ZA200405653B - Tetracyclic heterocompounds as estrogen receptor modulators - Google Patents
Tetracyclic heterocompounds as estrogen receptor modulatorsInfo
- Publication number
- ZA200405653B ZA200405653B ZA200405653A ZA200405653A ZA200405653B ZA 200405653 B ZA200405653 B ZA 200405653B ZA 200405653 A ZA200405653 A ZA 200405653A ZA 200405653 A ZA200405653 A ZA 200405653A ZA 200405653 B ZA200405653 B ZA 200405653B
- Authority
- ZA
- South Africa
- Prior art keywords
- heterocompounds
- tetracyclic
- estrogen receptor
- receptor modulators
- modulators
- Prior art date
Links
- 239000002834 estrogen receptor modulator Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Psychiatry (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pyrane Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US34195701P | 2001-12-19 | 2001-12-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200405653B true ZA200405653B (en) | 2006-06-28 |
Family
ID=23339719
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200405653A ZA200405653B (en) | 2001-12-19 | 2004-07-15 | Tetracyclic heterocompounds as estrogen receptor modulators |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP1467998B1 (xx) |
| JP (1) | JP2005513133A (xx) |
| CN (1) | CN1620457A (xx) |
| AR (1) | AR038661A1 (xx) |
| AT (1) | ATE321764T1 (xx) |
| AU (1) | AU2002362041A1 (xx) |
| BR (1) | BR0215152A (xx) |
| CA (1) | CA2471107A1 (xx) |
| CY (1) | CY1105361T1 (xx) |
| DE (1) | DE60210333T2 (xx) |
| DK (1) | DK1467998T3 (xx) |
| ES (1) | ES2264737T3 (xx) |
| HU (1) | HUP0500103A3 (xx) |
| IL (1) | IL162295A0 (xx) |
| MX (1) | MXPA04006034A (xx) |
| NZ (1) | NZ533281A (xx) |
| PL (1) | PL371045A1 (xx) |
| PT (1) | PT1467998E (xx) |
| RU (1) | RU2305099C2 (xx) |
| WO (1) | WO2003053977A1 (xx) |
| ZA (1) | ZA200405653B (xx) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7105679B2 (en) | 2001-12-19 | 2006-09-12 | Kanojia Ramesh M | Heteroatom containing tetracyclic derivatives as selective estrogen receptor modulators |
| US7329654B2 (en) * | 2001-12-19 | 2008-02-12 | Janssen Pharmaceutica N.V. | Heteroatom containing tetracyclic derivatives as selective estrogen receptor modulators |
| US8614204B2 (en) | 2003-06-06 | 2013-12-24 | Fibrogen, Inc. | Enhanced erythropoiesis and iron metabolism |
| EP1713820A1 (en) * | 2004-01-22 | 2006-10-25 | Eli Lilly And Company | Selective estrogen receptor modulators |
| SI1796664T1 (sl) | 2004-09-20 | 2014-02-28 | Janssen Pharmaceutica N.V. | Novi tetraciklični derivati, ki vsebujejo heteroatome, in so uporabni kot modulatorji receptorja spolnega steoidnega hormona |
| JP5410751B2 (ja) | 2005-06-15 | 2014-02-05 | ファイブローゲン、インコーポレーテッド | がん治療のための化合物および方法 |
| DE102006024032A1 (de) * | 2006-05-23 | 2007-11-29 | Voith Patent Gmbh | Anordnung zur Bandregelung |
| RU2360670C1 (ru) * | 2007-10-03 | 2009-07-10 | Закрытое акционерное общество "Биологические исследования и системы" | Фармацевтическая композиция для местного и наружного применения при климактерических расстройствах на основе сигетина |
| MX2012014431A (es) * | 2010-06-10 | 2013-02-26 | Aragon Pharmaceuticals Inc | Modulares del receptor de estrogenos y usos de los mismos. |
| MX357496B (es) * | 2011-12-14 | 2018-07-11 | Seragon Pharmaceuticals Inc | Moduladores del receptor de estrógenos fluorados y sus usos. |
| CN113135884B (zh) * | 2020-01-20 | 2023-03-10 | 西华大学 | 一种异色烯类化合物及其制备方法和用途 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL124481C (xx) * | 1964-11-04 | |||
| SU1607348A1 (ru) * | 1989-03-02 | 1994-09-30 | Пятигорский фармацевтический институт | 7-(3-фенилпропеноилокси)- 4' -фторизофлавон, обладающий гипотензивным действием |
| CA2214196A1 (en) * | 1996-09-26 | 1998-03-26 | Eli Lilly And Company | Benzo[b]indeno[2,1-d]thiophene compounds, intermediates, processes, compositions and methods |
| CN1120162C (zh) * | 1996-12-13 | 2003-09-03 | 中外制药株式会社 | 新的苯并吡喃衍生物 |
| RU2138669C1 (ru) * | 1997-07-02 | 1999-09-27 | Гнедых Александр Михайлович | Воздушный ракетный двигатель |
-
2002
- 2002-12-02 AT AT02797167T patent/ATE321764T1/de not_active IP Right Cessation
- 2002-12-02 IL IL16229502A patent/IL162295A0/xx unknown
- 2002-12-02 HU HU0500103A patent/HUP0500103A3/hu unknown
- 2002-12-02 PL PL02371045A patent/PL371045A1/xx not_active Application Discontinuation
- 2002-12-02 JP JP2003554693A patent/JP2005513133A/ja not_active Withdrawn
- 2002-12-02 CN CNA028281446A patent/CN1620457A/zh active Pending
- 2002-12-02 WO PCT/US2002/038486 patent/WO2003053977A1/en not_active Ceased
- 2002-12-02 EP EP02797167A patent/EP1467998B1/en not_active Expired - Lifetime
- 2002-12-02 RU RU2004118606/04A patent/RU2305099C2/ru not_active IP Right Cessation
- 2002-12-02 ES ES02797167T patent/ES2264737T3/es not_active Expired - Lifetime
- 2002-12-02 AU AU2002362041A patent/AU2002362041A1/en not_active Abandoned
- 2002-12-02 PT PT02797167T patent/PT1467998E/pt unknown
- 2002-12-02 NZ NZ533281A patent/NZ533281A/en unknown
- 2002-12-02 CA CA002471107A patent/CA2471107A1/en not_active Abandoned
- 2002-12-02 DK DK02797167T patent/DK1467998T3/da active
- 2002-12-02 BR BR0215152-9A patent/BR0215152A/pt not_active IP Right Cessation
- 2002-12-02 MX MXPA04006034A patent/MXPA04006034A/es active IP Right Grant
- 2002-12-02 DE DE60210333T patent/DE60210333T2/de not_active Expired - Fee Related
- 2002-12-18 AR ARP020104957A patent/AR038661A1/es unknown
-
2004
- 2004-07-15 ZA ZA200405653A patent/ZA200405653B/xx unknown
-
2006
- 2006-06-08 CY CY20061100768T patent/CY1105361T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1467998A1 (en) | 2004-10-20 |
| WO2003053977A1 (en) | 2003-07-03 |
| HUP0500103A2 (hu) | 2005-05-30 |
| CA2471107A1 (en) | 2003-07-03 |
| DE60210333D1 (de) | 2006-05-18 |
| HK1068875A1 (en) | 2005-05-06 |
| DE60210333T2 (de) | 2006-11-30 |
| ATE321764T1 (de) | 2006-04-15 |
| PL371045A1 (en) | 2005-06-13 |
| NZ533281A (en) | 2007-05-31 |
| HUP0500103A3 (en) | 2009-01-28 |
| MXPA04006034A (es) | 2005-03-31 |
| AU2002362041A1 (en) | 2003-07-09 |
| ES2264737T3 (es) | 2007-01-16 |
| CY1105361T1 (el) | 2010-03-03 |
| DK1467998T3 (da) | 2006-07-31 |
| CN1620457A (zh) | 2005-05-25 |
| BR0215152A (pt) | 2004-10-19 |
| IL162295A0 (en) | 2005-11-20 |
| PT1467998E (pt) | 2006-08-31 |
| JP2005513133A (ja) | 2005-05-12 |
| RU2004118606A (ru) | 2006-01-10 |
| EP1467998B1 (en) | 2006-03-29 |
| RU2305099C2 (ru) | 2007-08-27 |
| AR038661A1 (es) | 2005-01-26 |
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