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ZA200306727B - Aryl and biaryl compounds having MCH modulatory activity. - Google Patents

Aryl and biaryl compounds having MCH modulatory activity. Download PDF

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Publication number
ZA200306727B
ZA200306727B ZA200306727A ZA200306727A ZA200306727B ZA 200306727 B ZA200306727 B ZA 200306727B ZA 200306727 A ZA200306727 A ZA 200306727A ZA 200306727 A ZA200306727 A ZA 200306727A ZA 200306727 B ZA200306727 B ZA 200306727B
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South Africa
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compound
composition
group
prodrug
pharmaceutically acceptable
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ZA200306727A
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English (en)
Inventor
Douglas W Hobbs
Rachael C Hunter
Tao Guo
Huizhong Gu
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Pharmacopeia Drug Discovery
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Publication of ZA200306727B publication Critical patent/ZA200306727B/en

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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
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    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
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    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
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    • C—CHEMISTRY; METALLURGY
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CA2441235C (fr) 2011-05-24
US7034056B2 (en) 2006-04-25
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MXPA03008484A (es) 2003-12-08
CN1498205A (zh) 2004-05-19
HUP0400252A2 (hu) 2004-08-30
US20030092715A1 (en) 2003-05-15
WO2002076929A1 (fr) 2002-10-03
HUP0400252A3 (en) 2011-09-28
NZ527680A (en) 2005-07-29
CA2441235A1 (fr) 2002-10-03
JP2004526736A (ja) 2004-09-02
KR20030093257A (ko) 2003-12-06
EP1370520A1 (fr) 2003-12-17
CN100537527C (zh) 2009-09-09
IL157456A0 (en) 2004-03-28

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