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NO20080325L - Forbindelser og deres salter som er spesifikke overfor PPAR-reseptorer og EGF-reseptorer samt deres anvendelse innen medisin - Google Patents

Forbindelser og deres salter som er spesifikke overfor PPAR-reseptorer og EGF-reseptorer samt deres anvendelse innen medisin

Info

Publication number
NO20080325L
NO20080325L NO20080325A NO20080325A NO20080325L NO 20080325 L NO20080325 L NO 20080325L NO 20080325 A NO20080325 A NO 20080325A NO 20080325 A NO20080325 A NO 20080325A NO 20080325 L NO20080325 L NO 20080325L
Authority
NO
Norway
Prior art keywords
compounds
ppar
medicine
well
egf receptors
Prior art date
Application number
NO20080325A
Other languages
English (en)
Other versions
NO340680B1 (no
Inventor
Giancarlo Naccari
Sergio Baroni
Original Assignee
Giuliani Int Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37579831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20080325(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Giuliani Int Ltd filed Critical Giuliani Int Ltd
Publication of NO20080325L publication Critical patent/NO20080325L/no
Publication of NO340680B1 publication Critical patent/NO340680B1/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/38—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/40—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/42—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton with carboxyl groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by saturated carbon chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/52—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C07C229/54—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C229/60—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring with amino and carboxyl groups bound in meta- or para- positions

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)

Abstract

Foreliggende oppfinnelse angår forbindelser omfattende den generelle formel (I): (I) hvor: R1 og R2, som kan være like eller forskjellige, er valgt fra gruppen omfattende -H eller en lineær eller forgrenet alkylgruppe som har fra 1 til 6 karbonatomer eller sammen danner en aromatisk eller alifatisk ring med 5 eller 6 atomer; Y og Z, som kan være like eller forskjellige, er valgt fra gruppen omfattende -H, -OH, -COOH, -OR3, -CH(OR3)COOH, hvor R3 er valgt fra H, fenyl, benzyl, -CF3 eller -CF2CF3, vinyl, allyl og en lineær eller forgrenet alkylgruppe som har fra 1 til 6 karbonatomer.
NO20080325A 2005-07-22 2008-01-18 Forbindelser og deres salter som er spesifikke overfor PPAR-reseptorer og EGF-reseptorer samt deres anvendelse innen medisin NO340680B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT000389A ITRM20050389A1 (it) 2005-07-22 2005-07-22 Composti e loro sali specifici per i recettori ppar ed i recettori per l'egf e loro uso in campo medico.
PCT/IE2006/000078 WO2007010516A2 (en) 2005-07-22 2006-07-24 Compounds and their salts specific to the ppar receptors and the egf receptors and their use in the medical field

Publications (2)

Publication Number Publication Date
NO20080325L true NO20080325L (no) 2008-04-16
NO340680B1 NO340680B1 (no) 2017-05-29

Family

ID=37579831

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20080325A NO340680B1 (no) 2005-07-22 2008-01-18 Forbindelser og deres salter som er spesifikke overfor PPAR-reseptorer og EGF-reseptorer samt deres anvendelse innen medisin

Country Status (23)

Country Link
US (6) US8153841B2 (no)
EP (1) EP1910270B3 (no)
JP (1) JP5312026B2 (no)
KR (1) KR101317519B1 (no)
CN (2) CN101243039B (no)
AU (1) AU2006271165C1 (no)
CA (1) CA2616146C (no)
CY (1) CY1114294T1 (no)
DK (1) DK1910270T6 (no)
EA (2) EA014665B3 (no)
ES (1) ES2421260T7 (no)
HR (1) HRP20130549T4 (no)
IL (2) IL188878A (no)
IT (1) ITRM20050389A1 (no)
MX (1) MX366596B (no)
NO (1) NO340680B1 (no)
NZ (2) NZ592228A (no)
PL (1) PL1910270T6 (no)
PT (1) PT1910270E (no)
SI (1) SI1910270T1 (no)
UA (1) UA100359C2 (no)
WO (1) WO2007010516A2 (no)
ZA (2) ZA200801671B (no)

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Also Published As

Publication number Publication date
KR101317519B1 (ko) 2013-10-15
US9561202B2 (en) 2017-02-07
CY1114294T1 (el) 2016-08-31
WO2007010516A2 (en) 2007-01-25
HRP20130549T1 (en) 2013-07-31
CA2616146A1 (en) 2007-01-25
EA014665B3 (ru) 2016-09-30
PL1910270T3 (pl) 2013-09-30
US9133099B2 (en) 2015-09-15
NZ592228A (en) 2012-10-26
EP1910270B1 (en) 2013-05-08
ITRM20050389A1 (it) 2007-01-23
NO340680B1 (no) 2017-05-29
US8710100B2 (en) 2014-04-29
US20130005813A1 (en) 2013-01-03
PT1910270E (pt) 2013-07-17
CN101243039B (zh) 2013-04-03
UA100359C2 (uk) 2012-12-25
CN102020577A (zh) 2011-04-20
ES2421260T7 (es) 2016-10-11
US20170312239A1 (en) 2017-11-02
US20090048343A1 (en) 2009-02-19
DK1910270T3 (da) 2013-07-01
JP2009502777A (ja) 2009-01-29
CN101243039A (zh) 2008-08-13
EA200800372A1 (ru) 2008-06-30
US9345680B2 (en) 2016-05-24
US10016381B2 (en) 2018-07-10
IL188878A0 (en) 2008-04-13
CA2616146C (en) 2015-06-30
JP5312026B2 (ja) 2013-10-09
US20150045436A1 (en) 2015-02-12
US8153841B2 (en) 2012-04-10
US20150265562A1 (en) 2015-09-24
KR20080039428A (ko) 2008-05-07
EA014665B1 (ru) 2010-12-30
CN102020577B (zh) 2013-03-13
WO2007010516A3 (en) 2007-03-29
ZA200801671B (en) 2011-02-23
AU2006271165A1 (en) 2007-01-25
AU2006271165B2 (en) 2012-01-19
EP1910270B3 (en) 2016-05-11
BRPI0613396A2 (pt) 2011-01-11
DK1910270T6 (en) 2016-08-29
AU2006271165C1 (en) 2016-11-17
EP1910270A2 (en) 2008-04-16
EA201000708A1 (ru) 2010-10-29
ES2421260T3 (es) 2013-08-30
BRPI0613396A8 (pt) 2017-12-26
EA017566B1 (ru) 2013-01-30
HRP20130549T4 (hr) 2016-07-15
IL205992A (en) 2014-05-28
US20150265563A1 (en) 2015-09-24
IL188878A (en) 2013-04-30
ZA201008268B (en) 2012-04-25
PL1910270T6 (pl) 2017-05-31
NZ566045A (en) 2012-04-27
SI1910270T1 (sl) 2013-08-30
MX366596B (es) 2019-07-15

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