[go: up one dir, main page]

MX2017002853A - Nueva composicion farmaceutica para la prevencion y/o el tratamiento de la incontinencia urinaria. - Google Patents

Nueva composicion farmaceutica para la prevencion y/o el tratamiento de la incontinencia urinaria.

Info

Publication number
MX2017002853A
MX2017002853A MX2017002853A MX2017002853A MX2017002853A MX 2017002853 A MX2017002853 A MX 2017002853A MX 2017002853 A MX2017002853 A MX 2017002853A MX 2017002853 A MX2017002853 A MX 2017002853A MX 2017002853 A MX2017002853 A MX 2017002853A
Authority
MX
Mexico
Prior art keywords
pharmaceutical composition
urinary incontinence
treatment
novel pharmaceutical
incontinence prevention
Prior art date
Application number
MX2017002853A
Other languages
English (en)
Inventor
Mori Shinobu
Inamura Hiroko
Hirata Takuya
Kajihara Yusuke
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of MX2017002853A publication Critical patent/MX2017002853A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/136Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

El problema a resolver por la presente invención es proporcionar una nueva composición farmacéutica para la prevención y/o el tratamiento de la incontinencia urinaria, que difiere de los fármacos convencionales. La presente invención proporciona un agente terapéutico para la prevención y/o el tratamiento de la incontinencia urinaria que tiene 1-[2-({[trans-3-fluoro-1-(3-fluor opiridin-2-il) ciclobutil]metil}amino)pirimidin-5-il]-1H-pirrol-3- carboxamida o una sal de la misma, como ingrediente activo.
MX2017002853A 2014-09-09 2015-09-09 Nueva composicion farmaceutica para la prevencion y/o el tratamiento de la incontinencia urinaria. MX2017002853A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2014183434 2014-09-09
PCT/JP2015/075567 WO2016039367A1 (ja) 2014-09-09 2015-09-09 尿失禁予防用及び/又は治療用新規医薬組成物

Publications (1)

Publication Number Publication Date
MX2017002853A true MX2017002853A (es) 2018-01-12

Family

ID=55459111

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017002853A MX2017002853A (es) 2014-09-09 2015-09-09 Nueva composicion farmaceutica para la prevencion y/o el tratamiento de la incontinencia urinaria.

Country Status (18)

Country Link
US (1) US9987279B2 (es)
EP (1) EP3192512B1 (es)
JP (1) JP6573618B2 (es)
KR (1) KR102460731B1 (es)
CN (1) CN106687115B (es)
AU (1) AU2015313221B2 (es)
BR (1) BR112017004505A2 (es)
CA (1) CA2957804C (es)
ES (1) ES2750751T3 (es)
IL (1) IL250919B (es)
MX (1) MX2017002853A (es)
PH (1) PH12017500436A1 (es)
PL (1) PL3192512T3 (es)
PT (1) PT3192512T (es)
RU (1) RU2738886C9 (es)
SG (1) SG11201701019UA (es)
WO (1) WO2016039367A1 (es)
ZA (1) ZA201701671B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9133123B2 (en) 2010-04-23 2015-09-15 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
AR081331A1 (es) 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
AR081626A1 (es) 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
RU2743424C2 (ru) 2016-02-12 2021-02-18 Астеллас Фарма Инк. Производные тетрагидроизохинолина
KR20200109314A (ko) * 2017-12-26 2020-09-22 싸이토키네틱스, 인코포레이티드 아미노-피리미딘 및 이의 중간체의 제조 공정
MX2023004745A (es) 2020-11-06 2023-05-10 Cytokinetics Inc 1,4-diazepanonas biciclicas y sus usos terapeuticos.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR122018003623B8 (pt) 2004-03-05 2021-07-27 Hoffmann La Roche diaminopirimidinas, seus usos, e composição farmacêutica
CA2646729A1 (en) * 2005-03-21 2006-09-28 Dov Pharmaceutical, Inc. Methods and compositions for the treatment of urinary incontinence
JP2007176933A (ja) * 2005-11-29 2007-07-12 Tanabe Seiyaku Co Ltd 医薬組成物
JP2007290970A (ja) * 2006-04-21 2007-11-08 Astellas Pharma Inc 腹圧性及び混合型尿失禁治療剤
JPWO2008072778A1 (ja) 2006-12-13 2010-04-02 あすか製薬株式会社 尿路系疾患の処置剤
PL2216021T3 (pl) 2007-11-02 2013-03-29 Astellas Pharma Inc Kompozycja farmaceutyczna do leczenia zespołu pęcherza nadreaktywnego
JP5553547B2 (ja) 2009-07-14 2014-07-16 俊一 梶岡 トロポニン含有医薬組成物
AR081331A1 (es) * 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
US20150065525A1 (en) 2012-04-02 2015-03-05 Cytokinetics, Inc. Methods for improving diaphragm function
SG11201406359TA (en) 2012-04-11 2014-11-27 Cytokinetics Inc Improving resistance to skeletal muscle fatigue

Also Published As

Publication number Publication date
US9987279B2 (en) 2018-06-05
JP6573618B2 (ja) 2019-09-11
CA2957804A1 (en) 2016-03-17
PT3192512T (pt) 2019-10-29
PL3192512T3 (pl) 2020-03-31
RU2017111848A3 (es) 2019-07-17
ZA201701671B (en) 2019-06-26
RU2017111848A (ru) 2018-10-08
US20170273979A1 (en) 2017-09-28
JPWO2016039367A1 (ja) 2017-06-15
PH12017500436A1 (en) 2017-07-31
RU2738886C9 (ru) 2021-12-06
RU2738886C2 (ru) 2020-12-18
EP3192512B1 (en) 2019-08-14
KR102460731B1 (ko) 2022-10-28
AU2015313221A1 (en) 2017-03-09
BR112017004505A2 (pt) 2018-01-23
CN106687115A (zh) 2017-05-17
SG11201701019UA (en) 2017-03-30
EP3192512A1 (en) 2017-07-19
ES2750751T3 (es) 2020-03-27
CN106687115B (zh) 2019-07-19
KR20170045353A (ko) 2017-04-26
WO2016039367A1 (ja) 2016-03-17
EP3192512A4 (en) 2018-02-07
IL250919A0 (en) 2017-04-30
AU2015313221B2 (en) 2019-11-21
CA2957804C (en) 2023-04-04
IL250919B (en) 2019-10-31

Similar Documents

Publication Publication Date Title
NZ775660A (en) Combination therapy including a krasg12c inhibitor and one or more additional pharmaceutically active agents for the treatment of cancers
JOP20190186A1 (ar) مركب كينازولين
PH12017500436A1 (en) Novel pharmaceutical composition for prevention and/or treatment of urinary incontinence
SG11202106160WA (en) Pharmaceutical composition for prevention or treatment of cancer comprising weissella cibaria wikim28 as active ingredient
MX2023002507A (es) Inhibidores de cd73.
MY197700A (en) Compounds useful for inhibiting cdk7
ZA202204941B (en) Cd73 inhibitors
MX2016016593A (es) Nuevos derivados de aminoalquibenzotiazepina y usos de los mismos.
MX2016012574A (es) Compuestos heteroarilo sustituidos y metodos de uso.
SA518400356B1 (ar) مثبطات الأرجيناز واستخداماتها العلاجية
MX2020002271A (es) Composiciones farmaceuticas que comprenden sepiapterina y sus usos de las mismas.
WO2016028391A3 (en) Spiropyrrolidines as mdm2 inhibitors
JOP20180071A1 (ar) استخدام مشتقات أمينو ألكيل بنزوثيازبين
WO2015015378A3 (en) Heterobicycloaryl rorc2 inhibitors and methods of use thereof
PH12016501619A1 (en) Substituted fused heterocycles as gpr119 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders
SG11202112796YA (en) N-containing heteroaryl derivative and pharmaceutical composition comprising same as active ingredient for prevention or treatment of cancer
PH12016501527B1 (en) Pharmaceutical composition comprising diamino heterocyclic carboxamide compound as active ingredient
MX2019006863A (es) Inhibidores de heparanasa y uso de los mismos.
EP3541943A4 (en) MICRO-ORGANISM FOR ADMINISTERING A MEDICINAL PRODUCT FOR THE TREATMENT OF A GASTROINTESTINAL DISEASE, WHICH EXPRESSES AND SECRETS P8 PROTEIN, AND PHARMACEUTICAL COMPOSITION CONSISTING OF THIS MICRO-ORGANISM FOR THE PREVENTION OR TREATMENT OF A GASTROINTESTINAL DISEASE
EP3248603A4 (en) Pharmaceutical composition for prevention, treatment or delay of alzheimer's disease or dementia containing g protein-coupled receptor 19 agent as active ingredient
EP3909597A4 (en) PHARMACEUTICAL COMPOSITION FOR THE PREVENTION OR TREATMENT OF CANCER WITH OLIGOPEPTIDE AS THE ACTIVE SUBSTANCE
PH12019501642A1 (en) Novel compounds and their use in the treatment of schistosomiasis
MX2019008338A (es) Composicion farmaceutica que contiene sulglicotido o una sal farmaceuticamente aceptable del mismo para la prevencion o tratamiento del ojo seco.
MX2020008275A (es) Metodos para tratar trastornos mitocondriales.
EP4234021A3 (en) Pharmaceutical composition comprising an adenosine derivative for use in the prevention or treatment of diabetic nephropathy

Legal Events

Date Code Title Description
FG Grant or registration