NO20072634L - Antiinfektive lipopeptider - Google Patents
Antiinfektive lipopeptiderInfo
- Publication number
- NO20072634L NO20072634L NO20072634A NO20072634A NO20072634L NO 20072634 L NO20072634 L NO 20072634L NO 20072634 A NO20072634 A NO 20072634A NO 20072634 A NO20072634 A NO 20072634A NO 20072634 L NO20072634 L NO 20072634L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- lipopeptides
- infective
- relates
- methods
- Prior art date
Links
- 108010028921 Lipopeptides Proteins 0.000 title 1
- 230000002924 anti-infective effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- OHRURASPPZQGQM-GCCNXGTGSA-N romidepsin Chemical class O1C(=O)[C@H](C(C)C)NC(=O)C(=C/C)/NC(=O)[C@H]2CSSCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)C(=O)N2 OHRURASPPZQGQM-GCCNXGTGSA-N 0.000 abstract 2
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Biochemistry (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
Abstract
Foreliggende oppfinnelse angår nye depsipeptidforbindelser. Oppfinnelsen angår også farmasøytiske preparater av disse forbindelser og metoder for anvendelse av disse forbindelser som antibakterielle forbindelser. Oppfinnelsen angår også metoder for å produsere disse nye depsipeptidforbindelsene og mellomprodukter anvendt for fremstilling av disse forbindelsene.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US62705604P | 2004-11-12 | 2004-11-12 | |
| US71070505P | 2005-08-23 | 2005-08-23 | |
| PCT/US2005/040919 WO2006110185A2 (en) | 2004-11-12 | 2005-11-11 | Antiinfective lipopeptides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20072634L true NO20072634L (no) | 2007-08-09 |
Family
ID=37087468
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20072634A NO20072634L (no) | 2004-11-12 | 2007-05-24 | Antiinfektive lipopeptider |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP1814588A2 (no) |
| JP (1) | JP2008519848A (no) |
| KR (1) | KR20070086038A (no) |
| AU (1) | AU2005330517A1 (no) |
| BR (1) | BRPI0517830A (no) |
| CA (1) | CA2587848A1 (no) |
| IL (1) | IL183109A0 (no) |
| NO (1) | NO20072634L (no) |
| RU (1) | RU2007121705A (no) |
| WO (1) | WO2006110185A2 (no) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2379580T3 (da) * | 2008-12-22 | 2014-01-20 | Cubist Pharm Inc | Hidtil ukendte antibakterielle midler til behandling af gram-positive infektioner |
| RU2013157188A (ru) * | 2011-05-26 | 2015-07-10 | Кьюбист Фармасьютикалз, Инк. | Композиции св-183,315 и относящиеся к ним способы |
| KR101723649B1 (ko) | 2014-10-23 | 2017-04-06 | 서울대학교산학협력단 | 신규한 펩티드 화합물, 이의 생산 방법, 및 이의 용도 |
| CN113061164B (zh) * | 2021-03-29 | 2023-01-10 | 四川大学 | 环脂肽类化合物及其在抗类风湿关节炎药物中的应用 |
| EP4475890A1 (en) | 2022-02-09 | 2024-12-18 | Teitur Trophics ApS | Novel peptides |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2394350A1 (en) * | 1999-12-15 | 2001-06-21 | Cubist Pharmaceuticals, Inc. | Lipopeptides as antibacterial agents |
| WO2001044272A2 (en) * | 1999-12-15 | 2001-06-21 | Cubist Pharmaceuticals, Inc. | Daptomycin analogs as antibacterial agents |
| US6794490B2 (en) * | 1999-12-15 | 2004-09-21 | Cubist Pharmaceuticals, Inc. | Lipopeptides as antibacterial agents |
| CN100352836C (zh) * | 2001-08-06 | 2007-12-05 | 卡比斯特制药公司 | 新颖的缩肽和制备它们的方法 |
| CA2456552A1 (en) * | 2001-08-06 | 2003-02-20 | Cubist Pharmaceuticals, Inc. | Compositions and methods relating to the daptomycin biosynthetic gene cluster |
-
2005
- 2005-11-11 BR BRPI0517830-4A patent/BRPI0517830A/pt not_active IP Right Cessation
- 2005-11-11 RU RU2007121705/04A patent/RU2007121705A/ru not_active Application Discontinuation
- 2005-11-11 CA CA002587848A patent/CA2587848A1/en not_active Abandoned
- 2005-11-11 JP JP2007541346A patent/JP2008519848A/ja not_active Withdrawn
- 2005-11-11 WO PCT/US2005/040919 patent/WO2006110185A2/en not_active Ceased
- 2005-11-11 AU AU2005330517A patent/AU2005330517A1/en not_active Abandoned
- 2005-11-11 EP EP05857738A patent/EP1814588A2/en not_active Withdrawn
- 2005-11-11 KR KR1020077013150A patent/KR20070086038A/ko not_active Withdrawn
-
2007
- 2007-05-10 IL IL183109A patent/IL183109A0/en unknown
- 2007-05-24 NO NO20072634A patent/NO20072634L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0517830A (pt) | 2008-10-21 |
| WO2006110185A3 (en) | 2007-10-25 |
| WO2006110185A2 (en) | 2006-10-19 |
| IL183109A0 (en) | 2008-04-13 |
| KR20070086038A (ko) | 2007-08-27 |
| CA2587848A1 (en) | 2006-10-19 |
| AU2005330517A2 (en) | 2006-10-19 |
| JP2008519848A (ja) | 2008-06-12 |
| RU2007121705A (ru) | 2008-12-20 |
| AU2005330517A1 (en) | 2006-10-19 |
| EP1814588A2 (en) | 2007-08-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |