[go: up one dir, main page]

MX2018015067A - Solucion inyectable a ph 7 que comprende por lo menos una insulina basal cuyo pi esta comprendido entre 5.8 y 8.5, una insulina prandial y/o una hormona gastrointestinal y un co-poliamino acido que porta cargas de carboxilatos y de radicales hidrofobicos. - Google Patents

Solucion inyectable a ph 7 que comprende por lo menos una insulina basal cuyo pi esta comprendido entre 5.8 y 8.5, una insulina prandial y/o una hormona gastrointestinal y un co-poliamino acido que porta cargas de carboxilatos y de radicales hidrofobicos.

Info

Publication number
MX2018015067A
MX2018015067A MX2018015067A MX2018015067A MX2018015067A MX 2018015067 A MX2018015067 A MX 2018015067A MX 2018015067 A MX2018015067 A MX 2018015067A MX 2018015067 A MX2018015067 A MX 2018015067A MX 2018015067 A MX2018015067 A MX 2018015067A
Authority
MX
Mexico
Prior art keywords
insulin
acid bearing
injectable solution
carboxylate charges
gastrointestinal hormone
Prior art date
Application number
MX2018015067A
Other languages
English (en)
Inventor
Soula Olivier
Geissler Alexandre
Charvet Richard
LAAGE Ségolène
Original Assignee
Adocia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adocia filed Critical Adocia
Publication of MX2018015067A publication Critical patent/MX2018015067A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/28Insulins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/26Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se relaciona con composiciones estables físicamente en la forma de una solución acuosa inyectable, cuyo pH es de 6.0 a 8.0, que comprende por lo menos: a) una insulina basal cuyo punto isoeléctrico (pI) es de 5.8 a 8.5, b) una hormona de insulina prandial o gastrointestinal y c) un co-poliamino ácido que porta cargas de carboxilato y por lo menos un radical hidrofóbico.
MX2018015067A 2016-06-07 2017-06-07 Solucion inyectable a ph 7 que comprende por lo menos una insulina basal cuyo pi esta comprendido entre 5.8 y 8.5, una insulina prandial y/o una hormona gastrointestinal y un co-poliamino acido que porta cargas de carboxilatos y de radicales hidrofobicos. MX2018015067A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR1655222A FR3052072A1 (fr) 2016-06-07 2016-06-07 Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes
PCT/EP2017/063886 WO2017211916A1 (fr) 2016-06-07 2017-06-07 Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5, une insuline prandiale et/ou une hormone gastrointestinale, et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes

Publications (1)

Publication Number Publication Date
MX2018015067A true MX2018015067A (es) 2019-05-09

Family

ID=57348773

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2018015068A MX2018015068A (es) 2016-06-07 2017-06-07 Solucion inyectable a ph 7 que comprende por lo menos una insulina basal cuyo pi esta comprendido entre 5.8 y 8.5 y co-poliamino acido que porta cargas de carboxilatos y radicales hidrofobicos.
MX2018015067A MX2018015067A (es) 2016-06-07 2017-06-07 Solucion inyectable a ph 7 que comprende por lo menos una insulina basal cuyo pi esta comprendido entre 5.8 y 8.5, una insulina prandial y/o una hormona gastrointestinal y un co-poliamino acido que porta cargas de carboxilatos y de radicales hidrofobicos.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2018015068A MX2018015068A (es) 2016-06-07 2017-06-07 Solucion inyectable a ph 7 que comprende por lo menos una insulina basal cuyo pi esta comprendido entre 5.8 y 8.5 y co-poliamino acido que porta cargas de carboxilatos y radicales hidrofobicos.

Country Status (12)

Country Link
US (2) US10383920B2 (es)
EP (2) EP3463292B1 (es)
JP (1) JP2019517555A (es)
CN (2) CN109640953B (es)
BR (2) BR112018075140A2 (es)
EA (2) EA039333B1 (es)
FR (1) FR3052072A1 (es)
MX (2) MX2018015068A (es)
PH (1) PH12018502558B1 (es)
SA (2) SA518400588B1 (es)
SG (2) SG11201810937WA (es)
WO (2) WO2017211916A1 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR3070264A1 (fr) * 2017-08-24 2019-03-01 Adocia Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris de 5,8 a 8,5 et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes
FR3083089A1 (fr) * 2018-06-29 2020-01-03 Adocia Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes
KR20200106891A (ko) 2017-12-07 2020-09-15 아도시아 pI가 5.8 내지 8.5인 적어도 1종의 기저 인슐린, 및 카복실산염 전하 및 소수성 라디칼을 보유하는 코-폴리아미노산을 포함하는 pH 7의 주사용 용액
FR3083086A1 (fr) * 2018-06-29 2020-01-03 Adocia Compositions sous forme d'une solution aqueuse injectable comprenant de l'amyline, un agoniste au recepteur de l'amyline ou un analogue d'amyline et un co-polyaminoacide
IL275148B2 (en) 2017-12-07 2025-02-01 Adocia An injectable solution with a pH of 7 comprising at least one basic insulin with a PI between 5.8 and 8.5 and a copolyamino acid bearing carboxylate charges and hydrophobic radicals.
WO2019110773A1 (fr) 2017-12-07 2019-06-13 Adocia Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes
IL275146B2 (en) 2017-12-07 2025-01-01 Adocia Preparations in the form of an aqueous solution for injection comprising amylin, an amylin receptor agonist or an amylin analog and a copolyamino acid
WO2019110797A1 (fr) * 2017-12-07 2019-06-13 Adocia Compositions sous forme d'une solution aqueuse injectable comprenant de l'amyline, un agoniste au recepteur de l'amyline ou un analogue d'amyline et un co-polyaminoacide
WO2019115411A1 (fr) * 2017-12-07 2019-06-20 Adocia Compositions sous forme d'une solution aqueuse injectable comprenant de l'amyline, un agoniste au recepteur de l'amyline ou un analogue d'amyline et un co-polyaminoacide
BR112020011479A2 (pt) 2017-12-07 2020-11-17 Adocia composições na forma de uma solução aquosa injetável caracterizada pelo fato de que compreende amilina, um agonista do receptor de amilina ou um análogo de amilina e um co-poliaminoácido
FR3067247A1 (fr) * 2018-06-07 2018-12-14 Adocia Compositions sous forme d'une solution aqueuse injectable comprenant du glucagon humain et un co-polyaminoacide
WO2019243628A1 (fr) * 2018-06-22 2019-12-26 Adocia Composition injectable a ph 7 comprenant un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes et au moins une insuline basale presentant au moins un effet prandial et un effet basal
FR3084586B1 (fr) * 2018-08-03 2020-11-06 Adocia Compositions sous forme d'une solution aqueuse injectable comprenant de l'amyline, un agoniste au recepteur de l'amyline ou un analogue d'amyline et un compose amphiphile porteur de radicaux hydrophobes
FR3084585B1 (fr) * 2018-08-03 2020-11-06 Adocia Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un compose amphiphile porteur de radicaux hydrophobes
US20200179489A1 (en) * 2018-12-07 2020-06-11 Adocia Injectable solution at ph 7 comprising at least one basal insulin which pi is from 5.8 to 8.5 and a co-polyamino-acid bearing carboxylate charges and hydrophobic radicals and a limited amount of m-cresol
WO2020115334A1 (fr) * 2018-12-07 2020-06-11 Adocia Procede de preparation d'une composition stable sous forme d'une solution aqueuse injectable
WO2020245470A1 (fr) 2019-06-07 2020-12-10 Adocia Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5, du liraglutide et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985001890A1 (fr) 1983-10-26 1985-05-09 Kanebo, Ltd. Agent emulsifiant proteique, son procede de preparation et preparation cosmetique emulsifiee le contenant
DE3837825A1 (de) 1988-11-08 1990-05-10 Hoechst Ag Neue insulinderivate, ihre verwendung und eine sie enthaltende pharmazeutische zubereitung
FR2801226B1 (fr) 1999-11-23 2002-01-25 Flamel Tech Sa Suspension colloidale de particules submicroniques de vectorisation de principes actifs et son mode de preparation
EP1545460A4 (en) 2001-12-20 2005-11-16 Lilly Co Eli INSULIN MOLECULE WITH TEMPORARY EFFECT
FR2840614B1 (fr) 2002-06-07 2004-08-27 Flamel Tech Sa Polyaminoacides fonctionnalises par de l'alpha-tocopherol et leurs applications notamment therapeutiques
CA2518776A1 (en) 2003-04-29 2004-11-11 Eli Lilly And Company Insulin analogs having protracted time action
FR2862535B1 (fr) * 2003-11-21 2007-11-23 Flamel Tech Sa Formulations pharmaceutiques pour la liberation prolongee d'interleukines et leurs applications therapeutiques
FR2915683B1 (fr) * 2007-05-03 2009-08-07 Flamel Technologies Sa Formulations pharmaceutiques auto-precipitantes pour la liberation modifiee de principe actif
CN103889442B (zh) * 2011-08-10 2016-12-28 阿道恰公司 至少一种基础胰岛素的可注射溶液
FR2985429B1 (fr) 2012-01-09 2016-07-29 Adocia Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un polyaminoacide substitue obtenu par un procede de polymerisation controle
CN113730555A (zh) * 2012-01-09 2021-12-03 阿道恰公司 Ph为7且至少含pi为5.8至8.5之基础胰岛素和取代共聚(氨基酸)的可注射溶液
FR3001896B1 (fr) 2013-02-12 2015-07-03 Adocia Solution injectable a ph 7 comprenant au moins une insuline basale dont le point isolectrique est compris entre 5,8 et 8,5 et un polymere anionique hydrophobise
FR3001895B1 (fr) 2013-02-12 2015-07-03 Adocia Solution injectable a ph7 comprenant au moins une insuline basale dont le point isoelectrique est compris en 5,8 et 8,5 et un compose anionique porteur de charges carboxylates et de radicaux hydrophobes

Also Published As

Publication number Publication date
US20170348396A1 (en) 2017-12-07
US10548952B2 (en) 2020-02-04
CN109640953A (zh) 2019-04-16
CN109379888A (zh) 2019-02-22
EA039333B1 (ru) 2022-01-14
EA039363B1 (ru) 2022-01-18
SG11201810937WA (en) 2019-01-30
WO2017211916A1 (fr) 2017-12-14
EA201892737A1 (ru) 2019-05-31
BR112018075151A2 (pt) 2019-03-26
FR3052072A1 (fr) 2017-12-08
PH12018502558A1 (en) 2019-10-14
CN109640953B (zh) 2021-10-29
EP3463293A1 (fr) 2019-04-10
JP2019517555A (ja) 2019-06-24
WO2017211903A1 (fr) 2017-12-14
BR112018075140A2 (pt) 2019-03-26
EP3463292B1 (fr) 2020-08-05
MX2018015068A (es) 2019-05-09
PH12018502558B1 (en) 2024-02-02
SA518400588B1 (ar) 2022-03-07
EA201892736A1 (ru) 2019-05-31
SA518400596B1 (ar) 2022-03-16
US20170348423A1 (en) 2017-12-07
US10383920B2 (en) 2019-08-20
EP3463293B1 (fr) 2021-05-12
SG11201810935SA (en) 2019-01-30
EP3463292A1 (fr) 2019-04-10
CN109379888B (zh) 2021-10-29

Similar Documents

Publication Publication Date Title
PH12018502558B1 (en) Injectable solution at ph 7, comprising at least one basal insulin whose pi is between 5.8 and 8.5, a prandial insulin and/or a gastrointestinal hormone, and a copolyamino acid bearing carboxylate charges and hydrophobic radicals
MX2025009746A (es) Solucion inyectable a ph 7 que comprende al menos una insulina basal que tiene un pi de entre 5.8 y 8.5 y un copoliaminoacido con cargas de carboxilato y radicales hidrofobicos
MX2018015070A (es) Composiciones en forma de solucion acuosa inyectable, que comprende glucagon humano y un co-poliaminoacido injertado en el extremo.
WO2019110797A8 (fr) Compositions sous forme d'une solution aqueuse injectable comprenant de l'amyline, un agoniste au recepteur de l'amyline ou un analogue d'amyline et un co-polyaminoacide
PH12020550828A1 (en) Compositions in the form of an injectable aqueous solution comprising human glucagon and a copolyamino acid
SG11202005322RA (en) Injectable solution at ph 7 comprising at least one basal insulin having a pi of between 5.8 and 8.5 and a copolyamino acid carrying carboxylate charges and hydrophobic radicals
MY182507A (en) Aqueous ophthalmic solution
IL272141A (en) Preparations in the form of an aqueous solution for injection containing at least human insulin A21G and suppressing glucagon activity with a meal
FR3001896B1 (fr) Solution injectable a ph 7 comprenant au moins une insuline basale dont le point isolectrique est compris entre 5,8 et 8,5 et un polymere anionique hydrophobise
MX2025008231A (es) Composiciones en forma de una solucion acuosa inyectable que comprende amilina, un receptor agonista de amilina o un analogo de amilina y un copoliaminoacido
SG11202005320VA (en) Compositions in the form of an injectable aqueous solution comprising human glucagon and a copolyamino acid
MX2016004328A (es) Inmunopotenciador.
EA202091374A1 (ru) РАСТВОР ДЛЯ ИНЪЕКЦИЙ С pH 7, СОДЕРЖАЩИЙ ПО МЕНЬШЕЙ МЕРЕ ОДИН БАЗАЛЬНЫЙ ИНСУЛИН С pI МЕЖДУ 5,8 И 8,5 И СОПОЛИАМИНОКИСЛОТУ, НЕСУЩУЮ КАРБОКСИЛАТНЫЕ ЗАРЯДЫ И ГИДРОФОБНЫЕ РАДИКАЛЫ
FR3074681B1 (fr) Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes
MX2020006670A (es) Composicion acuosa que comprende acido 2-(dimetil-1h-pirazol-1-il) succinico y amoniaco.
EA202091387A1 (ru) Композиции в форме инъецируемого водного раствора, содержащие человеческий глюкагон и сополиаминокислоту
SG11201804902UA (en) A composition for improving memory, learning ability, and cognitive ability
FR3074683B1 (fr) Compositions sous forme d'une solution aqueuse injectable comprenant du glucagon humain et un co-polyaminoacide
FR3074422B1 (fr) Solution injectable a ph 7 comprenant au moins une insuline basale dont le pi est compris entre 5,8 et 8,5 et un co-polyaminoacide porteur de charges carboxylates et de radicaux hydrophobes
PL410126A1 (pl) Sposób otrzymywania zawiesiny nanocząstek chitozan-srebro i nanokompozytu chitozan-srebro