YU46418B - PROCEDURE FOR PREPARATION OF THE PHARMACEUTICAL PREPARATION METOPROLOL WITH CONTROLLED RELEASE - Google Patents
PROCEDURE FOR PREPARATION OF THE PHARMACEUTICAL PREPARATION METOPROLOL WITH CONTROLLED RELEASEInfo
- Publication number
- YU46418B YU46418B YU33987A YU33987A YU46418B YU 46418 B YU46418 B YU 46418B YU 33987 A YU33987 A YU 33987A YU 33987 A YU33987 A YU 33987A YU 46418 B YU46418 B YU 46418B
- Authority
- YU
- Yugoslavia
- Prior art keywords
- preparation
- controlled release
- metoprolol
- procedure
- pharmaceutical preparation
- Prior art date
Links
- 238000013270 controlled release Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000000825 pharmaceutical preparation Substances 0.000 title abstract 2
- IUBSYMUCCVWXPE-UHFFFAOYSA-N metoprolol Chemical compound COCCC1=CC=C(OCC(O)CNC(C)C)C=C1 IUBSYMUCCVWXPE-UHFFFAOYSA-N 0.000 title 1
- 229960002237 metoprolol Drugs 0.000 title 1
- 239000012528 membrane Substances 0.000 abstract 2
- 239000001856 Ethyl cellulose Substances 0.000 abstract 1
- ZZSNKZQZMQGXPY-UHFFFAOYSA-N Ethyl cellulose Chemical compound CCOCC1OC(OC)C(OCC)C(OCC)C1OC1C(O)C(O)C(OC)C(CO)O1 ZZSNKZQZMQGXPY-UHFFFAOYSA-N 0.000 abstract 1
- 239000001913 cellulose Substances 0.000 abstract 1
- 229920002678 cellulose Polymers 0.000 abstract 1
- 230000001419 dependent effect Effects 0.000 abstract 1
- 229920001249 ethyl cellulose Polymers 0.000 abstract 1
- 235000019325 ethyl cellulose Nutrition 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Abstract
POSTUPAK ZA DOBIVANJE FARMACEUTSKOG PREPARATA METOPROLOLA SA KONTROLISANIM OSLOBADJANJEM, naznačen time, što se mnoštvo čestica koji obuhvataju kao glavnu rastvornu komponentu najmanje 95 m/m% soli metoprolola sa rastvorljivošću ispod 600 mg/ml u vodi na 25В° C, prskanjem prevlači rastvorom koji obrazuje membranu, gradeći polimernu membranu koja sadrži derivate celuloze, prvenstveno etil celuloze, tako da se dobija proizvod sa oslobadjanjem aktivne komponente brzinom od 3-7 m/m%/h. Prijava sadrži još 12 zavisnih zahteva.PROCESS FOR THE PREPARATION OF A CONTROLLED RELEASE PHARMACEUTICAL PREPARATION METHOPROLOL membrane, building a polymeric membrane containing cellulose derivatives, preferably ethyl cellulose, so as to obtain a product with the release of the active component at a rate of 3-7 m / m% / h. The application contains 12 more dependent requests.
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| YU33987A YU46418B (en) | 1987-03-04 | 1987-03-04 | PROCEDURE FOR PREPARATION OF THE PHARMACEUTICAL PREPARATION METOPROLOL WITH CONTROLLED RELEASE |
| SI8710339A SI8710339A8 (en) | 1987-03-04 | 1987-03-04 | Process for obtaining pharmaceutical composition of metoprolol with controlled release |
| HR920590 HRP920590B1 (en) | 1987-03-04 | 1992-09-29 | New pharmaceutical preparation |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| YU33987A YU46418B (en) | 1987-03-04 | 1987-03-04 | PROCEDURE FOR PREPARATION OF THE PHARMACEUTICAL PREPARATION METOPROLOL WITH CONTROLLED RELEASE |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| YU33987A YU33987A (en) | 1988-12-31 |
| YU46418B true YU46418B (en) | 1993-10-20 |
Family
ID=25549458
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU33987A YU46418B (en) | 1987-03-04 | 1987-03-04 | PROCEDURE FOR PREPARATION OF THE PHARMACEUTICAL PREPARATION METOPROLOL WITH CONTROLLED RELEASE |
Country Status (2)
| Country | Link |
|---|---|
| SI (1) | SI8710339A8 (en) |
| YU (1) | YU46418B (en) |
-
1987
- 1987-03-04 YU YU33987A patent/YU46418B/en unknown
- 1987-03-04 SI SI8710339A patent/SI8710339A8/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| SI8710339A8 (en) | 1996-08-31 |
| YU33987A (en) | 1988-12-31 |
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