ZA201002700B - Compounds for inhibiting ksp kinesin activity - Google Patents

Compounds for inhibiting ksp kinesin activity

Info

Publication number: ZA201002700B
Authority: ZA; South Africa
Prior art keywords: compounds; ksp kinesin; kinesin activity; inhibiting ksp; inhibiting
Prior art date: 2007-11-09

Application number

ZA2010/02700A

Inventor

Chaoyang Dai

Umar Faruk Mansoor

Liping Yang

Lalalnthi Dilrukshi Vitharana

Angie R Angeles

Jr Gerald W Shipps

Xiaohua Huang

Cliff C Cheng

Arshad M Siddiqui

Original Assignee

Schering Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-11-09

Filing date

2010-04-16

Publication date

2010-12-29

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40254344&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA201002700(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2010-04-16 Application filed by Schering Corp filed Critical Schering Corp

2010-12-29 Publication of ZA201002700B publication Critical patent/ZA201002700B/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Oncology (AREA)
Rheumatology (AREA)
Heart & Thoracic Surgery (AREA)
Hematology (AREA)
Transplantation (AREA)
Communicable Diseases (AREA)
Pain & Pain Management (AREA)
Cardiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Plural Heterocyclic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

ZA2010/02700A 2007-11-09 2010-04-16 Compounds for inhibiting ksp kinesin activity ZA201002700B (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US98679907P	2007-11-09	2007-11-09
PCT/US2008/080176 WO2009061596A1 (en)	2007-11-09	2008-10-16	Compounds for inhibiting ksp kinesin activity

Publications (1)

Publication Number	Publication Date
ZA201002700B true ZA201002700B (en)	2010-12-29

Family

ID=40254344

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA2010/02700A ZA201002700B (en)	2007-11-09	2010-04-16	Compounds for inhibiting ksp kinesin activity

Country Status (14)

Country	Link
EP (1)	EP2215064A1 (en)
JP (1)	JP2011503076A (en)
KR (1)	KR20100075508A (en)
CN (1)	CN101952255A (en)
AR (1)	AR068889A1 (en)
AU (1)	AU2008325025A1 (en)
CA (1)	CA2702990A1 (en)
CL (1)	CL2008003062A1 (en)
IL (1)	IL205181A0 (en)
MX (1)	MX2010004314A (en)
PE (1)	PE20090968A1 (en)
TW (1)	TW200922559A (en)
WO (1)	WO2009061596A1 (en)
ZA (1)	ZA201002700B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CL2008003063A1 (en) *	2007-10-19	2010-01-04	Schering Corp	Compounds derived from 1,3,4-thiadiazole spiro-condensed, inhibitors of ksp kinesin activity; pharmaceutical composition; and its use in the treatment of proliferative diseases such as cancer, hyperplasia, cardiac hypertrophy, autoimmune diseases, fungal disorders, arthritis, graft rejection, among others.
DE102008001932A1 (en) *	2008-05-21	2009-11-26	Bayer Cropscience Ag	Substituted spiroisoxazolines
TWI683813B (en) *	2014-03-20	2020-02-01	美商卡佩拉醫療公司	Benzimidazole derivatives, and pharmaceutical compositions and methods of use thereof
WO2016057931A1 (en)	2014-10-10	2016-04-14	The Research Foundation For The State University Of New York	Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS5336470B2 (en) *	1971-08-09	1978-10-03
JP4399269B2 (en) *	2002-03-08	2010-01-13	メルクエンドカムパニーインコーポレーテッド	Mitotic kinesin inhibitor
US7449486B2 (en) *	2004-10-19	2008-11-11	Array Biopharma Inc.	Mitotic kinesin inhibitors and methods of use thereof
EP1868601A4 (en) *	2005-04-07	2008-12-10	Merck & Co Inc	INHIBITORS OF MITOTIC KINESIN

2008
- 2008-10-16 KR KR1020107008486A patent/KR20100075508A/en not_active Withdrawn
- 2008-10-16 MX MX2010004314A patent/MX2010004314A/en not_active Application Discontinuation
- 2008-10-16 CA CA2702990A patent/CA2702990A1/en not_active Abandoned
- 2008-10-16 AR ARP080104503A patent/AR068889A1/en not_active Application Discontinuation
- 2008-10-16 CN CN2008801214797A patent/CN101952255A/en active Pending
- 2008-10-16 PE PE2008001777A patent/PE20090968A1/en not_active Application Discontinuation
- 2008-10-16 AU AU2008325025A patent/AU2008325025A1/en not_active Abandoned
- 2008-10-16 WO PCT/US2008/080176 patent/WO2009061596A1/en not_active Ceased
- 2008-10-16 CL CL2008003062A patent/CL2008003062A1/en unknown
- 2008-10-16 JP JP2010533142A patent/JP2011503076A/en active Pending
- 2008-10-16 TW TW097139719A patent/TW200922559A/en unknown
- 2008-10-16 EP EP08847176A patent/EP2215064A1/en not_active Withdrawn
2010
- 2010-04-16 ZA ZA2010/02700A patent/ZA201002700B/en unknown
- 2010-04-18 IL IL205181A patent/IL205181A0/en unknown

Also Published As

Publication number	Publication date
WO2009061596A1 (en)	2009-05-14
EP2215064A1 (en)	2010-08-11
AU2008325025A1 (en)	2009-05-14
AR068889A1 (en)	2009-12-16
TW200922559A (en)	2009-06-01
CN101952255A (en)	2011-01-19
CA2702990A1 (en)	2009-05-14
JP2011503076A (en)	2011-01-27
PE20090968A1 (en)	2009-07-13
KR20100075508A (en)	2010-07-02
CL2008003062A1 (en)	2010-02-19
MX2010004314A (en)	2010-04-30
IL205181A0 (en)	2010-11-30

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IL205184A0 (en)	2010-11-30	Spiro-condensed 1, 3, 4 - thiadiazole derivatives for inhibiting ksp kinesin activity
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