ZA200901462B - Pharmacokinetically improved compounds - Google Patents
Pharmacokinetically improved compoundsInfo
- Publication number
- ZA200901462B ZA200901462B ZA200901462A ZA200901462A ZA200901462B ZA 200901462 B ZA200901462 B ZA 200901462B ZA 200901462 A ZA200901462 A ZA 200901462A ZA 200901462 A ZA200901462 A ZA 200901462A ZA 200901462 B ZA200901462 B ZA 200901462B
- Authority
- ZA
- South Africa
- Prior art keywords
- improved compounds
- pharmacokinetically improved
- pharmacokinetically
- compounds
- improved
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D257/08—Six-membered rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Dentistry (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US84030606P | 2006-08-24 | 2006-08-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200901462B true ZA200901462B (en) | 2010-07-28 |
Family
ID=39107450
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200901462A ZA200901462B (en) | 2006-08-24 | 2007-08-23 | Pharmacokinetically improved compounds |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US20100324037A1 (xx) |
| EP (2) | EP2061322B1 (xx) |
| JP (2) | JP2010501577A (xx) |
| KR (1) | KR20090042863A (xx) |
| CN (1) | CN101528042A (xx) |
| AU (1) | AU2007287024A1 (xx) |
| BR (1) | BRPI0716571A2 (xx) |
| CA (1) | CA2661483A1 (xx) |
| ES (1) | ES2548759T3 (xx) |
| IL (1) | IL197224A0 (xx) |
| MX (1) | MX2009002073A (xx) |
| NO (1) | NO20090896L (xx) |
| TW (1) | TW200826944A (xx) |
| WO (1) | WO2008024494A2 (xx) |
| ZA (1) | ZA200901462B (xx) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CR9465A (es) | 2005-03-25 | 2008-06-19 | Surface Logix Inc | Compuestos mejorados farmacocineticamente |
| JP6338601B2 (ja) * | 2013-03-01 | 2018-06-06 | フンダシオン パラ ラ インベスティガシオン メディカ アプリカダ | ホスホジエステラーゼとヒストンデアセチラーゼの二重阻害剤としての新規な化合物 |
| TW201639851A (zh) * | 2015-03-16 | 2016-11-16 | 大日本住友製藥股份有限公司 | 雙環咪唑衍生物 |
| CN114085225A (zh) * | 2021-06-04 | 2022-02-25 | 广东西捷药业有限公司 | 一种伐地那非类似物及其合成方法和应用 |
| TWI806144B (zh) * | 2021-09-01 | 2023-06-21 | 臺灣塑膠工業股份有限公司 | 纖維預浸布的含浸裝置及其方法 |
| US12258350B1 (en) * | 2024-11-14 | 2025-03-25 | Retension Pharmaceuticals, Inc. | Crystalline forms of 4-ethoxy-n-(2-methoxyethyl)-n-methyl-3-(5-methyl-4-oxo-7-propyl-3,4-dihydroimidazo[5, 1-f][1,2,4]triazin-2-yl)benzenesulfonamide |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4631211A (en) * | 1985-03-25 | 1986-12-23 | Scripps Clinic & Research Foundation | Means for sequential solid phase organic synthesis and methods using the same |
| US5143854A (en) * | 1989-06-07 | 1992-09-01 | Affymax Technologies N.V. | Large scale photolithographic solid phase synthesis of polypeptides and receptor binding screening thereof |
| EP0502060A4 (en) | 1989-11-13 | 1993-05-05 | Affymax Technologies N.V. | Spatially-addressable immobilization of anti-ligands on surfaces |
| DE69132531T2 (de) | 1990-12-06 | 2001-09-13 | Affymetrix, Inc. (N.D.Ges.D.Staates Delaware) | Verbindungen und ihre Verwendung in einer binären Synthesestrategie |
| AU675054B2 (en) | 1991-11-22 | 1997-01-23 | Affymetrix, Inc. | Combinatorial strategies for polymer synthesis |
| US5359115A (en) | 1992-03-26 | 1994-10-25 | Affymax Technologies, N.V. | Methods for the synthesis of phosphonate esters |
| US5573905A (en) | 1992-03-30 | 1996-11-12 | The Scripps Research Institute | Encoded combinatorial chemical libraries |
| JP2857540B2 (ja) | 1992-06-22 | 1999-02-17 | ファナック株式会社 | カッタパスの自動再作成を行うｃａｄ／ｃａｍ方法及び装置 |
| US5288514A (en) * | 1992-09-14 | 1994-02-22 | The Regents Of The University Of California | Solid phase and combinatorial synthesis of benzodiazepine compounds on a solid support |
| CA2143848C (en) | 1992-10-01 | 2007-09-11 | W. Clark Still | Complex combinatorial chemical libraries encoded with tags |
| US5480971A (en) | 1993-06-17 | 1996-01-02 | Houghten Pharmaceuticals, Inc. | Peralkylated oligopeptide mixtures |
| US5440016A (en) | 1993-06-18 | 1995-08-08 | Torrey Pines Institute For Molecular Studies | Peptides of the formula (KFmoc) ZZZ and their uses |
| US5362899A (en) * | 1993-09-09 | 1994-11-08 | Affymax Technologies, N.V. | Chiral synthesis of alpha-aminophosponic acids |
| DK1174431T3 (da) * | 1997-11-12 | 2012-08-20 | Bayer Pharma AG | 2-phenyl-substitueret imidazo triazinon som phoshodiesterase-inhibitorer |
| DE19827640A1 (de) * | 1998-06-20 | 1999-12-23 | Bayer Ag | 7-Alkyl- und Cycloalkyl-substituierte Imidazotriazinone |
| US6451807B1 (en) * | 1999-04-30 | 2002-09-17 | Lilly Icos, Llc. | Methods of treating sexual dysfunction in an individual suffering from a retinal disease, class 1 congestive heart failure, or myocardial infarction using a PDE5 inhibitor |
| MXPA02006240A (es) * | 1999-12-24 | 2003-01-28 | Bayer Ag | Nuevas imidazo[1,3,5,) triazinonas y su uso. |
| US6699665B1 (en) | 2000-11-08 | 2004-03-02 | Surface Logix, Inc. | Multiple array system for integrating bioarrays |
| DE10107639A1 (de) * | 2001-02-15 | 2002-08-22 | Bayer Ag | 2-Alkoxyphenyl-substituierte Imidazotriazinone |
| WO2003012392A2 (en) | 2001-07-27 | 2003-02-13 | Surface Logix, Inc. | Resealable and sealable devices for biochemical assays |
| JP2005509737A (ja) | 2001-08-27 | 2005-04-14 | サーフェイス ロジックス，インコーポレイティド | 単層で被覆された表面への生物学的分子の不動化 |
| DE10162435A1 (de) | 2001-12-19 | 2003-07-17 | Joerg Lahann | Verfahren zur Erzeugung von Oberflächenbeschichtungen, die die Adsorption von Proteinen bzw. die Adhäsion von Bakterien und/oder Zellen vermindern |
| JP2005529927A (ja) * | 2002-05-23 | 2005-10-06 | ファイザー インコーポレイテッド | 新規な組み合わせ |
| DE102004038328A1 (de) * | 2004-08-06 | 2006-03-16 | Bayer Healthcare Ag | Neue Verwendungen von 2-Phenyl-substituierten Imidazotriazinon-Derivaten |
| EP1848437A4 (en) * | 2005-02-18 | 2012-04-25 | Surface Logix Inc | METHOD FOR PRODUCING PHARMACOKINETIC IMPROVED COMPOUNDS WITH FUNCTIONAL RESTORATIONS OR GROUPS AND PHARMACEUTICAL COMPOSITIONS WITH THESE COMPOUNDS |
| CR9465A (es) * | 2005-03-25 | 2008-06-19 | Surface Logix Inc | Compuestos mejorados farmacocineticamente |
-
2007
- 2007-08-23 KR KR1020097005834A patent/KR20090042863A/ko not_active Withdrawn
- 2007-08-23 CN CNA2007800397724A patent/CN101528042A/zh active Pending
- 2007-08-23 CA CA002661483A patent/CA2661483A1/en not_active Abandoned
- 2007-08-23 EP EP07837341.2A patent/EP2061322B1/en active Active
- 2007-08-23 MX MX2009002073A patent/MX2009002073A/es not_active Application Discontinuation
- 2007-08-23 AU AU2007287024A patent/AU2007287024A1/en not_active Abandoned
- 2007-08-23 ES ES07837341.2T patent/ES2548759T3/es active Active
- 2007-08-23 WO PCT/US2007/018784 patent/WO2008024494A2/en not_active Ceased
- 2007-08-23 EP EP13180479.1A patent/EP2705753A1/en not_active Withdrawn
- 2007-08-23 US US12/438,504 patent/US20100324037A1/en not_active Abandoned
- 2007-08-23 BR BRPI0716571-4A patent/BRPI0716571A2/pt not_active IP Right Cessation
- 2007-08-23 JP JP2009525652A patent/JP2010501577A/ja active Pending
- 2007-08-23 ZA ZA200901462A patent/ZA200901462B/xx unknown
- 2007-08-24 TW TW096131544A patent/TW200826944A/zh unknown
-
2009
- 2009-02-24 IL IL197224A patent/IL197224A0/en unknown
- 2009-02-26 NO NO20090896A patent/NO20090896L/no not_active Application Discontinuation
-
2012
- 2012-12-07 US US13/708,420 patent/US8853394B2/en active Active
-
2013
- 2013-10-04 JP JP2013209390A patent/JP2014055136A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| ES2548759T3 (es) | 2015-10-20 |
| MX2009002073A (es) | 2009-05-25 |
| KR20090042863A (ko) | 2009-04-30 |
| WO2008024494A9 (en) | 2009-04-02 |
| EP2705753A1 (en) | 2014-03-12 |
| CA2661483A1 (en) | 2008-02-28 |
| US20130096114A1 (en) | 2013-04-18 |
| CN101528042A (zh) | 2009-09-09 |
| AU2007287024A1 (en) | 2008-02-28 |
| TW200826944A (en) | 2008-07-01 |
| EP2061322A4 (en) | 2011-01-05 |
| JP2014055136A (ja) | 2014-03-27 |
| WO2008024494A2 (en) | 2008-02-28 |
| WO2008024494A3 (en) | 2008-04-10 |
| JP2010501577A (ja) | 2010-01-21 |
| EP2061322A2 (en) | 2009-05-27 |
| IL197224A0 (en) | 2009-12-24 |
| EP2061322B1 (en) | 2015-07-01 |
| BRPI0716571A2 (pt) | 2013-11-05 |
| US8853394B2 (en) | 2014-10-07 |
| NO20090896L (no) | 2009-03-09 |
| US20100324037A1 (en) | 2010-12-23 |
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