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MX2011007195A - Derivado de ciclosporina para el uso en el tratamiento de infección de virus de hepatitis c (vhc) y virus de inmunodeficiencia humana (vih). - Google Patents

Derivado de ciclosporina para el uso en el tratamiento de infección de virus de hepatitis c (vhc) y virus de inmunodeficiencia humana (vih).

Info

Publication number
MX2011007195A
MX2011007195A MX2011007195A MX2011007195A MX2011007195A MX 2011007195 A MX2011007195 A MX 2011007195A MX 2011007195 A MX2011007195 A MX 2011007195A MX 2011007195 A MX2011007195 A MX 2011007195A MX 2011007195 A MX2011007195 A MX 2011007195A
Authority
MX
Mexico
Prior art keywords
hcv
treatment
hiv infection
cyclosporine derivative
cyclosporine
Prior art date
Application number
MX2011007195A
Other languages
English (en)
Inventor
Samuel Earl Hopkins
Original Assignee
Scynexis Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scynexis Inc filed Critical Scynexis Inc
Publication of MX2011007195A publication Critical patent/MX2011007195A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13Cyclosporins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)

Abstract

En la presente se proporciona dosis especificas de , o regímenes de dosificación para, usar SCY-635 en el tratamiento o prevención de enfermedades, en particular infección por virus de hepatitis C (VHC).
MX2011007195A 2009-01-07 2010-01-07 Derivado de ciclosporina para el uso en el tratamiento de infección de virus de hepatitis c (vhc) y virus de inmunodeficiencia humana (vih). MX2011007195A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14306209P 2009-01-07 2009-01-07
US15602609P 2009-02-27 2009-02-27
PCT/US2010/020316 WO2010080874A1 (en) 2009-01-07 2010-01-07 Cyclosporine derivative for use in the treatment of hcv and hiv infection

Publications (1)

Publication Number Publication Date
MX2011007195A true MX2011007195A (es) 2013-07-12

Family

ID=42101315

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011007195A MX2011007195A (es) 2009-01-07 2010-01-07 Derivado de ciclosporina para el uso en el tratamiento de infección de virus de hepatitis c (vhc) y virus de inmunodeficiencia humana (vih).

Country Status (13)

Country Link
US (1) US20100173837A1 (es)
EP (1) EP2385838A1 (es)
JP (1) JP2012514605A (es)
KR (1) KR20110116136A (es)
CN (1) CN102271699A (es)
AU (1) AU2010203656A1 (es)
CA (1) CA2750227A1 (es)
IL (1) IL213861A0 (es)
MX (1) MX2011007195A (es)
RU (1) RU2011127080A (es)
SG (1) SG172848A1 (es)
WO (1) WO2010080874A1 (es)
ZA (1) ZA201105343B (es)

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KR101089112B1 (ko) * 2006-06-02 2011-12-06 피씨 제스띠옹 에스.아.에스. 활성 전자 관리
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JP5780969B2 (ja) * 2008-12-31 2015-09-16 サイネクシス,インコーポレーテッド シクロスポリンaの誘導体
US9217015B2 (en) 2010-07-16 2015-12-22 S&T Global Inc. Cyclosporin derivatives for the treatment and prevention of a viral infection
US9573978B2 (en) 2010-08-12 2017-02-21 S&T Global, Inc. Cyclosporin derivatives for the treatment and prevention of a viral infection
JP6093307B2 (ja) * 2010-12-03 2017-03-08 エス アンド ティー グローバル インク. ウイルス感染の治療および予防のための新規シクロスポリン誘導体
US9890198B2 (en) 2010-12-03 2018-02-13 S&T Global Inc. Cyclosporin derivatives and uses thereof
WO2012097123A2 (en) * 2011-01-12 2012-07-19 Scynexis, Inc. New uses of cyclophilin inhibitors
EP2747569A4 (en) * 2011-08-24 2015-07-08 Glaxosmithkline Llc COMBINATION TREATMENTS FOR HEPATITIS C
MX381953B (es) 2016-02-25 2025-03-13 Asceneuron S A Sales de derivados de piperazina obtenidas por adicion de acidos.
CN106554392B (zh) * 2016-11-21 2019-10-25 石家庄中天生物技术有限责任公司 一种高纯度环孢菌素衍生物stg-175的制备方法
US11845809B2 (en) * 2018-12-14 2023-12-19 Waterstone Pharmaceuticals(Wuhan) Co., Ltd. Maleate of SCY-635 and uses thereof in medicine
WO2021068188A1 (en) * 2019-10-11 2021-04-15 Waterstone Pharmaceuticals(Wuhan) Co., Ltd. Ws-635 uses thereof in medicine
IL309862A (en) * 2021-07-05 2024-02-01 Ferrer Int Medicines that include glycosidase inhibitors
WO2024158815A1 (en) * 2023-01-24 2024-08-02 The General Hospital Corporation Use of ws635 to treat alzheimer's disease

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JP2012514605A (ja) 2012-06-28
RU2011127080A (ru) 2013-02-20
WO2010080874A1 (en) 2010-07-15
CN102271699A (zh) 2011-12-07
CA2750227A1 (en) 2010-07-15
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AU2010203656A2 (en) 2011-09-08

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