MC1769A1 - Diphenaylpiperidines n-substituees - Google Patents
Diphenaylpiperidines n-substitueesInfo
- Publication number
- MC1769A1 MC1769A1 MC861851A MC1851A MC1769A1 MC 1769 A1 MC1769 A1 MC 1769A1 MC 861851 A MC861851 A MC 861851A MC 1851 A MC1851 A MC 1851A MC 1769 A1 MC1769 A1 MC 1769A1
- Authority
- MC
- Monaco
- Prior art keywords
- formula
- pyridine
- diphenylethenyl
- piperidinyl
- het
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/785,113 US4632925A (en) | 1985-10-07 | 1985-10-07 | N-substituted diphenylpiperidines and antiobesity use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MC1769A1 true MC1769A1 (fr) | 1987-07-17 |
Family
ID=25134481
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MC861851A MC1769A1 (fr) | 1985-10-07 | 1986-10-06 | Diphenaylpiperidines n-substituees |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US4632925A (pt) |
| EP (1) | EP0221376B1 (pt) |
| JP (1) | JPH0633254B2 (pt) |
| KR (1) | KR870003984A (pt) |
| AR (1) | AR241422A1 (pt) |
| AT (1) | ATE53997T1 (pt) |
| AU (1) | AU593844B2 (pt) |
| CA (1) | CA1281326C (pt) |
| DE (1) | DE3672134D1 (pt) |
| DK (1) | DK168291B1 (pt) |
| ES (1) | ES2005074A6 (pt) |
| FI (1) | FI85020C (pt) |
| GR (1) | GR862513B (pt) |
| HU (1) | HU196200B (pt) |
| IE (1) | IE59434B1 (pt) |
| IL (1) | IL80232A0 (pt) |
| MC (1) | MC1769A1 (pt) |
| NO (1) | NO166127C (pt) |
| NZ (1) | NZ217798A (pt) |
| PH (1) | PH24167A (pt) |
| PT (1) | PT83495B (pt) |
| SG (1) | SG17593G (pt) |
| ZA (1) | ZA867375B (pt) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL78939A (en) * | 1986-01-17 | 1990-04-29 | Robins Co Inc A H | Pharmaceutical compositions containing n-substituted arylalkyl-and arylalkylene-piperidines and tetrahydropyridines and certain such novel compounds |
| GB9000305D0 (en) * | 1990-01-06 | 1990-03-07 | Pfizer Ltd | Anticholinergic agents |
| AU646519B2 (en) * | 1990-10-10 | 1994-02-24 | Schering Corporation | Pyridine and pyridine N-oxide derivatives of diaryl methyl piperidines or piperazines, and compositions and methods of use thereof |
| WO1993020063A1 (en) * | 1992-03-27 | 1993-10-14 | Schering Corporation | Unbridged bis-aryl carbinol derivatives, compositions and methods of use |
| TW381025B (en) * | 1993-08-05 | 2000-02-01 | Hoffmann La Roche | Pharmaceutical composition containing a glucosidase inhibitor and a lipase inhibitor |
| US6184234B1 (en) * | 1994-03-01 | 2001-02-06 | Fmc Corporation | Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines |
| US6030987A (en) * | 1996-05-17 | 2000-02-29 | Fmc Corporation | Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines |
| US5639763A (en) * | 1994-03-01 | 1997-06-17 | Fmc Corporation | Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl)methyl]piperidines |
| US6017931A (en) * | 1994-03-01 | 2000-01-25 | Fmc Corporation | Insecticidal compositions containing n-(substituted phenylmethyl)-4-[bis(substituted phenyl)methyl]piperidines |
| JP3168343B2 (ja) * | 1995-05-19 | 2001-05-21 | エフ エム シー コーポレーション | 殺虫性ｎ−（置換されたアリールメチル）−４−〔ビス（置換されたフェニル又はピリジル）メチル〕ピペリジン |
| JP4064460B2 (ja) * | 1996-03-01 | 2008-03-19 | ノボ ノルディスク アクティーゼルスカブ | 食欲抑制性ペプチドを含む医薬組成物の用途 |
| WO1999014203A1 (en) | 1997-09-16 | 1999-03-25 | Takeda Chemical Industries, Ltd. | Nitrogenous fused-ring compounds, process for the preparation of the same, and drugs |
| RU2241462C2 (ru) * | 2000-07-28 | 2004-12-10 | Ф. Хоффманн-Ля Рош Аг | Новая фармацевтическая композиция |
| US20100064413A1 (en) * | 2008-03-14 | 2010-03-18 | Simply Weights, LLC | Exercise clothing and accessories |
| WO2009132979A1 (en) * | 2008-04-29 | 2009-11-05 | F. Hoffmann-La Roche Ag | 4-trimethylammonio-butyrates as cpt2 inhibitors |
| MX2010008196A (es) * | 2008-04-29 | 2010-08-11 | Hoffmann La Roche | Derivados de acido 4-dimetilaminobutirico. |
| EP3737680A1 (en) | 2018-01-08 | 2020-11-18 | F. Hoffmann-La Roche AG | Octahydropyrido[1,2-alpha]pyrazines as magl inhibitors |
| WO2022049134A1 (en) | 2020-09-03 | 2022-03-10 | F. Hoffmann-La Roche Ag | Heterocyclic compounds |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4076717A (en) * | 1971-12-15 | 1978-02-28 | G. D. Searle & Co. | Derivatives of 1-(3-cyano-3,3-diphenylpropyl)-4-phenylpiperidine-4-carboxylic acid |
| US3931197A (en) * | 1974-02-08 | 1976-01-06 | Richardson-Merrell Inc. | Substituted piperidine derivatives |
| US4650874A (en) * | 1984-11-26 | 1987-03-17 | G. D. Searle & Co. | N-(aralkoxybenzyl)-4(benzhydryl) piperidines |
-
1985
- 1985-10-07 US US06/785,113 patent/US4632925A/en not_active Expired - Fee Related
-
1986
- 1986-09-26 ZA ZA867375A patent/ZA867375B/xx unknown
- 1986-10-03 DK DK475286A patent/DK168291B1/da active
- 1986-10-03 HU HU864167A patent/HU196200B/hu not_active IP Right Cessation
- 1986-10-03 CA CA000519718A patent/CA1281326C/en not_active Expired - Lifetime
- 1986-10-03 NZ NZ217798A patent/NZ217798A/xx unknown
- 1986-10-03 IL IL80232A patent/IL80232A0/xx not_active IP Right Cessation
- 1986-10-03 AU AU63501/86A patent/AU593844B2/en not_active Ceased
- 1986-10-06 JP JP61236364A patent/JPH0633254B2/ja not_active Expired - Lifetime
- 1986-10-06 ES ES8602424A patent/ES2005074A6/es not_active Expired
- 1986-10-06 AT AT86113837T patent/ATE53997T1/de not_active IP Right Cessation
- 1986-10-06 EP EP86113837A patent/EP0221376B1/de not_active Expired - Lifetime
- 1986-10-06 DE DE8686113837T patent/DE3672134D1/de not_active Expired - Lifetime
- 1986-10-06 PT PT83495A patent/PT83495B/pt not_active IP Right Cessation
- 1986-10-06 NO NO863978A patent/NO166127C/no unknown
- 1986-10-06 IE IE263686A patent/IE59434B1/en not_active IP Right Cessation
- 1986-10-06 MC MC861851A patent/MC1769A1/fr unknown
- 1986-10-07 FI FI864051A patent/FI85020C/fi not_active IP Right Cessation
- 1986-10-07 GR GR862513A patent/GR862513B/el unknown
- 1986-10-07 PH PH34329A patent/PH24167A/en unknown
- 1986-10-07 KR KR1019860008388A patent/KR870003984A/ko not_active Ceased
- 1986-10-23 AR AR86305473A patent/AR241422A1/es active
-
1993
- 1993-02-17 SG SG175/93A patent/SG17593G/en unknown
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| YP | Annual fee paid |