MC1985A1 - Derives d'acides amines - Google Patents
Derives d'acides aminesInfo
- Publication number
- MC1985A1 MC1985A1 MC882008A MC2008A MC1985A1 MC 1985 A1 MC1985 A1 MC 1985A1 MC 882008 A MC882008 A MC 882008A MC 2008 A MC2008 A MC 2008A MC 1985 A1 MC1985 A1 MC 1985A1
- Authority
- MC
- Monaco
- Prior art keywords
- hydroxy
- isopropyl
- cyclohexylmethyl
- acid
- carbamoyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
- C07C237/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
- C07C237/08—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atom of at least one of the carboxamide groups bound to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0227—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the (partial) peptide sequence -Phe-His-NH-(X)2-C(=0)-, e.g. Renin-inhibitors with n = 2 - 6; for n > 6 see C07K5/06 - C07K5/10
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
- C07K5/0823—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Furan Compounds (AREA)
- Pyridine Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Indole Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH390387 | 1987-10-06 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MC1985A1 true MC1985A1 (fr) | 1989-11-23 |
Family
ID=4265984
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MC882008A MC1985A1 (fr) | 1987-10-06 | 1988-10-03 | Derives d'acides amines |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP0310918A3 (pt) |
| JP (1) | JPH02256658A (pt) |
| KR (1) | KR890006572A (pt) |
| AU (1) | AU627156B2 (pt) |
| DK (1) | DK523288A (pt) |
| FI (1) | FI884598A7 (pt) |
| HU (1) | HUT49322A (pt) |
| IL (1) | IL87871A0 (pt) |
| MC (1) | MC1985A1 (pt) |
| NO (1) | NO884434L (pt) |
| NZ (1) | NZ226395A (pt) |
| PT (1) | PT88679A (pt) |
| YU (1) | YU185188A (pt) |
| ZA (1) | ZA887322B (pt) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU595309B2 (en) * | 1986-05-09 | 1990-03-29 | Dainippon Pharmaceutical Co. Ltd. | Tripeptide derivatives |
| US4895834A (en) * | 1986-12-15 | 1990-01-23 | Warner-Lambert Company | Renin inhibitors III |
| US5023236A (en) * | 1988-04-07 | 1991-06-11 | Corvas, Inc. | Factor VII/VIIA active site inhibitors |
| EP0391180A3 (de) * | 1989-04-04 | 1991-04-03 | F. Hoffmann-La Roche Ag | Peptidartige Aminosäurederivate mit reninhemmender Wirkung |
| CA2012901A1 (en) * | 1989-04-05 | 1990-10-05 | Quirico Branca | Amino acid derivatives |
| US5374731A (en) * | 1989-09-12 | 1994-12-20 | Hoechst Aktiengesellschaft | Amino acid derivatives with renin-inhibiting properties, a process for the preparation thereof, agents containing these, and the use thereof |
| DE4008403A1 (de) * | 1990-03-16 | 1991-09-19 | Merck Patent Gmbh | Glykolsaeurederivate |
| US5516784A (en) * | 1991-08-13 | 1996-05-14 | Schering Corporation | Anti-HIV (AIDS) agents |
| US5422349A (en) * | 1992-08-14 | 1995-06-06 | G. D. Seale & Co. | Morpholino-oxazinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension |
| US5693815A (en) * | 1993-01-17 | 1997-12-02 | Schering Corporation | Peptides |
| US5563127A (en) * | 1993-03-24 | 1996-10-08 | The Dupont Merck Pharmaceutical Company | Boronic acid and ester inhibitors of thrombin |
| FR2741066B1 (fr) * | 1995-11-14 | 1997-12-12 | Rhone Poulenc Rorer Sa | Nouveaux agents de transfection et leurs applications pharmaceutiques |
| FR2752422B1 (fr) * | 1996-08-16 | 1998-11-06 | Lipha | Composition pharmaceutique contenant des acides 4-oxo-butanoiques |
| YU68900A (sh) * | 1998-05-12 | 2002-12-10 | Warner-Lambert Company | Kombinacije inhibitora protein farnesiltransferaze i hmg coa reduktaze i njihova upotreba u tretmanu raka |
| AU2008247488B2 (en) * | 2007-05-04 | 2014-02-27 | Marina Biotech, Inc. | Amino acid lipids and uses thereof |
| GB0919194D0 (en) | 2009-11-02 | 2009-12-16 | Lytix Biopharma As | Compounds |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4652551A (en) * | 1984-06-22 | 1987-03-24 | Abbott Laboratories | Renin inhibiting compounds |
| DK34086A (da) * | 1985-01-23 | 1986-07-24 | Abbott Lab | Peptidylaminodioler |
| IL81234A (en) * | 1986-01-16 | 1992-09-06 | Abbott Lab | Peptidylaminodiols,process for their preparation and pharmaceutical compositions comprising them |
| US4792555A (en) * | 1987-03-20 | 1988-12-20 | American Home Products Corporation | Phospholipase A2 inhibitors |
-
1988
- 1988-09-20 DK DK523288A patent/DK523288A/da not_active Application Discontinuation
- 1988-09-27 EP EP19880115878 patent/EP0310918A3/de not_active Withdrawn
- 1988-09-29 NZ NZ226395A patent/NZ226395A/en unknown
- 1988-09-29 IL IL87871A patent/IL87871A0/xx unknown
- 1988-09-29 ZA ZA887322A patent/ZA887322B/xx unknown
- 1988-09-30 AU AU23307/88A patent/AU627156B2/en not_active Ceased
- 1988-10-03 HU HU885114A patent/HUT49322A/hu unknown
- 1988-10-03 MC MC882008A patent/MC1985A1/fr unknown
- 1988-10-04 YU YU01851/88A patent/YU185188A/xx unknown
- 1988-10-05 KR KR1019880012964A patent/KR890006572A/ko not_active Withdrawn
- 1988-10-05 NO NO88884434A patent/NO884434L/no unknown
- 1988-10-06 FI FI884598A patent/FI884598A7/fi not_active IP Right Cessation
- 1988-10-06 JP JP63252886A patent/JPH02256658A/ja active Pending
- 1988-10-06 PT PT88679A patent/PT88679A/pt unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA887322B (en) | 1989-06-28 |
| FI884598A0 (fi) | 1988-10-06 |
| EP0310918A2 (de) | 1989-04-12 |
| NZ226395A (en) | 1991-12-23 |
| PT88679A (pt) | 1989-07-31 |
| YU185188A (en) | 1990-12-31 |
| AU2330788A (en) | 1989-06-08 |
| IL87871A0 (en) | 1989-03-31 |
| AU627156B2 (en) | 1992-08-20 |
| DK523288A (da) | 1989-04-07 |
| FI884598A7 (fi) | 1989-04-07 |
| EP0310918A3 (de) | 1990-12-12 |
| DK523288D0 (da) | 1988-09-20 |
| NO884434L (no) | 1989-04-07 |
| KR890006572A (ko) | 1989-06-14 |
| HUT49322A (en) | 1989-09-28 |
| NO884434D0 (no) | 1988-10-05 |
| JPH02256658A (ja) | 1990-10-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| YP | Annual fee paid |