[go: up one dir, main page]

NO143459C - ANALOGUE PROCEDURE FOR PREPARING PHYSIOLOGICALLY ACTIVE 2-PHENYLIMINO-IMIDAZOLIDINE DERIVATIVES - Google Patents

ANALOGUE PROCEDURE FOR PREPARING PHYSIOLOGICALLY ACTIVE 2-PHENYLIMINO-IMIDAZOLIDINE DERIVATIVES

Info

Publication number
NO143459C
NO143459C NO753314A NO753314A NO143459C NO 143459 C NO143459 C NO 143459C NO 753314 A NO753314 A NO 753314A NO 753314 A NO753314 A NO 753314A NO 143459 C NO143459 C NO 143459C
Authority
NO
Norway
Prior art keywords
phenylimino
physiologically active
imidazolidine derivatives
analogue procedure
preparing physiologically
Prior art date
Application number
NO753314A
Other languages
Norwegian (no)
Other versions
NO753314L (en
NO143459B (en
Inventor
Helmut Staehle
Herbert Koeppe
Werner Kummer
Wolfgang Hoefke
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of NO753314L publication Critical patent/NO753314L/no
Publication of NO143459B publication Critical patent/NO143459B/en
Publication of NO143459C publication Critical patent/NO143459C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
    • C07D233/50Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO753314A 1974-10-01 1975-09-30 ANALOGUE PROCEDURE FOR PREPARING PHYSIOLOGICALLY ACTIVE 2-PHENYLIMINO-IMIDAZOLIDINE DERIVATIVES NO143459C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2446758A DE2446758C3 (en) 1974-10-01 1974-10-01 2- (2-Fluoro-6-trifluoromethylphenylimino) -imidazolidine, its acid addition salts, processes for the preparation of these compounds and their use in combating hypertension

Publications (3)

Publication Number Publication Date
NO753314L NO753314L (en) 1976-04-02
NO143459B NO143459B (en) 1980-11-10
NO143459C true NO143459C (en) 1981-02-18

Family

ID=5927202

Family Applications (1)

Application Number Title Priority Date Filing Date
NO753314A NO143459C (en) 1974-10-01 1975-09-30 ANALOGUE PROCEDURE FOR PREPARING PHYSIOLOGICALLY ACTIVE 2-PHENYLIMINO-IMIDAZOLIDINE DERIVATIVES

Country Status (27)

Country Link
JP (1) JPS6018653B2 (en)
AT (1) AT344159B (en)
BE (1) BE834051A (en)
BG (2) BG25221A3 (en)
CA (1) CA1056836A (en)
CH (5) CH620682A5 (en)
CS (1) CS193524B2 (en)
DD (1) DD123602A5 (en)
DE (1) DE2446758C3 (en)
DK (1) DK441875A (en)
ES (4) ES441385A1 (en)
FI (1) FI61883C (en)
FR (1) FR2286649A1 (en)
GB (1) GB1515019A (en)
HU (1) HU178469B (en)
IE (1) IE42130B1 (en)
IL (1) IL48214A (en)
LU (1) LU73472A1 (en)
NL (1) NL7511490A (en)
NO (1) NO143459C (en)
NZ (1) NZ178810A (en)
PH (1) PH13653A (en)
PL (2) PL98984B1 (en)
SE (1) SE418497B (en)
SU (1) SU575026A3 (en)
YU (1) YU230281A (en)
ZA (1) ZA756185B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2630060C2 (en) * 1976-07-03 1984-04-19 C.H. Boehringer Sohn, 6507 Ingelheim 2- (2-Bromo-6-fluoro-phenylimino) -imidazolidine, its acid addition salts, medicaments containing them and processes for their preparation
DE2806775A1 (en) * 1978-02-17 1979-08-30 Boehringer Sohn Ingelheim NEW SUBSTITUTED 2-PHENYLIMINO IMIDAZOLIDINE THEIR ACID ADDITION SALTS, MEDICINAL PRODUCTS CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF
DE2806811A1 (en) * 1978-02-17 1979-08-23 Boehringer Sohn Ingelheim NEW SUBSTITUTED 2-PHENYLIMINO-IMIDAZOLIDINE, THEIR ACID-ADDITIONAL SALTS, THESE MEDICINAL PRODUCTS AND METHOD FOR MANUFACTURING THE SAME
ZA801680B (en) * 1979-04-03 1981-03-25 Fujisawa Pharmaceutical Co 2-imidazoline derivatives,process for the preparation thereof and the pharmaceutical composition of the same
HU192986B (en) * 1984-05-23 1987-08-28 Egyt Gyogyszervegyeszeti Gyar Process for production of imidasodiline derivatives
CA2637292A1 (en) * 2006-01-27 2007-08-16 F. Hoffmann-La Roche Ag Use of 2-imidazoles for the treatment of cns disorders
KR101174191B1 (en) 2007-02-02 2012-08-14 에프. 호프만-라 로슈 아게 Novel 2-aminooxazolines as taar1 ligands for cns disorders
EP2121641B1 (en) 2007-02-15 2014-09-24 F. Hoffmann-La Roche AG 2-aminooxazolines as taar1 ligands
US8242153B2 (en) 2008-07-24 2012-08-14 Hoffmann-La Roche Inc. 4,5-dihydro-oxazol-2YL derivatives
US8354441B2 (en) 2009-11-11 2013-01-15 Hoffmann-La Roche Inc. Oxazoline derivatives
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
BR112018015389B1 (en) 2016-03-17 2023-12-19 F. Hoffmann-La Roche Ag 5-Ethyl-4-methyl-pyrazol-3-carboxamide derivative, its manufacturing process, oral pharmaceutical preparation and use

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3236857A (en) * 1961-10-09 1966-02-22 Boehringer Sohn Ingelheim 2-(phenyl-amino)-1, 3-diazacyclopentene-(2) substitution products
DE1670807A1 (en) * 1967-02-17 1971-03-11 Bayer Ag Process for the preparation of cyclic guanidines
DE1670918A1 (en) * 1967-09-07 1971-04-08 Bayer Ag Process for the preparation of 2-aryl-amino-substituted nitrogen-containing heterocycles
BE787683A (en) * 1971-08-20 1973-02-19 Boehringer Sohn Ingelheim 2-PHENYLIMINO-IMIDAZOLIDINES, THEIR ADDITIONAL SALTS WITH ACIDS AND METHODS FOR MAKING THEM

Also Published As

Publication number Publication date
CH626352A5 (en) 1981-11-13
CA1056836A (en) 1979-06-19
IL48214A0 (en) 1975-11-25
PL98984B1 (en) 1978-06-30
NO753314L (en) 1976-04-02
DE2446758A1 (en) 1976-04-22
CH627453A5 (en) 1982-01-15
ES444900A1 (en) 1977-04-16
LU73472A1 (en) 1977-05-16
AT344159B (en) 1978-07-10
JPS5159863A (en) 1976-05-25
FI61883C (en) 1982-10-11
NZ178810A (en) 1978-04-03
IE42130B1 (en) 1980-06-04
ATA722875A (en) 1977-11-15
DK441875A (en) 1976-04-02
SU575026A3 (en) 1977-09-30
JPS6018653B2 (en) 1985-05-11
CH627452A5 (en) 1982-01-15
ES441385A1 (en) 1977-08-01
NL7511490A (en) 1976-04-05
DE2446758B2 (en) 1978-05-18
ZA756185B (en) 1977-06-29
SE418497B (en) 1981-06-09
FR2286649A1 (en) 1976-04-30
NO143459B (en) 1980-11-10
IE42130L (en) 1976-04-01
FI61883B (en) 1982-06-30
FI752728A7 (en) 1976-04-02
HU178469B (en) 1982-05-28
AU8529875A (en) 1977-04-07
DD123602A5 (en) 1977-01-05
DE2446758C3 (en) 1979-01-04
FR2286649B1 (en) 1979-09-14
BE834051A (en) 1976-03-30
ES444901A1 (en) 1977-04-16
PH13653A (en) 1980-08-21
GB1515019A (en) 1978-06-21
CH627454A5 (en) 1982-01-15
CS193524B2 (en) 1979-10-31
BG25221A3 (en) 1978-08-10
YU230281A (en) 1982-02-28
PL97003B1 (en) 1978-01-31
ES444898A1 (en) 1977-05-16
CH620682A5 (en) 1980-12-15
BG25220A3 (en) 1978-08-10
IL48214A (en) 1979-10-31
SE7511028L (en) 1976-04-02

Similar Documents

Publication Publication Date Title
SE420199B (en) PROCEDURE FOR PREPARING 16-OXIDATED PROSTANIC ACID DERIVATIVES
NO145382C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 3-AMINO-INDAZOLCARBOXYLIC ACID DERIVATIVES.
NO149035C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE ACYLANILIDE DERIVATIVES
SE428562C (en) PROCEDURE FOR PURINATE DERIVATIVES
SE431652B (en) PROCEDURE FOR PREPARING 7BETA-AMINO-3CEFEM-3OL-4-CARBOXYLIC ACID DERIVATIVES
NO141013C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE BIFENYLYL DERIVATIVES
NO147986C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE PHENYLETYLAMINES
NO146865C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 16-DEHYDRO ANDROSTAND DERIVATIVES
NO143459C (en) ANALOGUE PROCEDURE FOR PREPARING PHYSIOLOGICALLY ACTIVE 2-PHENYLIMINO-IMIDAZOLIDINE DERIVATIVES
SE412066B (en) PROCEDURE FOR PREPARING PHAMACOLOGICALLY EFFECTIVE TIENODIAZINE DERIVATIVES
SE409452B (en) PROCEDURE FOR THE PREPARATION OF STILBENDER DERIVATIVES
SE7506237L (en) PROCEDURE FOR THE PREPARATION OF DEKAHYDROISOKINOLINE DERIVATIVES
NO147672C (en) ANALOGUE PROCEDURE FOR PREPARING N-ARYL-N- (1-L1-4-PIPERIDINYL) -ARYLACETAMIDES
NO144928C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE ZANTINE DERIVATIVES.
SE418292B (en) PROCEDURE FOR PREPARING 5-ARYL-2-FURAMIDINES
SE421612B (en) PROCEDURE FOR PREPARING ALFA-6-DEOXI-5-HYDROXYTETRACYCLINE
SE425739B (en) PROCEDURE FOR PREPARING CERTAIN STATED TETRAZOLYL-BENZOPYRANOPYRIDINE DERIVATIVES
NO145383C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE SUBSTITUTED INDOLS.
SE417509B (en) PROCEDURE FOR PREPARING ANTHELMINTICALLY ACTIVE 2-CARBAL COXYAMINO-5 (6) -PHENYL-SULPHONYLOXY-BENZIMIDAZOLES
NO143317C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE TIAZINE Dioxides
SE414926B (en) PROCEDURE FOR PREPARING 1-ALKYL-2- (PHENOXIMETHYL) -5-NITROIMIDAZOLES
SE414029B (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE FENTIAZINE DERIVATIVES
NO143499C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE INHANDER DERIVATIVES
SE7513739L (en) PROCEDURE FOR THE PREPARATION OF 2-SCYL-4-OXO-PYRAZINO-ISOCONOLINE DERIVATIVES
NO142525C (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF PHYSIOLOGICALLY ACTIVE ISOTIOR INGREDIENTS