trpv1
US8969325B2 (en) 2011-12-19 2015-03-03 Abbvie Inc. TRPV1 antagonists
US8796328B2 (en) 2012-06-20 2014-08-05 Abbvie Inc. TRPV1 antagonists
WO2014203217A1 (fr) 2013-06-21 2014-12-24 Lupin Limited Composés hétérocycliques substitués utiles en tant que modulateurs de crac
EP3013810A1 (fr) 2013-06-24 2016-05-04 Lupin Limited Dérivés de chromane et de chromène et leur utilisation en tant que modulateurs de crac
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AR057543A1 (es) 2007-12-05
US20110021549A1 (en) 2011-01-27
US20120041011A1 (en) 2012-02-16
US20080269253A1 (en) 2008-10-30
EA200801013A1 (ru) 2008-10-30
KR20080064972A (ko) 2008-07-10
CA2624307A1 (fr) 2007-04-19
AU2006300871A1 (en) 2007-04-19
EP1931681A1 (fr) 2008-06-18
US7842703B2 (en) 2010-11-30
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US20120277259A1 (en) 2012-11-01

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