FI864051L - N-substituerade difenylpiperidiner. - Google Patents

N-substituerade difenylpiperidiner. Download PDF

Info

Publication number: FI864051L
Authority: FI; Finland
Prior art keywords: diphenylpiperidine; substituerade; substituerade diphenylpiperidine
Prior art date: 1985-10-07

Application number

FI864051A

Other languages

English (en)

Other versions

FI85020C (fi

FI85020B (fi

FI864051A0 (fi

Inventor

Jr John Guilfoyle Mullin

Richard Wightman Kierstead

Joseph Triscari

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-10-07

Filing date

1986-10-07

Publication date

1987-04-08

1986-10-07 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

1986-10-07 Publication of FI864051A0 publication Critical patent/FI864051A0/fi

1987-04-08 Publication of FI864051L publication Critical patent/FI864051L/fi

1991-11-15 Application granted granted Critical

1991-11-15 Publication of FI85020B publication Critical patent/FI85020B/fi

1992-02-25 Publication of FI85020C publication Critical patent/FI85020C/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Diabetes (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Hematology (AREA)
Obesity (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

FI864051A 1985-10-07 1986-10-07 Foerfarande foer framstaellning av terapeutiskt aktiva n-substituerade difenylpiperidiner. FI85020C (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US06/785,113 US4632925A (en)	1985-10-07	1985-10-07	N-substituted diphenylpiperidines and antiobesity use thereof
US78511385		1985-10-07

Publications (4)

Publication Number	Publication Date
FI864051A0 FI864051A0 (fi)	1986-10-07
FI864051L true FI864051L (fi)	1987-04-08
FI85020B FI85020B (fi)	1991-11-15
FI85020C FI85020C (fi)	1992-02-25

Family

ID=25134481

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI864051A FI85020C (fi)	1985-10-07	1986-10-07	Foerfarande foer framstaellning av terapeutiskt aktiva n-substituerade difenylpiperidiner.

Country Status (23)

Country	Link
US (1)	US4632925A (fi)
EP (1)	EP0221376B1 (fi)
JP (1)	JPH0633254B2 (fi)
KR (1)	KR870003984A (fi)
AR (1)	AR241422A1 (fi)
AT (1)	ATE53997T1 (fi)
AU (1)	AU593844B2 (fi)
CA (1)	CA1281326C (fi)
DE (1)	DE3672134D1 (fi)
DK (1)	DK168291B1 (fi)
ES (1)	ES2005074A6 (fi)
FI (1)	FI85020C (fi)
GR (1)	GR862513B (fi)
HU (1)	HU196200B (fi)
IE (1)	IE59434B1 (fi)
IL (1)	IL80232A0 (fi)
MC (1)	MC1769A1 (fi)
NO (1)	NO166127C (fi)
NZ (1)	NZ217798A (fi)
PH (1)	PH24167A (fi)
PT (1)	PT83495B (fi)
SG (1)	SG17593G (fi)
ZA (1)	ZA867375B (fi)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IN163948B (fi) *	1986-01-17	1988-12-10	Robins Co Inc A H
GB9000305D0 (en) *	1990-01-06	1990-03-07	Pfizer Ltd	Anticholinergic agents
SK31793A3 (en) *	1990-10-10	1993-09-08	Schering Corp	Pyridine and pyridine n-oxide derivatives of diaryl methyl piperidines and piperazines and compositions and methods of use thereof
EP0635012B1 (en) *	1992-03-27	1996-07-10	Schering Corporation	Unbridged bis-aryl carbinol derivatives, compositions and methods of use
TW381025B (en) *	1993-08-05	2000-02-01	Hoffmann La Roche	Pharmaceutical composition containing a glucosidase inhibitor and a lipase inhibitor
US5639763A (en) *	1994-03-01	1997-06-17	Fmc Corporation	Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl)methyl]piperidines
US6017931A (en) *	1994-03-01	2000-01-25	Fmc Corporation	Insecticidal compositions containing n-(substituted phenylmethyl)-4-[bis(substituted phenyl)methyl]piperidines
US6184234B1 (en) *	1994-03-01	2001-02-06	Fmc Corporation	Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines
US6030987A (en) *	1996-05-17	2000-02-29	Fmc Corporation	Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines
HUP9802550A3 (en) *	1995-05-19	2000-06-28	Fmc Corp	Insecticidal n-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines
BR9707807A (pt) *	1996-03-01	1999-07-27	Novo Nordisk As	Uso de uma composição farmacêutica composição farmacêutica processo de tratar doenças ou distúrbios associados com a regulação do apetite prejudicado e uso de um peptideo
US6407116B1 (en)	1997-09-16	2002-06-18	Takeda Chemical Industries, Inc.	Nitrogenous fused-ring compounds, process for the preparation of the same, and drugs
AU2001289699B2 (en) *	2000-07-28	2006-06-01	Cheplapharm Arzneimittel Gmbh	New pharmaceutical composition
US20100064413A1 (en) *	2008-03-14	2010-03-18	Simply Weights, LLC	Exercise clothing and accessories
KR101225223B1 (ko)	2008-04-29	2013-01-22	에프. 호프만-라 로슈 아게	4-다이메틸아미노부티르산 유도체
RU2502727C2 (ru) *	2008-04-29	2013-12-27	Ф.Хоффманн-Ля Рош Аг	4-триметиламмониобутираты в качестве ингибиторов срт2
CN111566105A (zh)	2018-01-08	2020-08-21	豪夫迈·罗氏有限公司	作为MAGL抑制剂的八氢吡啶并[1,2-α]吡嗪类化合物
CA3190277A1 (en) *	2020-09-03	2022-03-10	Joerg Benz	Heterocyclic compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4076717A (en) *	1971-12-15	1978-02-28	G. D. Searle & Co.	Derivatives of 1-(3-cyano-3,3-diphenylpropyl)-4-phenylpiperidine-4-carboxylic acid
US3931197A (en) *	1974-02-08	1976-01-06	Richardson-Merrell Inc.	Substituted piperidine derivatives
US4650874A (en) *	1984-11-26	1987-03-17	G. D. Searle & Co.	N-(aralkoxybenzyl)-4(benzhydryl) piperidines

1985
- 1985-10-07 US US06/785,113 patent/US4632925A/en not_active Expired - Fee Related
1986
- 1986-09-26 ZA ZA867375A patent/ZA867375B/xx unknown
- 1986-10-03 HU HU864167A patent/HU196200B/hu not_active IP Right Cessation
- 1986-10-03 NZ NZ217798A patent/NZ217798A/xx unknown
- 1986-10-03 CA CA000519718A patent/CA1281326C/en not_active Expired - Lifetime
- 1986-10-03 DK DK475286A patent/DK168291B1/da active
- 1986-10-03 IL IL80232A patent/IL80232A0/xx not_active IP Right Cessation
- 1986-10-03 AU AU63501/86A patent/AU593844B2/en not_active Ceased
- 1986-10-06 DE DE8686113837T patent/DE3672134D1/de not_active Expired - Lifetime
- 1986-10-06 AT AT86113837T patent/ATE53997T1/de not_active IP Right Cessation
- 1986-10-06 JP JP61236364A patent/JPH0633254B2/ja not_active Expired - Lifetime
- 1986-10-06 PT PT83495A patent/PT83495B/pt not_active IP Right Cessation
- 1986-10-06 MC MC861851A patent/MC1769A1/fr unknown
- 1986-10-06 ES ES8602424A patent/ES2005074A6/es not_active Expired
- 1986-10-06 EP EP86113837A patent/EP0221376B1/de not_active Expired - Lifetime
- 1986-10-06 NO NO863978A patent/NO166127C/no unknown
- 1986-10-06 IE IE263686A patent/IE59434B1/en not_active IP Right Cessation
- 1986-10-07 KR KR1019860008388A patent/KR870003984A/ko not_active Ceased
- 1986-10-07 GR GR862513A patent/GR862513B/el unknown
- 1986-10-07 FI FI864051A patent/FI85020C/fi not_active IP Right Cessation
- 1986-10-07 PH PH34329A patent/PH24167A/en unknown
- 1986-10-23 AR AR86305473A patent/AR241422A1/es active
1993
- 1993-02-17 SG SG175/93A patent/SG17593G/en unknown

Also Published As

Publication number	Publication date
EP0221376B1 (de)	1990-06-20
PH24167A (en)	1990-03-22
DK475286D0 (da)	1986-10-03
AR241422A1 (es)	1992-07-31
IL80232A0 (en)	1987-01-30
JPS6287585A (ja)	1987-04-22
EP0221376A2 (de)	1987-05-13
PT83495A (en)	1986-11-01
SG17593G (en)	1993-05-21
NO863978D0 (no)	1986-10-06
FI85020C (fi)	1992-02-25
JPH0633254B2 (ja)	1994-05-02
DK168291B1 (da)	1994-03-07
US4632925A (en)	1986-12-30
ATE53997T1 (de)	1990-07-15
DE3672134D1 (de)	1990-07-26
EP0221376A3 (en)	1987-09-02
PT83495B (pt)	1989-05-31
FI85020B (fi)	1991-11-15
AU593844B2 (en)	1990-02-22
IE59434B1 (en)	1994-02-23
ZA867375B (en)	1987-05-27
NO166127B (no)	1991-02-25
IE862636L (en)	1987-04-07
CA1281326C (en)	1991-03-12
NZ217798A (en)	1989-10-27
AU6350186A (en)	1987-04-09
MC1769A1 (fr)	1987-07-17
ES2005074A6 (es)	1989-03-01
NO863978L (no)	1987-04-08
FI864051A0 (fi)	1986-10-07
DK475286A (da)	1987-04-08
HUT41768A (en)	1987-05-28
KR870003984A (ko)	1987-05-06
NO166127C (no)	1991-06-05
HU196200B (en)	1988-10-28
GR862513B (en)	1987-02-09

Publication	Publication Date	Title
FI852073L (fi)	1986-11-24	Andningsbehandlingsapparat.
FI860542A7 (fi)	1986-08-08	Foerkopplingsanordning foer hoegtrycksurladdningslampor speciellt foer natriumaonglampor.
FI860285L (fi)	1986-08-08	6-tioxantinderivat.
FI865074L (fi)	1987-06-14	Folieelement foer elektrisk uppvaermning.
FI862399A7 (fi)	1986-12-08	Antibakteriskt verkande kinolonkarboxylsyraestrar.
FI864051A0 (fi)	1986-10-07	N-substituerade difenylpiperidiner.
FI851763L (fi)	1986-11-04	Hydrauliskt klassifiseringsfoerfarande och -anordning.
FI865092A0 (fi)	1986-12-15	Avbrytningskrest foer gitterbryttyristor.
FI851079A0 (fi)	1985-03-19	Kausticeringsfoerfarande.
FI864374A0 (fi)	1986-10-28	Brotsch.
FI851027L (fi)	1986-09-15	Kalciumsulfatuppslamning.
FI850220L (fi)	1986-07-18	Skivpress.
FI851829L (fi)	1986-11-09	Varmluftsutvecklare.
FI851052L (fi)	1986-09-16	Noskapinsalt.
FI73492B (fi)	1987-06-30	Fasadplatta.
FI850177A0 (fi)	1985-01-15	Vaermesystem.
FI851878A0 (fi)	1985-05-13	Hammare.
ES286448Y (es)	1986-07-01	Tapon-dosificador.
FI850395A0 (fi)	1985-01-30	Lysroersarmatur.
FI850548A0 (fi)	1985-02-08	Anordning avsedd foer dragutraetningsbommar foer bilkaross.
FI850444A0 (fi)	1985-02-01	Slitstarkt foeremaol.
FI850494A0 (fi)	1985-02-06	Foertoejningslina.
NO871412D0 (no)	1987-04-03	Overvaakningsanlegg.
FI852175A0 (fi)	1985-05-30	Gallerrenare.
FI850312A0 (fi)	1985-01-24	Kombinerad rotationstryckmaskin.

Legal Events

Date	Code	Title	Description
1995-05-15	MM	Patent lapsed
2004-08-31	MM	Patent lapsed	Owner name: F. HOFFMANN-LA ROCHE AG