ZA200606073B - Methods and dosage forms for increasing solubility of drug compositions for controlled delivery - Google Patents

Methods and dosage forms for increasing solubility of drug compositions for controlled delivery Download PDF

Info

Publication number: ZA200606073B
Authority: ZA; South Africa
Prior art keywords: composition; drug; therapeutic agent; surfactant; dosage form
Prior art date: 2003-12-23

Application number

ZA200606073A

Other languages

English (en)

Inventor

Jao Frank

Skluzacek Robert

Edgren David

Yam Noymi

Original Assignee

Alza Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-12-23

Filing date

2006-07-21

Publication date

2008-02-27

2006-07-21 Application filed by Alza Corp filed Critical Alza Corp

2008-02-27 Publication of ZA200606073B publication Critical patent/ZA200606073B/en

Links

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MSRILKIQRXUYCT-UHFFFAOYSA-M valproate semisodium Chemical compound [Na+].CCCC(C(O)=O)CCC.CCCC(C([O-])=O)CCC MSRILKIQRXUYCT-UHFFFAOYSA-M 0.000 description 1
229960000604 valproic acid Drugs 0.000 description 1
235000013311 vegetables Nutrition 0.000 description 1
229960001722 verapamil Drugs 0.000 description 1
229960003048 vinblastine Drugs 0.000 description 1
JXLYSJRDGCGARV-XQKSVPLYSA-N vincaleukoblastine Chemical compound C([C@@H](C[C@]1(C(=O)OC)C=2C(=CC3=C([C@]45[C@H]([C@@]([C@H](OC(C)=O)[C@]6(CC)C=CCN([C@H]56)CC4)(O)C(=O)OC)N3C)C=2)OC)C[C@@](C2)(O)CC)N2CCC2=C1NC1=CC=CC=C21 JXLYSJRDGCGARV-XQKSVPLYSA-N 0.000 description 1
235000019156 vitamin B Nutrition 0.000 description 1
239000011720 vitamin B Substances 0.000 description 1
235000019165 vitamin E Nutrition 0.000 description 1
229940046009 vitamin E Drugs 0.000 description 1
239000011709 vitamin E Substances 0.000 description 1
229960005080 warfarin Drugs 0.000 description 1
PJVWKTKQMONHTI-UHFFFAOYSA-N warfarin Chemical compound OC=1C2=CC=CC=C2OC(=O)C=1C(CC(=O)C)C1=CC=CC=C1 PJVWKTKQMONHTI-UHFFFAOYSA-N 0.000 description 1
230000003442 weekly effect Effects 0.000 description 1
238000009736 wetting Methods 0.000 description 1
239000000080 wetting agent Substances 0.000 description 1
239000000811 xylitol Substances 0.000 description 1
229960002555 zidovudine Drugs 0.000 description 1
HBOMLICNUCNMMY-XLPZGREQSA-N zidovudine Chemical compound O=C1NC(=O)C(C)=CN1[C@@H]1O[C@H](CO)[C@@H](N=[N+]=[N-])C1 HBOMLICNUCNMMY-XLPZGREQSA-N 0.000 description 1
229910052725 zinc Inorganic materials 0.000 description 1
239000011701 zinc Substances 0.000 description 1
239000002076 α-tocopherol Substances 0.000 description 1
235000004835 α-tocopherol Nutrition 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/18—Sulfonamides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7004—Monosaccharides having only carbon, hydrogen and oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Molecular Biology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

ZA200606073A 2003-12-23 2006-07-21 Methods and dosage forms for increasing solubility of drug compositions for controlled delivery ZA200606073B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US53245003P	2003-12-23	2003-12-23

Publications (1)

Publication Number	Publication Date
ZA200606073B true ZA200606073B (en)	2008-02-27

Family

ID=34738800

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200606073A ZA200606073B (en)	2003-12-23	2006-07-21	Methods and dosage forms for increasing solubility of drug compositions for controlled delivery

Country Status (11)

Country	Link
US (1)	US20050169992A1 (fr)
EP (1)	EP1703894A1 (fr)
JP (1)	JP2007516297A (fr)
KR (1)	KR20060123493A (fr)
CN (1)	CN1905856A (fr)
AU (1)	AU2004308973A1 (fr)
CA (1)	CA2550866A1 (fr)
IL (1)	IL176108A0 (fr)
NO (1)	NO20063411L (fr)
WO (1)	WO2005063206A1 (fr)
ZA (1)	ZA200606073B (fr)

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2004
- 2004-12-22 JP JP2006547435A patent/JP2007516297A/ja not_active Withdrawn
- 2004-12-22 AU AU2004308973A patent/AU2004308973A1/en not_active Abandoned
- 2004-12-22 CA CA002550866A patent/CA2550866A1/fr not_active Abandoned
- 2004-12-22 US US11/023,257 patent/US20050169992A1/en not_active Abandoned
- 2004-12-22 CN CNA2004800388651A patent/CN1905856A/zh active Pending
- 2004-12-22 WO PCT/US2004/043525 patent/WO2005063206A1/fr not_active Ceased
- 2004-12-22 KR KR1020067014086A patent/KR20060123493A/ko not_active Withdrawn
- 2004-12-22 EP EP04817055A patent/EP1703894A1/fr not_active Withdrawn
2006
- 2006-06-04 IL IL176108A patent/IL176108A0/en unknown
- 2006-07-21 ZA ZA200606073A patent/ZA200606073B/en unknown
- 2006-07-24 NO NO20063411A patent/NO20063411L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
AU2004308973A1 (en)	2005-07-14
JP2007516297A (ja)	2007-06-21
NO20063411L (no)	2006-09-19
WO2005063206A1 (fr)	2005-07-14
CA2550866A1 (fr)	2005-07-14
US20050169992A1 (en)	2005-08-04
EP1703894A1 (fr)	2006-09-27
CN1905856A (zh)	2007-01-31
KR20060123493A (ko)	2006-12-01
IL176108A0 (en)	2006-10-05

Publication	Publication Date	Title
US20050169992A1 (en)	2005-08-04	Methods and dosage forms for increasing solubility of drug compositions for controlled delivery
US20040091529A1 (en)	2004-05-13	Methods and dosage forms for increasing solubility of drug compositions for controlled delivery
US20040115262A1 (en)	2004-06-17	Formulations and dosage forms for controlled delivery of topiramate
US20050175690A1 (en)	2005-08-11	Novel drug compositions and dosage forms
US20050058707A1 (en)	2005-03-17	Uniform delivery of topiramate over prolonged period of time with enhanced dispersion formulation
US20070243254A1 (en)	2007-10-18	Novel drug compositions and dosage forms of topiramate
US20050136108A1 (en)	2005-06-23	Stepwise delivery of topiramate over prolonged period of time
US20050175697A1 (en)	2005-08-11	Novel drug compositions and dosage forms of topiramate
US20050175696A1 (en)	2005-08-11	Drug granule coatings that impart smear resistance during mechanical compression
AU2004312083A1 (en)	2005-07-21	Drug granule coatings that impart smear resistance during mechanical compression
MXPA06007289A (en)	2007-04-20	Methods and dosage forms for increasing solubility of drug compositions for controlled delivery