NL7511490A - PROCESS FOR THE PREPARATION OF NEW 2,6-DIGITAL SUBSTITUTED 2-PHENYLIMINOIMIDAZOLIDINS AND THEIR ACID ADDITIONAL SALTS. - Google Patents
PROCESS FOR THE PREPARATION OF NEW 2,6-DIGITAL SUBSTITUTED 2-PHENYLIMINOIMIDAZOLIDINS AND THEIR ACID ADDITIONAL SALTS.Info
- Publication number
- NL7511490A NL7511490A NL7511490A NL7511490A NL7511490A NL 7511490 A NL7511490 A NL 7511490A NL 7511490 A NL7511490 A NL 7511490A NL 7511490 A NL7511490 A NL 7511490A NL 7511490 A NL7511490 A NL 7511490A
- Authority
- NL
- Netherlands
- Prior art keywords
- phenyliminoimidazolidins
- substituted
- digital
- preparation
- new
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2446758A DE2446758C3 (en) | 1974-10-01 | 1974-10-01 | 2- (2-Fluoro-6-trifluoromethylphenylimino) -imidazolidine, its acid addition salts, processes for the preparation of these compounds and their use in combating hypertension |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NL7511490A true NL7511490A (en) | 1976-04-05 |
Family
ID=5927202
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL7511490A NL7511490A (en) | 1974-10-01 | 1975-09-30 | PROCESS FOR THE PREPARATION OF NEW 2,6-DIGITAL SUBSTITUTED 2-PHENYLIMINOIMIDAZOLIDINS AND THEIR ACID ADDITIONAL SALTS. |
Country Status (27)
| Country | Link |
|---|---|
| JP (1) | JPS6018653B2 (en) |
| AT (1) | AT344159B (en) |
| BE (1) | BE834051A (en) |
| BG (2) | BG25221A3 (en) |
| CA (1) | CA1056836A (en) |
| CH (5) | CH620682A5 (en) |
| CS (1) | CS193524B2 (en) |
| DD (1) | DD123602A5 (en) |
| DE (1) | DE2446758C3 (en) |
| DK (1) | DK441875A (en) |
| ES (4) | ES441385A1 (en) |
| FI (1) | FI61883C (en) |
| FR (1) | FR2286649A1 (en) |
| GB (1) | GB1515019A (en) |
| HU (1) | HU178469B (en) |
| IE (1) | IE42130B1 (en) |
| IL (1) | IL48214A (en) |
| LU (1) | LU73472A1 (en) |
| NL (1) | NL7511490A (en) |
| NO (1) | NO143459C (en) |
| NZ (1) | NZ178810A (en) |
| PH (1) | PH13653A (en) |
| PL (2) | PL98984B1 (en) |
| SE (1) | SE418497B (en) |
| SU (1) | SU575026A3 (en) |
| YU (1) | YU230281A (en) |
| ZA (1) | ZA756185B (en) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2630060C2 (en) * | 1976-07-03 | 1984-04-19 | C.H. Boehringer Sohn, 6507 Ingelheim | 2- (2-Bromo-6-fluoro-phenylimino) -imidazolidine, its acid addition salts, medicaments containing them and processes for their preparation |
| DE2806775A1 (en) * | 1978-02-17 | 1979-08-30 | Boehringer Sohn Ingelheim | NEW SUBSTITUTED 2-PHENYLIMINO IMIDAZOLIDINE THEIR ACID ADDITION SALTS, MEDICINAL PRODUCTS CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF |
| DE2806811A1 (en) * | 1978-02-17 | 1979-08-23 | Boehringer Sohn Ingelheim | NEW SUBSTITUTED 2-PHENYLIMINO-IMIDAZOLIDINE, THEIR ACID-ADDITIONAL SALTS, THESE MEDICINAL PRODUCTS AND METHOD FOR MANUFACTURING THE SAME |
| ZA801680B (en) * | 1979-04-03 | 1981-03-25 | Fujisawa Pharmaceutical Co | 2-imidazoline derivatives,process for the preparation thereof and the pharmaceutical composition of the same |
| HU192986B (en) | 1984-05-23 | 1987-08-28 | Egyt Gyogyszervegyeszeti Gyar | Process for production of imidasodiline derivatives |
| JP2009524619A (en) * | 2006-01-27 | 2009-07-02 | エフ.ホフマン−ラ ロシュ アーゲー | Use of 2-imidazole for the treatment of CNS disorders |
| JP5248528B2 (en) | 2007-02-02 | 2013-07-31 | エフ.ホフマン−ラ ロシュ アーゲー | Novel 2-aminooxazolines as TAAR1 ligands for CNS diseases |
| MX2009008465A (en) | 2007-02-15 | 2009-08-20 | Hoffmann La Roche | 2-aminooxazolines as taar1 ligands. |
| US8242153B2 (en) | 2008-07-24 | 2012-08-14 | Hoffmann-La Roche Inc. | 4,5-dihydro-oxazol-2YL derivatives |
| US8354441B2 (en) | 2009-11-11 | 2013-01-15 | Hoffmann-La Roche Inc. | Oxazoline derivatives |
| US9452980B2 (en) | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
| PE20181446A1 (en) | 2016-03-17 | 2018-09-12 | Hoffmann La Roche | DERIVATIVES OF 5-ETHYL-4-METHYL-PIRAZOL-3-CARBOXAMIDE WITH ACTIVITY AS OF TAAR |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3236857A (en) * | 1961-10-09 | 1966-02-22 | Boehringer Sohn Ingelheim | 2-(phenyl-amino)-1, 3-diazacyclopentene-(2) substitution products |
| DE1670807A1 (en) * | 1967-02-17 | 1971-03-11 | Bayer Ag | Process for the preparation of cyclic guanidines |
| DE1670918A1 (en) * | 1967-09-07 | 1971-04-08 | Bayer Ag | Process for the preparation of 2-aryl-amino-substituted nitrogen-containing heterocycles |
| BE787683A (en) * | 1971-08-20 | 1973-02-19 | Boehringer Sohn Ingelheim | 2-PHENYLIMINO-IMIDAZOLIDINES, THEIR ADDITIONAL SALTS WITH ACIDS AND METHODS FOR MAKING THEM |
-
1974
- 1974-10-01 DE DE2446758A patent/DE2446758C3/en not_active Expired
-
1975
- 1975-09-22 AT AT722875A patent/AT344159B/en not_active IP Right Cessation
- 1975-09-23 SU SU7502174605A patent/SU575026A3/en active
- 1975-09-26 PH PH17613A patent/PH13653A/en unknown
- 1975-09-29 BG BG032014A patent/BG25221A3/en unknown
- 1975-09-29 CS CS756573A patent/CS193524B2/en unknown
- 1975-09-29 LU LU73472A patent/LU73472A1/xx unknown
- 1975-09-29 BG BG031110A patent/BG25220A3/en unknown
- 1975-09-29 DD DD188613A patent/DD123602A5/xx unknown
- 1975-09-30 IL IL48214A patent/IL48214A/en unknown
- 1975-09-30 DK DK441875A patent/DK441875A/en not_active Application Discontinuation
- 1975-09-30 JP JP50118196A patent/JPS6018653B2/en not_active Expired
- 1975-09-30 NO NO753314A patent/NO143459C/en unknown
- 1975-09-30 PL PL1975197816A patent/PL98984B1/en unknown
- 1975-09-30 HU HU75BO1573A patent/HU178469B/en unknown
- 1975-09-30 CH CH1267875A patent/CH620682A5/en not_active IP Right Cessation
- 1975-09-30 CA CA236,670A patent/CA1056836A/en not_active Expired
- 1975-09-30 FI FI752728A patent/FI61883C/en not_active IP Right Cessation
- 1975-09-30 NZ NZ178810A patent/NZ178810A/en unknown
- 1975-09-30 PL PL1975183670A patent/PL97003B1/en unknown
- 1975-09-30 ZA ZA756185A patent/ZA756185B/en unknown
- 1975-09-30 ES ES441385A patent/ES441385A1/en not_active Expired
- 1975-09-30 NL NL7511490A patent/NL7511490A/en not_active Application Discontinuation
- 1975-09-30 GB GB40012/75A patent/GB1515019A/en not_active Expired
- 1975-09-30 BE BE160578A patent/BE834051A/en not_active IP Right Cessation
- 1975-10-01 SE SE7511028A patent/SE418497B/en not_active IP Right Cessation
- 1975-10-01 FR FR7530117A patent/FR2286649A1/en active Granted
- 1975-10-01 IE IE2150/75A patent/IE42130B1/en unknown
-
1976
- 1976-02-04 ES ES444898A patent/ES444898A1/en not_active Expired
- 1976-02-04 ES ES444900A patent/ES444900A1/en not_active Expired
- 1976-02-04 ES ES444901A patent/ES444901A1/en not_active Expired
-
1980
- 1980-07-01 CH CH506380A patent/CH627453A5/en not_active IP Right Cessation
- 1980-07-01 CH CH506280A patent/CH627452A5/en not_active IP Right Cessation
- 1980-07-01 CH CH506480A patent/CH626352A5/en not_active IP Right Cessation
- 1980-07-01 CH CH506580A patent/CH627454A5/en not_active IP Right Cessation
-
1981
- 1981-09-24 YU YU02302/81A patent/YU230281A/en unknown
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BA | A request for search or an international-type search has been filed | ||
| BB | A search report has been drawn up | ||
| BC | A request for examination has been filed | ||
| A85 | Still pending on 85-01-01 | ||
| BV | The patent application has lapsed |