[go: up one dir, main page]

MX2018015275A - Compuestos de tetrahidropiranilcarbonil-2,3-dihidro-1h-indol para tratar cancer. - Google Patents

Compuestos de tetrahidropiranilcarbonil-2,3-dihidro-1h-indol para tratar cancer.

Info

Publication number
MX2018015275A
MX2018015275A MX2018015275A MX2018015275A MX2018015275A MX 2018015275 A MX2018015275 A MX 2018015275A MX 2018015275 A MX2018015275 A MX 2018015275A MX 2018015275 A MX2018015275 A MX 2018015275A MX 2018015275 A MX2018015275 A MX 2018015275A
Authority
MX
Mexico
Prior art keywords
cancer
compounds
dihydro
tetrahydropyranylcarbonyl
indole compounds
Prior art date
Application number
MX2018015275A
Other languages
English (en)
Other versions
MX382877B (es
Inventor
Robert Henry James
Rubio Almudena
Anne Bastian Jolie
Chen Jiehao
Daniel Cohen Jeffrey
Thomas Mcmillen William
Earl Reaman Bradley
Jon Sall Daniel
Zhao Gaiying
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MX2018015275A publication Critical patent/MX2018015275A/es
Publication of MX382877B publication Critical patent/MX382877B/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/10Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/4045Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/57Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/01Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invención se refiere a ciertos nuevos compuestos de 2,3-dihidro-1H-indol, composiciones farmacéuticas que comprenden los compuestos, y métodos para usar los compuestos para tratar cáncer, más particularmente para el tratamiento de cáncer seleccionado a partir del grupo que consiste de melanoma, leucemia mieloide aguda, leucemia linfocítica crónica, cáncer colorrectal, cáncer de mama, cáncer de pulmón, cáncer de ovario, carcinoma de tubos de falopio, carcinoma peritoneal primario, cáncer cervical, cáncer gástrico, cáncer hepático, cáncer pancreático, cáncer tiroideo, glioma, linfoma no Hodgkin, y linfoma de Hodgkin.
MX2018015275A 2016-06-10 2017-05-31 Compuestos de tetrahidropiranilcarbonil-2,3-dihidro-1h-indol para tratar cancer. MX382877B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662348457P 2016-06-10 2016-06-10
PCT/US2017/035097 WO2017213919A1 (en) 2016-06-10 2017-05-31 1-tetrahydropyranylcarbonyl-2,3-dihydro-1h-indole compounds for treating cancer

Publications (2)

Publication Number Publication Date
MX2018015275A true MX2018015275A (es) 2019-04-11
MX382877B MX382877B (es) 2025-03-13

Family

ID=59031409

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018015275A MX382877B (es) 2016-06-10 2017-05-31 Compuestos de tetrahidropiranilcarbonil-2,3-dihidro-1h-indol para tratar cancer.

Country Status (40)

Country Link
US (2) US10759786B2 (es)
EP (1) EP3468965B1 (es)
JP (1) JP6632746B2 (es)
KR (1) KR102241258B1 (es)
CN (1) CN109641881B (es)
AR (1) AR108586A1 (es)
AU (1) AU2017277833B2 (es)
BR (1) BR112018072872A2 (es)
CA (1) CA3027035C (es)
CL (1) CL2018003543A1 (es)
CO (1) CO2018013251A2 (es)
CR (1) CR20180579A (es)
CY (1) CY1123660T1 (es)
DK (1) DK3468965T3 (es)
DO (1) DOP2018000278A (es)
EA (1) EA037419B1 (es)
EC (1) ECSP19001734A (es)
ES (1) ES2797981T3 (es)
HR (1) HRP20200769T1 (es)
HU (1) HUE050155T2 (es)
IL (1) IL263497B (es)
JO (1) JOP20170131B1 (es)
LT (1) LT3468965T (es)
MA (1) MA45224B1 (es)
MD (1) MD3468965T2 (es)
ME (1) ME03744B (es)
MX (1) MX382877B (es)
MY (1) MY197462A (es)
NZ (1) NZ748500A (es)
PE (1) PE20190378A1 (es)
PH (1) PH12018502572A1 (es)
PL (1) PL3468965T3 (es)
PT (1) PT3468965T (es)
RS (1) RS60322B1 (es)
SG (1) SG11201809625RA (es)
SI (1) SI3468965T1 (es)
TW (1) TWI671294B (es)
UA (1) UA122526C2 (es)
WO (1) WO2017213919A1 (es)
ZA (1) ZA201807688B (es)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10738035B2 (en) 2015-05-13 2020-08-11 Enanta Pharmaceuticals, Inc. Hepatitis B antiviral agents
SG11201807543YA (en) 2016-03-07 2018-09-27 Enanta Pharm Inc Hepatitis b antiviral agents
AU2018326474B2 (en) 2017-08-28 2024-07-25 Enanta Pharmaceuticals, Inc. Hepatitis B antiviral agents
US12275729B2 (en) * 2017-11-01 2025-04-15 Merck Sharp & Dohme Llc Substituted tetrahydroquinolin compounds as indoleamine 2,3-dioxygenase (IDO) inhibitors
WO2019126257A1 (en) * 2017-12-21 2019-06-27 Merck Patent Gmbh Combination of an anti-pd-l1 antibody and ido1 inhibitor for the treatment of cancer
US11058678B2 (en) 2018-01-22 2021-07-13 Enanta Pharmaceuticals, Inc. Substituted heterocycles as antiviral agents
WO2020036837A1 (en) 2018-08-17 2020-02-20 Merck Sharp & Dohme Corp. Novel substituted tetrahydroquinoline compounds as indoleamine 2,3-dioxygenase inhibitors
CN112955142A (zh) 2018-09-21 2021-06-11 英安塔制药有限公司 官能化杂环化合物作为抗病毒剂
WO2020096871A1 (en) * 2018-11-06 2020-05-14 Merck Sharp & Dohme Corp. Novel substituted tricyclic compounds as indoleamine 2,3-dioxygenase inhibitors
CN113271946A (zh) 2018-11-21 2021-08-17 英安塔制药有限公司 官能化杂环化合物作为抗病毒剂
WO2020247444A1 (en) 2019-06-03 2020-12-10 Enanta Pharmaceuticals, Inc, Hepatitis b antiviral agents
US11760755B2 (en) 2019-06-04 2023-09-19 Enanta Pharmaceuticals, Inc. Hepatitis B antiviral agents
US11472808B2 (en) 2019-06-04 2022-10-18 Enanta Pharmaceuticals, Inc. Substituted pyrrolo[1,2-c]pyrimidines as hepatitis B antiviral agents
WO2021007488A1 (en) 2019-07-11 2021-01-14 Enanta Pharmaceuticals, Inc. Substituted heterocycles as antiviral agents
WO2021055425A2 (en) 2019-09-17 2021-03-25 Enanta Pharmaceuticals, Inc. Functionalized heterocycles as antiviral agents
WO2021188414A1 (en) 2020-03-16 2021-09-23 Enanta Pharmaceuticals, Inc. Functionalized heterocyclic compounds as antiviral agents
CN114105961B (zh) * 2021-12-10 2023-09-12 海南梵圣生物科技有限公司 一种ido1抑制剂(ly-3381916)制备方法
CN114213310B (zh) * 2021-12-31 2024-02-23 中国药科大学 吲哚啉化合物及其衍生物、制备方法、药物组合物和应用
WO2025072355A1 (en) * 2023-09-25 2025-04-03 Biohybrid Solutions Holdings, Inc. Methods for and compositions of non-peg bioconjugates with ultra-high drug-to-agent ratio
WO2025140363A1 (zh) * 2023-12-27 2025-07-03 海思科医药集团股份有限公司 一种苯基哌啶衍生物的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE602004027171D1 (de) * 2003-04-11 2010-06-24 High Point Pharmaceuticals Llc Verbindungen mit Aktivität an der 11Beta-Hydroxasteroiddehydrogenase
BR122020016659B8 (pt) * 2005-05-10 2021-07-27 Incyte Holdings Corp moduladores de 2,3-dioxigenase de indolamina e métodos de modulação de atividade de inibição e de imunossupressão
US7622495B2 (en) * 2006-10-03 2009-11-24 Neurim Pharmaceuticals (1991) Ltd. Substituted aryl-indole compounds and their kynurenine/kynuramine-like metabolites as therapeutic agents
CN101990537A (zh) * 2008-02-07 2011-03-23 雅培制药有限公司 作为阳性别构调节剂的酰胺衍生物和其使用方法
RS57132B1 (sr) * 2008-07-08 2018-07-31 Incyte Holdings Corp 1,2,5-oksadiazoli kao inhibitori indolamin 2,3-dioksigenaze
NO2694640T3 (es) * 2011-04-15 2018-03-17
KR20150129010A (ko) * 2013-03-15 2015-11-18 브리스톨-마이어스 스큅 컴퍼니 Ido 억제제
WO2015150097A1 (en) * 2014-04-04 2015-10-08 Iomet Pharma Ltd Indole derivatives for use in medicine
AR102537A1 (es) * 2014-11-05 2017-03-08 Flexus Biosciences Inc Agentes inmunomoduladores
CA3048193A1 (en) * 2015-12-23 2017-06-29 Moonshot Pharma Llc Methods for inducing an immune response by promoting premature termination codon read-through

Also Published As

Publication number Publication date
EP3468965B1 (en) 2020-04-29
AR108586A1 (es) 2018-09-05
MD3468965T2 (ro) 2020-08-31
MA45224B1 (fr) 2020-06-30
KR20190003750A (ko) 2019-01-09
SI3468965T1 (sl) 2020-07-31
EA037419B1 (ru) 2021-03-25
IL263497A (en) 2019-01-31
JP2019518027A (ja) 2019-06-27
PL3468965T3 (pl) 2020-09-21
CR20180579A (es) 2019-02-08
CA3027035A1 (en) 2017-12-14
KR102241258B1 (ko) 2021-04-16
US20190161477A1 (en) 2019-05-30
NZ748500A (en) 2020-04-24
WO2017213919A1 (en) 2017-12-14
ZA201807688B (en) 2020-08-26
TW201806948A (zh) 2018-03-01
AU2017277833B2 (en) 2020-07-02
SG11201809625RA (en) 2018-11-29
IL263497B (en) 2020-11-30
CN109641881B (zh) 2022-01-07
UA122526C2 (uk) 2020-11-25
CA3027035C (en) 2021-05-04
LT3468965T (lt) 2020-06-10
DOP2018000278A (es) 2018-12-31
CO2018013251A2 (es) 2019-01-18
PH12018502572A1 (en) 2019-10-28
ME03744B (me) 2021-04-20
EA201892479A1 (ru) 2019-07-31
DK3468965T3 (da) 2020-06-15
US9872853B2 (en) 2018-01-23
US20170354641A1 (en) 2017-12-14
US10759786B2 (en) 2020-09-01
RS60322B1 (sr) 2020-07-31
JP6632746B2 (ja) 2020-01-22
PE20190378A1 (es) 2019-03-08
EP3468965A1 (en) 2019-04-17
BR112018072872A2 (pt) 2019-03-06
MY197462A (en) 2023-06-19
CY1123660T1 (el) 2022-03-24
ECSP19001734A (es) 2019-01-31
ES2797981T3 (es) 2020-12-04
CN109641881A (zh) 2019-04-16
CL2018003543A1 (es) 2019-03-22
JOP20170131B1 (ar) 2021-08-17
MX382877B (es) 2025-03-13
TWI671294B (zh) 2019-09-11
AU2017277833A1 (en) 2018-11-15
HRP20200769T1 (hr) 2020-07-24
PT3468965T (pt) 2020-07-16
HUE050155T2 (hu) 2020-12-28

Similar Documents

Publication Publication Date Title
CO2018013251A2 (es) Compuestos derivados de 1-tetrahidropiranilcarbonil-2,3-dihidro-1h-indol para tratar el cancer
UY36419A (es) Composiciones farmacéuticas que contienen anticuerpos anti-cd38 para el tratamiento de la leucemia mieloide aguda
CL2017002637A1 (es) Compuestos nucleósidos 5'-sustituidos.
MX375746B (es) Combinación de lenalidomida y constructo de polipéptido, y sus usos.
CR20170596A (es) Derivados de amidas policiclicas como inhibidores de cdk9
CL2016002157A1 (es) Anticuerpos anti-cd38 para el tratamiento de leucemia linfoide aguda
MD3395820T2 (ro) Compuși antitumorali
KR102247795B9 (ko) 급성 골수성 백혈병 또는 전이성 유방암의 예방 또는 치료용 약제학적 조성물
EP3925969C0 (en) Peptide compounds and peptide conjugates for the treatment of cancer by receptor-mediated chemotherapy
CL2017001336A1 (es) Nuevos aminoácidos ester fosforamidatos 2' y/o 5', 3' deoxiadenosina derivativos como compuestos anticancerígenos
PH12017501879A1 (en) Methods for treating cancer
GB201709405D0 (en) Compounds for treating ovarian cancer
MX387515B (es) Inhibidores de factor xia.
EA201691549A1 (ru) Ариллактамные ингибиторы киназы
MX381092B (es) Inhibidores de fucosidasa.
KR102004959B9 (ko) 전이성 난소암, 자궁내막암 또는 유방암의 예방 또는 치료용 조성물
MX2017009445A (es) Inhibidores del factor xia.
MX388409B (es) Composiciones y metodos para tratar canceres.
MX2019003311A (es) Metodos para tratamiento de cancer de ovario.
UA111303C2 (uk) Пігмент зеленого світіння для плівкового маскуючого матеріалу
UA104379U (uk) Біс(оксифеніленімінометилен)дифеноли з перфторованими моно- та біфеніленовими центральними фрагментами як прекурсори для синтезу бензоксазинів
MY198135A (en) Combination of therapeutic agents for treating ovarian cancer