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NO20021566L - Bicykliske imidazo-5-yl-aminderivater - Google Patents

Bicykliske imidazo-5-yl-aminderivater

Info

Publication number
NO20021566L
NO20021566L NO20021566A NO20021566A NO20021566L NO 20021566 L NO20021566 L NO 20021566L NO 20021566 A NO20021566 A NO 20021566A NO 20021566 A NO20021566 A NO 20021566A NO 20021566 L NO20021566 L NO 20021566L
Authority
NO
Norway
Prior art keywords
amine derivatives
bicyclic imidazo
imidazo
bicyclic
amine
Prior art date
Application number
NO20021566A
Other languages
English (en)
Other versions
NO20021566D0 (no
Inventor
Matthias Gerlach
Corinna Maul
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19948434A external-priority patent/DE19948434A1/de
Priority claimed from DE1999148436 external-priority patent/DE19948436B4/de
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of NO20021566D0 publication Critical patent/NO20021566D0/no
Publication of NO20021566L publication Critical patent/NO20021566L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO20021566A 1999-10-08 2002-04-03 Bicykliske imidazo-5-yl-aminderivater NO20021566L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19948434A DE19948434A1 (de) 1999-10-08 1999-10-08 Substanzbibliothek enthaltend bicyclische Imidazo-5-amine und/oder bicyclische Imidazo-3-amine
DE1999148436 DE19948436B4 (de) 1999-10-08 1999-10-08 Bicyclische Imidazo-5-aminderivate
PCT/EP2000/009097 WO2001027118A2 (de) 1999-10-08 2000-09-18 Bicyclische imidazo-5-yl-aminderivate

Publications (2)

Publication Number Publication Date
NO20021566D0 NO20021566D0 (no) 2002-04-03
NO20021566L true NO20021566L (no) 2002-05-27

Family

ID=26055216

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20021566A NO20021566L (no) 1999-10-08 2002-04-03 Bicykliske imidazo-5-yl-aminderivater

Country Status (28)

Country Link
US (2) US6657064B2 (no)
EP (1) EP1218383B1 (no)
JP (1) JP2003511456A (no)
KR (1) KR20020068515A (no)
CN (1) CN1211385C (no)
AR (1) AR030030A1 (no)
AT (1) ATE413403T1 (no)
AU (1) AU781227B2 (no)
BR (1) BR0014817A (no)
CA (1) CA2388476C (no)
CO (1) CO5200851A1 (no)
CY (1) CY1110416T1 (no)
CZ (1) CZ20021242A3 (no)
DE (1) DE50015443D1 (no)
DK (1) DK1218383T3 (no)
ES (1) ES2316388T3 (no)
HU (1) HUP0203140A3 (no)
IL (2) IL149010A0 (no)
MX (1) MXPA02002837A (no)
NO (1) NO20021566L (no)
PE (1) PE20010638A1 (no)
PL (1) PL355019A1 (no)
PT (1) PT1218383E (no)
RU (1) RU2002110112A (no)
SI (1) SI1218383T1 (no)
SK (1) SK4642002A3 (no)
UY (1) UY26370A1 (no)
WO (1) WO2001027118A2 (no)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1218383E (pt) * 1999-10-08 2009-01-29 Gruenenthal Gmbh Derivados bicíclicos de imidazo-5-il-amina
AU2001251444A1 (en) 2000-04-10 2001-10-23 Merck And Co., Inc. Inhibitors of prenyl-protein transferase
DE10043845A1 (de) * 2000-09-06 2002-03-14 Gruenenthal Gmbh Verfahren zur Messung der Aktivität der NO-Synthase
KR100647583B1 (ko) * 2003-10-07 2006-11-17 삼성에스디아이 주식회사 이미다졸 고리 함유 화합물 및 이를 이용한 유기 전계발광 소자
WO2006065788A2 (en) * 2004-12-13 2006-06-22 Glaxo Group Limited Novel muscarinic acetylcholine receptor antagonists
US7923041B2 (en) * 2005-02-03 2011-04-12 Signum Biosciences, Inc. Compositions and methods for enhancing cognitive function
DE102006011574A1 (de) 2006-03-10 2007-10-31 Grünenthal GmbH Substituierte Imidazo[2,1-b]thiazol-Verbindungen und ihre Verwendung zur Herstellung von Arzneimitteln
WO2007138072A2 (en) * 2006-05-31 2007-12-06 Galapagos N.V. Triazolopyrazine compounds useful for the treatment of degenerative & inflammatory diseases
US8227603B2 (en) * 2006-08-01 2012-07-24 Cytokinetics, Inc. Modulating skeletal muscle
WO2008016648A2 (en) * 2006-08-01 2008-02-07 Cytokinetics, Incorporated Certain chemical entities, compositions and methods
US8299248B2 (en) 2006-08-02 2012-10-30 Cytokinetics, Incorporated Certain 1H-imidazo[4,5-b]pyrazin-2(3H)-ones and 1H-imidazo[4,5-b]pyrazin-2-ols and methods for their use
PT2583970E (pt) * 2006-08-02 2016-02-08 Cytokinetics Inc Certas entidades químicas, composições e métodos compreendendo imidazopirimidinas
EP2139478A4 (en) * 2007-03-30 2010-05-05 Cytokinetics Inc CHEMICAL ENTITIES, COMPOSITIONS AND METHODS
CA2704645A1 (en) * 2007-11-09 2009-05-14 The Salk Institute For Biological Studies Non-nucleoside reverse transcriptase inhibitors
NZ588376A (en) 2008-04-15 2011-06-30 Eisai R&D Man Co Ltd 3-phenylpyrazolo[5,1-b]thiazole compound having antagonism against corticotropin-releasing factor (CRF) receptor
EP2443123B1 (en) * 2009-06-15 2017-04-05 Rigel Pharmaceuticals, Inc. Small molecule inhibitors of spleen tyrosine kinase (syk)
AR078521A1 (es) 2009-10-08 2011-11-16 Eisai R&D Man Co Ltd Compuesto pirazolotiazol
EA201791043A1 (ru) 2011-07-13 2017-09-29 Сайтокинетикс, Инк. Комбинированная терапия бокового амиотрофического склероза
HUE060743T2 (hu) 2012-04-26 2023-04-28 Bristol Myers Squibb Co Gyógyszerészeti kompozíciók, amelyek tartalmaznak imidazothiadiazol- és imidazopiridazinszármazékokat mint proteáz aktívált receptor 4 (PAR4) inhibitorokat trombocitaaggregációk kezelésére
JP6181744B2 (ja) 2012-04-26 2017-08-16 ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ 血小板凝集を治療するためのプロテアーゼ活性化受容体４（ｐａｒ４）阻害剤としてのイミダゾチアジアゾール誘導体
JP6101343B2 (ja) 2012-04-26 2017-03-22 ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ 血小板凝集を治療するためのプロテアーゼ活性化受容体４（ｐａｒ４）阻害剤としてのイミダゾチアジアゾールおよびイミダゾピリダジン誘導体
US9598419B1 (en) 2014-06-24 2017-03-21 Universite De Montreal Imidazotriazine and imidazodiazine compounds
US9617279B1 (en) 2014-06-24 2017-04-11 Bristol-Myers Squibb Company Imidazooxadiazole compounds
KR102599388B1 (ko) * 2017-09-01 2023-11-09 현대자동차주식회사 피드백 제어방법 및 시스템

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW274551B (no) * 1991-04-16 1996-04-21 Takeda Pharm Industry Co Ltd
PT1218383E (pt) * 1999-10-08 2009-01-29 Gruenenthal Gmbh Derivados bicíclicos de imidazo-5-il-amina

Also Published As

Publication number Publication date
EP1218383B1 (de) 2008-11-05
US20020183320A1 (en) 2002-12-05
ES2316388T3 (es) 2009-04-16
HUP0203140A2 (hu) 2003-01-28
NO20021566D0 (no) 2002-04-03
US6657064B2 (en) 2003-12-02
SI1218383T1 (sl) 2009-04-30
CZ20021242A3 (cs) 2002-08-14
WO2001027118A2 (de) 2001-04-19
HK1047746A1 (zh) 2003-03-07
DK1218383T3 (da) 2009-01-19
IL149010A (en) 2007-06-17
KR20020068515A (ko) 2002-08-27
CA2388476A1 (en) 2001-04-19
CO5200851A1 (es) 2002-09-27
CN1402726A (zh) 2003-03-12
BR0014817A (pt) 2002-06-18
UY26370A1 (es) 2000-12-29
AU7777200A (en) 2001-04-23
ATE413403T1 (de) 2008-11-15
RU2002110112A (ru) 2003-12-20
US20040023927A1 (en) 2004-02-05
WO2001027118A3 (de) 2001-09-20
AU781227B2 (en) 2005-05-12
CA2388476C (en) 2008-08-05
JP2003511456A (ja) 2003-03-25
CY1110416T1 (el) 2015-04-29
CN1211385C (zh) 2005-07-20
PE20010638A1 (es) 2001-07-07
EP1218383A2 (de) 2002-07-03
MXPA02002837A (es) 2002-08-30
PL355019A1 (en) 2004-03-22
US6936631B2 (en) 2005-08-30
PT1218383E (pt) 2009-01-29
HUP0203140A3 (en) 2004-06-28
IL149010A0 (en) 2002-11-10
DE50015443D1 (de) 2008-12-18
AR030030A1 (es) 2003-08-13
SK4642002A3 (en) 2002-09-10

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application