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MX2016007266A - Metodo para preparar composiciones secas para inhalacion en polvo. - Google Patents

Metodo para preparar composiciones secas para inhalacion en polvo.

Info

Publication number
MX2016007266A
MX2016007266A MX2016007266A MX2016007266A MX2016007266A MX 2016007266 A MX2016007266 A MX 2016007266A MX 2016007266 A MX2016007266 A MX 2016007266A MX 2016007266 A MX2016007266 A MX 2016007266A MX 2016007266 A MX2016007266 A MX 2016007266A
Authority
MX
Mexico
Prior art keywords
excipient
active ingredient
dry powder
powder inhalation
preparing dry
Prior art date
Application number
MX2016007266A
Other languages
English (en)
Other versions
MX368857B (es
Inventor
Mattila Terhi
Happonen Anita
Haikarainen Jussi
Original Assignee
Orion Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52146529&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2016007266(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Orion Corp filed Critical Orion Corp
Publication of MX2016007266A publication Critical patent/MX2016007266A/es
Publication of MX368857B publication Critical patent/MX368857B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Otolaryngology (AREA)
  • Emergency Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se describe un método para preparar composiciones secas para inhalación en polvo que comprenden dos o más ingredientes activos y excipiente en partículas inerte y un método para ajustar el rendimiento de tales composiciones. El método comprende mezclar el primer ingrediente activo y una porción del segundo ingrediente activo con un primer excipiente para proporcionar una primera premezcla, mezclar la porción restante del segundo ingrediente activo con un segundo excipiente para proporcionar una segunda premezcla y finalmente mezclar juntas la primera y la segunda premezcla, en donde los dos grados del excipiente difieren en su tamaño medio de partícula. El nivel de la FPD del segundo ingrediente activo se puede ajustar simplemente al cambiar la relación de cómo se divide el primero y el segundo excipiente.
MX2016007266A 2013-12-06 2014-12-05 Metodo para preparar composiciones secas para inhalacion en polvo. MX368857B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361913024P 2013-12-06 2013-12-06
PCT/FI2014/000038 WO2015082756A1 (en) 2013-12-06 2014-12-05 Method for preparing dry powder inhalation compositions

Publications (2)

Publication Number Publication Date
MX2016007266A true MX2016007266A (es) 2016-09-07
MX368857B MX368857B (es) 2019-10-18

Family

ID=52146529

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016007266A MX368857B (es) 2013-12-06 2014-12-05 Metodo para preparar composiciones secas para inhalacion en polvo.

Country Status (26)

Country Link
EP (1) EP3076957B1 (es)
JP (1) JP6353049B2 (es)
KR (1) KR102255402B1 (es)
CN (2) CN105873575A (es)
AU (1) AU2014359111B2 (es)
BR (1) BR112016012871B1 (es)
CA (1) CA2928695C (es)
CL (1) CL2016001359A1 (es)
CY (1) CY1122797T1 (es)
DK (1) DK3076957T3 (es)
EA (1) EA033247B1 (es)
ES (1) ES2776350T3 (es)
HR (1) HRP20200618T1 (es)
HU (1) HUE049162T2 (es)
LT (1) LT3076957T (es)
MA (1) MA39089B1 (es)
MX (1) MX368857B (es)
MY (1) MY185073A (es)
PH (1) PH12016501045B1 (es)
PL (1) PL3076957T3 (es)
PT (1) PT3076957T (es)
SA (1) SA516371266B1 (es)
SI (1) SI3076957T1 (es)
UA (1) UA118861C2 (es)
WO (1) WO2015082756A1 (es)
ZA (1) ZA201602909B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3082692A1 (en) * 2013-12-20 2016-10-26 The Procter & Gamble Company Diaper with improved cuffs and fit
US20230225973A1 (en) * 2020-06-26 2023-07-20 Mylan Pharma Uk Limited Multi-layered medicament for inhalation
WO2024010539A1 (en) * 2022-07-07 2024-01-11 Arven Ilac Sanayi Ve Ticaret Anonim Sirketi A process for the preparation of dry powder compositions for inhalation using different mixers
CN115364075B (zh) * 2022-09-16 2023-11-10 苏州易合医药有限公司 一种吸入颗粒组合物及其制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4140689B4 (de) * 1991-12-10 2007-11-22 Boehringer Ingelheim Kg Inhalationspulver und Verfahren zu ihrer Herstellung
US6369115B1 (en) * 2000-03-20 2002-04-09 Dura Pharmaceuticals, Inc. Stabilized powder formulations
GB0012260D0 (en) * 2000-05-19 2000-07-12 Astrazeneca Ab Novel composition
WO2003024396A2 (en) * 2001-09-17 2003-03-27 Glaxo Group Limited Dry powder medicament formulations
JP3691459B2 (ja) * 2002-06-14 2005-09-07 久光メディカル株式会社 粉末状吸入剤組成物
JP4744876B2 (ja) * 2002-08-21 2011-08-10 ノートン・ヘルスケアー リミテッド 乾燥粉末吸入組成物の製造方法
GB0219512D0 (en) * 2002-08-21 2002-10-02 Norton Healthcare Ltd Inhalation compositions with high drug ratios
GB0714134D0 (en) * 2007-07-19 2007-08-29 Norton Healthcare Ltd Dry-powder medicament
EP2221048A1 (en) * 2009-02-18 2010-08-25 Siegfried Generics International AG Pharmaceutical composition for inhalation
WO2011145109A1 (en) * 2010-05-20 2011-11-24 Sun Pharma Advanced Research Company Ltd., Dry powder inhalation composition
FI3412277T3 (fi) * 2012-01-25 2023-03-23 Chiesi Farm Spa Kortikosteroidia ja beeta-adrenergista ainetta käsittävä kuivajauheformulaatio annettavaksi inhalaatiolla

Also Published As

Publication number Publication date
LT3076957T (lt) 2020-03-10
WO2015082756A1 (en) 2015-06-11
CA2928695A1 (en) 2015-06-11
CL2016001359A1 (es) 2016-11-18
JP6353049B2 (ja) 2018-07-04
ES2776350T3 (es) 2020-07-30
CA2928695C (en) 2022-03-29
KR20160093718A (ko) 2016-08-08
PT3076957T (pt) 2020-03-05
MY185073A (en) 2021-04-30
CN113908142A (zh) 2022-01-11
ZA201602909B (en) 2017-04-26
HRP20200618T1 (hr) 2020-07-10
KR102255402B1 (ko) 2021-05-24
MA39089A1 (fr) 2017-10-31
PL3076957T3 (pl) 2020-06-29
UA118861C2 (uk) 2019-03-25
SI3076957T1 (sl) 2020-04-30
PH12016501045A1 (en) 2016-07-25
BR112016012871B1 (pt) 2022-10-11
MA39089B1 (fr) 2019-03-29
AU2014359111A1 (en) 2016-05-19
JP2016539151A (ja) 2016-12-15
BR112016012871A2 (pt) 2020-08-04
DK3076957T3 (da) 2020-04-27
MX368857B (es) 2019-10-18
PH12016501045B1 (en) 2016-07-25
CN105873575A (zh) 2016-08-17
AU2014359111B2 (en) 2019-06-13
HUE049162T2 (hu) 2020-09-28
EP3076957A1 (en) 2016-10-12
NZ719346A (en) 2021-01-29
EA201691181A1 (ru) 2016-09-30
EP3076957B1 (en) 2020-02-05
SA516371266B1 (ar) 2019-08-01
CY1122797T1 (el) 2021-05-05
EA033247B1 (ru) 2019-09-30

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