NO20033700L - Isoksazolinderivater som anti-depressive midler - Google Patents

Isoksazolinderivater som anti-depressive midler

Info

Publication number: NO20033700L
Authority: NO; Norway
Prior art keywords: depressants; isoxazoline derivatives; isoxazoline; derivatives
Prior art date: 2001-02-21

Application number

NO20033700A

Other languages

English (en)

Other versions

NO20033700D0 (no

Inventor

Antonius Adrianus Hendrikus Petrus Megens

Manuel Jesus Alcazar-Vaca

Jose Ignacio Andres-Gil

Jose Maria Cid-Nunez

Joaquin Pastor-Fernandez

Godelieve Irma Christine Heylen

Xavier Jean Michel Langlois

Margaretha Henrica Maria Bakker

Thomas Horst Wolfgang Steckler

Francisco Javier Fernandez-Gadea

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-02-21

Filing date

2003-08-20

Publication date

2003-10-21

2003-08-20 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2003-08-20 Publication of NO20033700D0 publication Critical patent/NO20033700D0/no

2003-10-21 Publication of NO20033700L publication Critical patent/NO20033700L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Epidemiology (AREA)
Psychiatry (AREA)
Child & Adolescent Psychology (AREA)
Hematology (AREA)
Obesity (AREA)
Pain & Pain Management (AREA)
Diabetes (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

NO20033700A 2001-02-21 2003-08-20 Isoksazolinderivater som anti-depressive midler NO20033700L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP01200611		2001-02-21
EP01201264		2001-04-05
PCT/EP2002/001567 WO2002066484A1 (en)	2001-02-21	2002-02-13	Isoxazoline derivatives as anti-depressants

Publications (2)

Publication Number	Publication Date
NO20033700D0 NO20033700D0 (no)	2003-08-20
NO20033700L true NO20033700L (no)	2003-10-21

Family

ID=26076836

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20033700A NO20033700L (no)	2001-02-21	2003-08-20	Isoksazolinderivater som anti-depressive midler

Country Status (32)

Country	Link
US (1)	US7169786B2 (no)
EP (1)	EP1368358B1 (no)
JP (1)	JP3953424B2 (no)
KR (1)	KR100848898B1 (no)
CN (1)	CN100400540C (no)
AR (1)	AR035685A1 (no)
AT (1)	ATE337322T1 (no)
AU (1)	AU2002244717B2 (no)
BG (1)	BG107984A (no)
BR (1)	BR0207433A (no)
CA (1)	CA2437505C (no)
CY (1)	CY1106448T1 (no)
CZ (1)	CZ20032515A3 (no)
DE (1)	DE60214138T2 (no)
DK (1)	DK1368358T3 (no)
EA (1)	EA006747B1 (no)
EE (1)	EE200300398A (no)
EG (1)	EG23929A (no)
ES (1)	ES2271230T3 (no)
HR (1)	HRP20030647A2 (no)
HU (1)	HUP0303270A3 (no)
IL (2)	IL157470A0 (no)
MX (1)	MXPA03007432A (no)
MY (1)	MY137836A (no)
NO (1)	NO20033700L (no)
NZ (1)	NZ526741A (no)
PL (1)	PL208593B1 (no)
PT (1)	PT1368358E (no)
SI (1)	SI1368358T1 (no)
SK (1)	SK11612003A3 (no)
TW (1)	TWI257392B (no)
WO (1)	WO2002066484A1 (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0203299D0 (en) *	2002-02-12	2002-03-27	Glaxo Group Ltd	Novel compounds
IL164341A0 (en) *	2002-04-02	2005-12-18	Janssen Pharmaceutica Nv	Substituted amino isoxazoline derivatives and their use as anti-depressants
TW200409777A (en) *	2002-08-12	2004-06-16	Janssen Pharmaceutica Nv	C-substituted tricyclic isoxazoline derivatives and their use as anti-depressants
EP1554286B1 (en) *	2002-08-15	2010-01-27	Janssen Pharmaceutica N.V.	Fused heterocyclic isoxazoline derivatives and their use as anti-depressants
ATE387455T1 (de) *	2002-08-21	2008-03-15	Janssen Pharmaceutica Nv	C6- und c9-substituierte chromeno(4,3- c)isoxazoline und ihre verwendung als anti- depressiva
CN100516040C (zh)	2003-03-07	2009-07-22	安斯泰来制药有限公司	具有2,6-二取代苯乙烯基的含氮杂环衍生物
EP1944306A1 (en) *	2003-09-17	2008-07-16	Janssen Pharmaceutica, N.V.	Fused heterocyclic compounds as serotonin receptor modulators
KR101151653B1 (ko) *	2003-09-17	2012-06-28	얀센 파마슈티카 엔.브이.	융합된 헤테로사이클릭 화합물
AU2005308778B2 (en) *	2004-11-26	2011-03-24	Janssen Pharmaceutica N.V.	Isoxazoline-indole derivatives with an improved antipsychotic and anxiolytic activity
RU2470937C2 (ru)	2007-03-09	2012-12-27	Санофи-Авентис	Получение и применение замещенных дигидро- и тетрагидрооксазолопиримидинонов
AU2008261888A1 (en) *	2007-06-08	2008-12-18	Helicon Therapeutics, Inc.	Therapeutic pyrazoloquinoline urea derivatives
JP2011507835A (ja)	2007-12-21	2011-03-10	アンドレイ・アレクサンドロビッチ・イワシェンコ	α−アドレナリン受容体、ドーパミン、ヒスタミン、イミダゾリン及びセロトニン受容体のリガンド並びにその使用
AR078171A1 (es)	2009-09-15	2011-10-19	Sanofi Aventis	Dihidrobenzocicloalquiloximetil-oxazolopirimidinonas sustituidas, preparacion y uso de las mismas

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0361577B1 (en)	1988-09-19	1993-05-05	Akzo N.V.	Tetrahydronaphthalene and indane derivatives
US5880121A (en) *	1996-01-05	1999-03-09	Hoechst Marion Roussel Inc.	4,5-dihydronaphth (1,2-c) isoxazoles and derivatives thereof
PT892804E (pt) *	1996-04-12	2003-01-31	Janssen Pharmaceutica Nv	Derivados de isoxazolidina
HUP9602763A3 (en) *	1996-10-09	1999-05-28	Egyt Gyogyszervegyeszeti Gyar	3-phenyl isoxazole derivatives, process for producing them and pharmaceutical compositions containing the same
CA2346396C (en) *	1998-10-09	2009-04-28	Janssen Pharmaceutica N.V.	4,5-dihydro-isoxazole derivatives and their pharmaceutical use

2002
- 2002-02-13 AT AT02712909T patent/ATE337322T1/de not_active IP Right Cessation
- 2002-02-13 JP JP2002565998A patent/JP3953424B2/ja not_active Expired - Lifetime
- 2002-02-13 DK DK02712909T patent/DK1368358T3/da active
- 2002-02-13 EP EP02712909A patent/EP1368358B1/en not_active Expired - Lifetime
- 2002-02-13 ES ES02712909T patent/ES2271230T3/es not_active Expired - Lifetime
- 2002-02-13 EE EEP200300398A patent/EE200300398A/xx unknown
- 2002-02-13 NZ NZ526741A patent/NZ526741A/en unknown
- 2002-02-13 MX MXPA03007432A patent/MXPA03007432A/es active IP Right Grant
- 2002-02-13 AU AU2002244717A patent/AU2002244717B2/en not_active Expired
- 2002-02-13 CN CNB028052439A patent/CN100400540C/zh not_active Expired - Fee Related
- 2002-02-13 WO PCT/EP2002/001567 patent/WO2002066484A1/en not_active Ceased
- 2002-02-13 DE DE60214138T patent/DE60214138T2/de not_active Expired - Lifetime
- 2002-02-13 PL PL363264A patent/PL208593B1/pl unknown
- 2002-02-13 IL IL15747002A patent/IL157470A0/xx unknown
- 2002-02-13 SI SI200230433T patent/SI1368358T1/sl unknown
- 2002-02-13 EA EA200300915A patent/EA006747B1/ru not_active IP Right Cessation
- 2002-02-13 HU HU0303270A patent/HUP0303270A3/hu unknown
- 2002-02-13 PT PT02712909T patent/PT1368358E/pt unknown
- 2002-02-13 SK SK1161-2003A patent/SK11612003A3/sk unknown
- 2002-02-13 CZ CZ20032515A patent/CZ20032515A3/cs unknown
- 2002-02-13 US US10/468,555 patent/US7169786B2/en not_active Expired - Lifetime
- 2002-02-13 HR HR20030647A patent/HRP20030647A2/hr not_active Application Discontinuation
- 2002-02-13 KR KR1020037008328A patent/KR100848898B1/ko not_active Expired - Fee Related
- 2002-02-13 BR BR0207433-8A patent/BR0207433A/pt not_active IP Right Cessation
- 2002-02-13 CA CA2437505A patent/CA2437505C/en not_active Expired - Lifetime
- 2002-02-19 MY MYPI20020548A patent/MY137836A/en unknown
- 2002-02-19 EG EG20020197A patent/EG23929A/xx active
- 2002-02-20 TW TW091102853A patent/TWI257392B/zh not_active IP Right Cessation
- 2002-02-20 AR ARP020100583A patent/AR035685A1/es unknown
2003
- 2003-07-08 BG BG107984A patent/BG107984A/bg unknown
- 2003-08-19 IL IL157470A patent/IL157470A/en unknown
- 2003-08-20 NO NO20033700A patent/NO20033700L/no not_active Application Discontinuation
2006
- 2006-11-22 CY CY20061101693T patent/CY1106448T1/el unknown

Also Published As

Publication number	Publication date
HUP0303270A3 (en)	2007-03-28
JP3953424B2 (ja)	2007-08-08
US20040122037A1 (en)	2004-06-24
PL208593B1 (pl)	2011-05-31
PT1368358E (pt)	2007-01-31
AR035685A1 (es)	2004-06-23
CA2437505A1 (en)	2002-08-29
EA006747B1 (ru)	2006-04-28
KR20030076590A (ko)	2003-09-26
DE60214138D1 (de)	2006-10-05
DE60214138T2 (de)	2007-03-29
JP2004518748A (ja)	2004-06-24
TWI257392B (en)	2006-07-01
SK11612003A3 (sk)	2004-04-06
EP1368358B1 (en)	2006-08-23
MXPA03007432A (es)	2003-11-18
HUP0303270A2 (hu)	2004-01-28
EG23929A (en)	2008-01-14
HK1065537A1 (zh)	2005-02-25
ES2271230T3 (es)	2007-04-16
NO20033700D0 (no)	2003-08-20
MY137836A (en)	2009-03-31
PL363264A1 (en)	2004-11-15
CN1492871A (zh)	2004-04-28
ATE337322T1 (de)	2006-09-15
EE200300398A (et)	2003-12-15
BR0207433A (pt)	2004-06-01
HRP20030647A2 (en)	2005-06-30
CZ20032515A3 (cs)	2003-12-17
WO2002066484A1 (en)	2002-08-29
BG107984A (bg)	2004-09-30
EP1368358A1 (en)	2003-12-10
CA2437505C (en)	2010-02-09
EA200300915A1 (ru)	2004-06-24
SI1368358T1 (sl)	2007-02-28
IL157470A (en)	2008-07-08
US7169786B2 (en)	2007-01-30
CN100400540C (zh)	2008-07-09
DK1368358T3 (da)	2007-01-02
KR100848898B1 (ko)	2008-07-29
NZ526741A (en)	2004-04-30
AU2002244717B2 (en)	2007-07-19
IL157470A0 (en)	2004-03-28
CY1106448T1 (el)	2011-10-12

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Legal Events

Date	Code	Title	Description
2010-05-10	FC2A	Withdrawal, rejection or dismissal of laid open patent application