MX2017003780A - Composicion farmaceutica para tratar colitis ulcerativa. - Google Patents
Composicion farmaceutica para tratar colitis ulcerativa.Info
- Publication number
- MX2017003780A MX2017003780A MX2017003780A MX2017003780A MX2017003780A MX 2017003780 A MX2017003780 A MX 2017003780A MX 2017003780 A MX2017003780 A MX 2017003780A MX 2017003780 A MX2017003780 A MX 2017003780A MX 2017003780 A MX2017003780 A MX 2017003780A
- Authority
- MX
- Mexico
- Prior art keywords
- ulcerative colitis
- pharmaceutical composition
- treat ulcerative
- pharmaceutically acceptable
- acceptable salt
- Prior art date
Links
- 206010009900 Colitis ulcerative Diseases 0.000 title abstract 3
- 201000006704 Ulcerative Colitis Diseases 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Se proporciona una composición farmacéutica para tratar colitis ulcerativa, que comprende un compuesto representado por una fórmula (1) o una sal farmacéuticamente aceptable del mismo, en donde el compuesto o la sal farmacéuticamente aceptable se administra en una cantidad de 600 mg o más por día a un paciente con colitis ulcerativa.(ver Fórmula).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014198681 | 2014-09-29 | ||
| PCT/JP2015/059717 WO2016051828A1 (ja) | 2014-09-29 | 2015-03-27 | 潰瘍性大腸炎の治療用医薬組成物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX2017003780A true MX2017003780A (es) | 2017-06-30 |
| MX381440B MX381440B (es) | 2025-03-12 |
Family
ID=55629887
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2017003780A MX381440B (es) | 2014-09-29 | 2015-03-27 | Composicion farmaceutica para tratar colitis ulcerativa. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US10183022B2 (es) |
| JP (1) | JP6580053B2 (es) |
| KR (1) | KR102319078B1 (es) |
| AU (1) | AU2015326196B2 (es) |
| BR (1) | BR112017006272A2 (es) |
| CA (1) | CA2961311C (es) |
| EA (1) | EA034956B1 (es) |
| MX (1) | MX381440B (es) |
| WO (1) | WO2016051828A1 (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2973216T3 (es) * | 2018-01-18 | 2024-06-19 | Sterna Biologicals Gmbh | Composición para el tratamiento de un paciente que padece colitis ulcerosa y uso de la composición como medicamento |
| CN112969687B (zh) | 2018-10-30 | 2024-08-23 | 吉利德科学公司 | 作为α4β7整合素抑制剂的喹啉衍生物 |
| ES3003232T3 (en) | 2018-10-30 | 2025-03-10 | Gilead Sciences Inc | Compounds for inhibition of alpha4beta7 integrin |
| CA3115820A1 (en) | 2018-10-30 | 2020-05-07 | Gilead Sciences, Inc. | Compounds for inhibition of .alpha.4.beta.7 integrin |
| EP3873900B1 (en) | 2018-10-30 | 2025-01-08 | Gilead Sciences, Inc. | Imidazo[1,2-a]pyridine derivatives as alpha4beta7 integrin inhibitors for the treatment of inflammatory diseases |
| CA3148613A1 (en) | 2019-08-14 | 2021-02-18 | Gilead Sciences, Inc. | Phenylalanine derived compounds and their use as inhinitors of alpha 4 beta 7 integrin |
| GB202002926D0 (en) * | 2020-02-28 | 2020-04-15 | Benevolentai Tech Limited | Compositions and uses thereof |
| KR102758046B1 (ko) | 2021-11-05 | 2025-01-23 | (주) 넥셀 | 궤양성 대장염 예방 또는 치료용 재조합 단백질 및 이를 포함하는 궤양성 대장염 예방 또는 치료용 조성물 |
| CN114668775B (zh) * | 2022-02-28 | 2023-12-19 | 中国药科大学 | 纤维素衍生物在制备治疗溃疡性结肠炎药物中的应用 |
| WO2023171789A1 (ja) | 2022-03-11 | 2023-09-14 | 国立大学法人大阪大学 | Vla-4の阻害物質を含む、心筋炎を予防、又は治療するための組成物 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2286340C2 (ru) | 2000-08-18 | 2006-10-27 | Адзиномото Ко., Инк. | Новые производные фенилаланина |
| EP1595870B1 (en) | 2003-02-20 | 2015-09-23 | Ajinomoto Co., Inc. | Process for producing phenylalanine derivative having quinazolinedione skeleton and intermediate for the same |
| JP4780522B2 (ja) | 2003-11-14 | 2011-09-28 | 味の素株式会社 | フェニルアラニン誘導体の固体分散体または固体分散体医薬製剤 |
| WO2005046697A1 (ja) | 2003-11-14 | 2005-05-26 | Ajinomoto Co., Inc. | フェニルアラニン誘導体の徐放性経口投与製剤 |
| WO2005051525A1 (en) | 2003-11-25 | 2005-06-09 | Polyvalor, Limited Partnership | Permeation barrier coating or layer with modulated properties and methods of making the same |
| JP4748449B2 (ja) | 2003-11-27 | 2011-08-17 | 味の素株式会社 | フェニルアラニン誘導体の結晶及びその製造方法 |
| CN102503899B (zh) | 2005-06-21 | 2014-09-24 | 味之素株式会社 | 苯基丙氨酸衍生物的结晶、其制备方法及其应用 |
| AU2007322637B2 (en) | 2006-11-22 | 2012-07-05 | Ea Pharma Co., Ltd. | Process for production of phenylalanine derivatives having quinazolinedione skeletons and intermediates for the production |
| US7987289B2 (en) | 2008-06-24 | 2011-07-26 | Microsoft Corporation | Participating in cloud as totally stubby edge |
| EP2993173A1 (en) * | 2010-03-29 | 2016-03-09 | Ajinomoto Co., Inc. | Crystals of salts of phenylalanine derivatives |
| WO2011122620A1 (ja) | 2010-03-29 | 2011-10-06 | 味の素株式会社 | フェニルアラニン誘導体を含有する医薬製剤 |
-
2015
- 2015-03-27 BR BR112017006272-0A patent/BR112017006272A2/pt not_active Application Discontinuation
- 2015-03-27 KR KR1020177011379A patent/KR102319078B1/ko not_active Expired - Fee Related
- 2015-03-27 JP JP2016551565A patent/JP6580053B2/ja active Active
- 2015-03-27 MX MX2017003780A patent/MX381440B/es unknown
- 2015-03-27 EA EA201790726A patent/EA034956B1/ru not_active IP Right Cessation
- 2015-03-27 CA CA2961311A patent/CA2961311C/en active Active
- 2015-03-27 WO PCT/JP2015/059717 patent/WO2016051828A1/ja not_active Ceased
- 2015-03-27 AU AU2015326196A patent/AU2015326196B2/en not_active Ceased
-
2017
- 2017-03-28 US US15/471,745 patent/US10183022B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| BR112017006272A2 (pt) | 2018-03-13 |
| AU2015326196A1 (en) | 2017-03-23 |
| CA2961311C (en) | 2022-12-06 |
| KR20170057435A (ko) | 2017-05-24 |
| CA2961311A1 (en) | 2016-04-07 |
| JPWO2016051828A1 (ja) | 2017-07-27 |
| AU2015326196B2 (en) | 2020-05-14 |
| US20170196870A1 (en) | 2017-07-13 |
| JP6580053B2 (ja) | 2019-09-25 |
| MX381440B (es) | 2025-03-12 |
| EA201790726A1 (ru) | 2017-11-30 |
| KR102319078B1 (ko) | 2021-10-29 |
| US10183022B2 (en) | 2019-01-22 |
| EA034956B1 (ru) | 2020-04-10 |
| WO2016051828A1 (ja) | 2016-04-07 |
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