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NO20000227L - Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat, fremgangsmåte for dens fremstilling og dens anvendelse - Google Patents

Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat, fremgangsmåte for dens fremstilling og dens anvendelse

Info

Publication number
NO20000227L
NO20000227L NO20000227A NO20000227A NO20000227L NO 20000227 L NO20000227 L NO 20000227L NO 20000227 A NO20000227 A NO 20000227A NO 20000227 A NO20000227 A NO 20000227A NO 20000227 L NO20000227 L NO 20000227L
Authority
NO
Norway
Prior art keywords
phenyl
preparation
crystal modification
pyrimidinamine derivative
pyrimidinamine
Prior art date
Application number
NO20000227A
Other languages
English (en)
Other versions
NO20000227D0 (no
NO319486B1 (no
Inventor
Juerg Zimmermann
Bertrand Sutter
Hans Michael Buerger
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4218028&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20000227(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20000227D0 publication Critical patent/NO20000227D0/no
Publication of NO20000227L publication Critical patent/NO20000227L/no
Publication of NO319486B1 publication Critical patent/NO319486B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C30—CRYSTAL GROWTH
    • C30B—SINGLE-CRYSTAL GROWTH; UNIDIRECTIONAL SOLIDIFICATION OF EUTECTIC MATERIAL OR UNIDIRECTIONAL DEMIXING OF EUTECTOID MATERIAL; REFINING BY ZONE-MELTING OF MATERIAL; PRODUCTION OF A HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; SINGLE CRYSTALS OR HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; AFTER-TREATMENT OF SINGLE CRYSTALS OR A HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; APPARATUS THEREFOR
    • C30B7/00—Single-crystal growth from solutions using solvents which are liquid at normal temperature, e.g. aqueous solutions

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Materials Engineering (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Metallurgy (AREA)
  • Dermatology (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
NO20000227A 1997-07-18 2000-01-17 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat, farmasøytisk sammensetning innbefattende samme, fremgangsmåte for fremstilling av samme og anvendelse av samme for fremstilling av preparat NO319486B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH176497 1997-07-18
PCT/EP1998/004427 WO1999003854A1 (en) 1997-07-18 1998-07-16 Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use

Publications (3)

Publication Number Publication Date
NO20000227D0 NO20000227D0 (no) 2000-01-17
NO20000227L true NO20000227L (no) 2000-01-17
NO319486B1 NO319486B1 (no) 2005-08-22

Family

ID=4218028

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20000227A NO319486B1 (no) 1997-07-18 2000-01-17 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat, farmasøytisk sammensetning innbefattende samme, fremgangsmåte for fremstilling av samme og anvendelse av samme for fremstilling av preparat
NO20052755A NO331016B1 (no) 1997-07-18 2005-06-07 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20052755A NO331016B1 (no) 1997-07-18 2005-06-07 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat

Country Status (30)

Country Link
US (5) US6894051B1 (no)
EP (1) EP0998473B1 (no)
JP (1) JP3276359B2 (no)
KR (1) KR100450356B1 (no)
CN (1) CN1134430C (no)
AR (2) AR016351A1 (no)
AT (1) ATE251152T1 (no)
AU (1) AU740713B2 (no)
BR (1) BR9810920A (no)
CA (1) CA2296604C (no)
CO (1) CO4940418A1 (no)
CZ (1) CZ298531B6 (no)
DE (1) DE69818674T2 (no)
DK (1) DK0998473T3 (no)
ES (1) ES2209194T3 (no)
HU (1) HU230185B1 (no)
ID (1) ID24093A (no)
IL (5) IL133906A0 (no)
MY (2) MY128664A (no)
NO (2) NO319486B1 (no)
NZ (1) NZ502295A (no)
PE (1) PE97899A1 (no)
PL (1) PL188348B1 (no)
PT (1) PT998473E (no)
RU (1) RU2208012C2 (no)
SK (2) SK286551B6 (no)
TR (1) TR200000060T2 (no)
TW (1) TW491845B (no)
WO (1) WO1999003854A1 (no)
ZA (1) ZA986362B (no)

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