ZA983046B - 4-Halogenated steroids their preparation process and intermediates their use as medicaments and the pharmaceutical compositions containing them - Google Patents

4-Halogenated steroids their preparation process and intermediates their use as medicaments and the pharmaceutical compositions containing them

Info

Publication number: ZA983046B
Authority: ZA; South Africa
Prior art keywords: medicaments; intermediates; pharmaceutical compositions; preparation process; compositions containing
Prior art date: 1997-04-09

Application number

ZA983046A

Other languages

English (en)

Inventor

Yamina Bouali

Francois Nique

Jean-Georges Teutsch

Patrick Van De Velde

Original Assignee

Hoechst Marion Roussel Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-04-09

Filing date

1998-04-09

Publication date

1999-04-09

1998-04-09 Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc

1999-04-09 Publication of ZA983046B publication Critical patent/ZA983046B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
- C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Physical Education & Sports Medicine (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Cardiology (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Heart & Thoracic Surgery (AREA)
Dermatology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

ZA983046A 1997-04-09 1998-04-09 4-Halogenated steroids their preparation process and intermediates their use as medicaments and the pharmaceutical compositions containing them ZA983046B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9704321A FR2761992B1 (fr)	1997-04-09	1997-04-09	Nouveaux steroides 4-halogenes, leur procede et intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant

Publications (1)

Publication Number	Publication Date
ZA983046B true ZA983046B (en)	1999-04-09

Family

ID=9505672

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA983046A ZA983046B (en)	1997-04-09	1998-04-09	4-Halogenated steroids their preparation process and intermediates their use as medicaments and the pharmaceutical compositions containing them

Country Status (31)

Country	Link
US (5)	US6239121B1 (xx)
EP (1)	EP0973793B1 (xx)
JP (1)	JP4347420B2 (xx)
KR (1)	KR20010006149A (xx)
CN (1)	CN1259956A (xx)
AP (1)	AP1137A (xx)
AR (1)	AR012377A1 (xx)
AT (1)	ATE220408T1 (xx)
AU (1)	AU750030B2 (xx)
BR (1)	BR9809578A (xx)
CA (1)	CA2285679A1 (xx)
DE (1)	DE69806473T2 (xx)
DK (1)	DK0973793T3 (xx)
EA (1)	EA002116B1 (xx)
ES (1)	ES2178208T3 (xx)
FR (1)	FR2761992B1 (xx)
HR (1)	HRP980196B1 (xx)
HU (1)	HUP0002457A3 (xx)
ID (1)	ID22930A (xx)
IL (1)	IL132202A (xx)
NO (1)	NO315049B1 (xx)
NZ (1)	NZ337947A (xx)
PL (1)	PL190629B1 (xx)
PT (1)	PT973793E (xx)
SK (1)	SK284480B6 (xx)
TR (1)	TR199902507T2 (xx)
TW (1)	TW505621B (xx)
UA (1)	UA57073C2 (xx)
WO (1)	WO1998045316A1 (xx)
YU (1)	YU51199A (xx)
ZA (1)	ZA983046B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2757519B1 (fr) *	1996-12-23	1999-06-11	Hoechst Marion Roussel Inc	Steroides substitues en position 11, leur procede de preparation, leur application comme medicament et les compositions pharmaceutiques les renfermant
FR2780060B1 (fr) *	1998-06-23	2000-08-04	Hoechst Marion Roussel Inc	Nouveaux 19-nor steroides 17-halogenes, procede et intermediaires de preparation, application comme medicaments et compositions pharmaceutiques les renfermant
FR2826004B1 (fr) *	2001-06-13	2008-03-28	Aventis Pharma Sa	Procede de preparation de derives estrogenes
FR2854402B1 (fr) *	2003-04-29	2008-07-04	Aventis Pharma Sa	Nouveau procede et intermediaires de preparation de composes 19-nor-steroides
EP2125827B1 (en) *	2006-12-29	2010-11-03	F. Hoffmann-La Roche AG	Azaspiro derivatives
US20120046461A1 (en) *	2009-01-23	2012-02-23	Northeastern University	Steroidal anti-hormone hybrids
FR2942409B1 (fr) *	2009-02-20	2013-07-26	Natacha Voillot	Composition pharmaceutique pour la prevention des avortements a repetition.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2640977A2 (en) *	1982-06-11	1990-06-29	Roussel Uclaf	New position-11 substituted 19-norsteroids and their application as medicinal products.
US4676932A (en) *	1984-04-09	1987-06-30	The University Of New Mexico	Synthesis of 1-haloestradiols
US4859585A (en) *	1986-04-17	1989-08-22	Trustees Of Tufts College	In-vitro methods for identifying compositions which are agonists and antagonists of estrogens

1997
- 1997-04-09 FR FR9704321A patent/FR2761992B1/fr not_active Expired - Fee Related
1998
- 1998-04-01 TW TW087104892A patent/TW505621B/zh not_active IP Right Cessation
- 1998-04-08 SK SK1362-99A patent/SK284480B6/sk unknown
- 1998-04-08 AP APAP/P/1999/001656A patent/AP1137A/en active
- 1998-04-08 NZ NZ337947A patent/NZ337947A/en unknown
- 1998-04-08 CN CN98805963A patent/CN1259956A/zh active Pending
- 1998-04-08 CA CA002285679A patent/CA2285679A1/fr not_active Abandoned
- 1998-04-08 EA EA199900909A patent/EA002116B1/ru not_active IP Right Cessation
- 1998-04-08 AT AT98920587T patent/ATE220408T1/de not_active IP Right Cessation
- 1998-04-08 KR KR1019997009228A patent/KR20010006149A/ko not_active Ceased
- 1998-04-08 HU HU0002457A patent/HUP0002457A3/hu unknown
- 1998-04-08 AR ARP980101631A patent/AR012377A1/es active IP Right Grant
- 1998-04-08 TR TR1999/02507T patent/TR199902507T2/xx unknown
- 1998-04-08 ES ES98920587T patent/ES2178208T3/es not_active Expired - Lifetime
- 1998-04-08 DK DK98920587T patent/DK0973793T3/da active
- 1998-04-08 WO PCT/FR1998/000709 patent/WO1998045316A1/fr not_active Ceased
- 1998-04-08 US US09/402,705 patent/US6239121B1/en not_active Expired - Lifetime
- 1998-04-08 HR HR980196A patent/HRP980196B1/xx not_active IP Right Cessation
- 1998-04-08 EP EP98920587A patent/EP0973793B1/fr not_active Expired - Lifetime
- 1998-04-08 DE DE69806473T patent/DE69806473T2/de not_active Expired - Lifetime
- 1998-04-08 JP JP54246298A patent/JP4347420B2/ja not_active Expired - Fee Related
- 1998-04-08 YU YU51199A patent/YU51199A/sh unknown
- 1998-04-08 PT PT98920587T patent/PT973793E/pt unknown
- 1998-04-08 AU AU73396/98A patent/AU750030B2/en not_active Ceased
- 1998-04-08 ID IDW991174A patent/ID22930A/id unknown
- 1998-04-08 BR BR9809578-1A patent/BR9809578A/pt not_active IP Right Cessation
- 1998-04-08 PL PL98336116A patent/PL190629B1/pl unknown
- 1998-04-08 IL IL13220298A patent/IL132202A/en active IP Right Grant
- 1998-04-09 ZA ZA983046A patent/ZA983046B/xx unknown
- 1998-08-04 UA UA99116107A patent/UA57073C2/uk unknown
1999
- 1999-10-08 NO NO19994908A patent/NO315049B1/no not_active IP Right Cessation
2000
- 2000-12-08 US US09/733,377 patent/US6472382B2/en not_active Expired - Lifetime
- 2000-12-22 US US09/746,245 patent/US6462211B1/en not_active Expired - Lifetime
2001
- 2001-01-10 US US09/757,678 patent/US20010005756A1/en not_active Abandoned
- 2001-01-10 US US09/757,679 patent/US6399766B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
US6239121B1 (en)	2001-05-29
IL132202A0 (en)	2001-03-19
US6462211B1 (en)	2002-10-08
US20010005756A1 (en)	2001-06-28
US20020040135A1 (en)	2002-04-04
FR2761992A1 (fr)	1998-10-16
NO994908L (no)	1999-12-07
HRP980196B1 (en)	2003-08-31
CA2285679A1 (fr)	1998-10-15
ES2178208T3 (es)	2002-12-16
NO315049B1 (no)	2003-06-30
DK0973793T3 (da)	2002-10-28
EP0973793B1 (fr)	2002-07-10
CN1259956A (zh)	2000-07-12
YU51199A (sh)	2002-09-19
SK284480B6 (sk)	2005-04-01
PT973793E (pt)	2002-11-29
US20010008941A1 (en)	2001-07-19
US6399766B2 (en)	2002-06-04
AP1137A (en)	2003-01-12
ID22930A (id)	1999-12-16
IL132202A (en)	2004-02-19
NZ337947A (en)	2001-04-27
EA002116B1 (ru)	2001-12-24
BR9809578A (pt)	2000-07-04
WO1998045316A1 (fr)	1998-10-15
PL336116A1 (en)	2000-06-05
JP4347420B2 (ja)	2009-10-21
TW505621B (en)	2002-10-11
FR2761992B1 (fr)	1999-06-11
US6472382B2 (en)	2002-10-29
HUP0002457A3 (en)	2002-07-29
TR199902507T2 (xx)	2000-07-21
AU7339698A (en)	1998-10-30
EP0973793A1 (fr)	2000-01-26
KR20010006149A (ko)	2001-01-26
DE69806473T2 (de)	2003-02-13
UA57073C2 (uk)	2003-06-16
US20010039268A1 (en)	2001-11-08
PL190629B1 (pl)	2005-12-30
ATE220408T1 (de)	2002-07-15
JP2001518891A (ja)	2001-10-16
NO994908D0 (no)	1999-10-08
DE69806473D1 (de)	2002-08-14
AR012377A1 (es)	2000-10-18
EA199900909A1 (ru)	2000-04-24
AP9901656A0 (en)	1999-09-30
SK136299A3 (en)	2000-05-16
HUP0002457A1 (hu)	2001-02-28
HRP980196A2 (en)	1998-12-31
AU750030B2 (en)	2002-07-11

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