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ZA200600579B - Piperazine derivatives and methods of use - Google Patents

Piperazine derivatives and methods of use

Info

Publication number
ZA200600579B
ZA200600579B ZA200600579A ZA200600579A ZA200600579B ZA 200600579 B ZA200600579 B ZA 200600579B ZA 200600579 A ZA200600579 A ZA 200600579A ZA 200600579 A ZA200600579 A ZA 200600579A ZA 200600579 B ZA200600579 B ZA 200600579B
Authority
ZA
South Africa
Prior art keywords
methods
diseases
compounds
processes
treatment
Prior art date
Application number
ZA200600579A
Other languages
English (en)
Inventor
Jian J Chen
Ben C Askew
Biswas Kaustav
Jennifer N Chau
Derin C D'amicio
Harried Scott
Nguyen Thomas
Qian Wenyuan
Zhu Jiawang
Christopher H Fotsch
Han Nianhe
Li Aiwen
Liu Qingyian
Nishimura Nobuko
Nomak Rana
Peterkin Tanya
Riahi Babak
Yang Kevin
Yuan Chester Chenguang
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of ZA200600579B publication Critical patent/ZA200600579B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
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    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
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    • C07D243/08—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D245/00—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07—ORGANIC CHEMISTRY
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    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
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    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Virology (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Toxicology (AREA)
  • Molecular Biology (AREA)
  • Addiction (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Vascular Medicine (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
ZA200600579A 2003-06-20 2006-01-20 Piperazine derivatives and methods of use ZA200600579B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US48030303P 2003-06-20 2003-06-20

Publications (1)

Publication Number Publication Date
ZA200600579B true ZA200600579B (en) 2007-04-25

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Application Number Title Priority Date Filing Date
ZA200600579A ZA200600579B (en) 2003-06-20 2006-01-20 Piperazine derivatives and methods of use

Country Status (18)

Country Link
US (2) US7393852B2 (xx)
EP (1) EP1656355B1 (xx)
JP (1) JP2007516176A (xx)
KR (1) KR20060036399A (xx)
CN (1) CN1849121A (xx)
AT (1) ATE388708T1 (xx)
AU (1) AU2004303757B2 (xx)
BR (1) BRPI0411673A (xx)
CA (1) CA2529314A1 (xx)
DE (1) DE602004012418T2 (xx)
ES (1) ES2302079T3 (xx)
IL (1) IL172419A0 (xx)
IS (1) IS8175A (xx)
MX (1) MXPA05013469A (xx)
NO (1) NO20060278L (xx)
RU (1) RU2006101541A (xx)
WO (1) WO2005061467A2 (xx)
ZA (1) ZA200600579B (xx)

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US20040073617A1 (en) * 2000-06-19 2004-04-15 Milliken Walter Clark Hash-based systems and methods for detecting and preventing transmission of unwanted e-mail
US7328349B2 (en) 2001-12-14 2008-02-05 Bbn Technologies Corp. Hash-based systems and methods for detecting, preventing, and tracing network worms and viruses
US7200105B1 (en) * 2001-01-12 2007-04-03 Bbn Technologies Corp. Systems and methods for point of ingress traceback of a network attack
WO2005061467A2 (en) * 2003-06-20 2005-07-07 Amgen Inc. Piperazine derivatives as bradykinin antagonists
CA2573730A1 (en) * 2004-07-15 2006-02-23 Amgen Inc. 1,2,3,4-tetrahydropyrazin-2-yl acetamides and their use as bradykinin antagonists for the treatment of inflammation related disorders
US20060217362A1 (en) * 2004-12-29 2006-09-28 Tung Jay S Novel compounds useful for bradykinin B1 receptor antagonism
US20060173037A1 (en) * 2005-01-10 2006-08-03 Nathalie Schlienger Aminophenyl derivatives as selective androgen receptor modulators
US8059551B2 (en) * 2005-02-15 2011-11-15 Raytheon Bbn Technologies Corp. Method for source-spoofed IP packet traceback
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US20090054460A1 (en) 2009-02-26
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US20050014749A1 (en) 2005-01-20
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NO20060278L (no) 2006-03-15

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