YU38200A - Antagonisti integrinskog receptora - Google Patents
Antagonisti integrinskog receptoraInfo
- Publication number
- YU38200A YU38200A YU38200A YU38200A YU38200A YU 38200 A YU38200 A YU 38200A YU 38200 A YU38200 A YU 38200A YU 38200 A YU38200 A YU 38200A YU 38200 A YU38200 A YU 38200A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- receptor antagonists
- integrin receptor
- compounds
- present
- antagonists
- Prior art date
Links
- 229940127449 Integrin Receptor Antagonists Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 201000001320 Atherosclerosis Diseases 0.000 abstract 1
- 208000006386 Bone Resorption Diseases 0.000 abstract 1
- 206010012689 Diabetic retinopathy Diseases 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 206010027476 Metastases Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 230000033115 angiogenesis Effects 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 230000024279 bone resorption Effects 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 102000006495 integrins Human genes 0.000 abstract 1
- 108010044426 integrins Proteins 0.000 abstract 1
- 208000002780 macular degeneration Diseases 0.000 abstract 1
- 230000009401 metastasis Effects 0.000 abstract 1
- 208000037803 restenosis Diseases 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
- 230000004614 tumor growth Effects 0.000 abstract 1
- 230000002792 vascular Effects 0.000 abstract 1
- 230000003612 virological effect Effects 0.000 abstract 1
- 230000029663 wound healing Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Predmetni pronalazak se odnosi na jedinjenja i njihove derivate, njihovu sintezu i korišćenje, kao antagonista integrinskog receptora. Preciznije, jedinjenja predmetnog pronalaska su antagonisti integrinskih receptora ανГџ3, ανГџ5, i/ili ανГџ6 i upotrebljavaju se za sprečavanje resorpcije kostiju, lečenje i prevenciju osteoporoze i sprečavanje vaskularne restenoze, dijabetične retinopatije, makularne degeneracije, angiogeneze, ateroskleroze, zapaljenja, zarastanja rana, virusnih oboljenja, rasta tumora, i metastaza.[The present invention relates to compounds and derivatives thereof, their synthesis, and their use as integrin receptor antagonists. More particularly, the compounds of the present invention are antagonists of the integrin receptors ανГџ3, ανГџ5, and/or ανГџ6 and are useful for inhibiting bone resorption, treating and preventing osteoporosis, and inhibiting vascular restenosis, diabetic retinopathy, macular degeneration, angiogenesis, atherosclerosis, inflammation, wound healing, viral disease, tumor growth, and metastasis.
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6989997P | 1997-12-17 | 1997-12-17 | |
| GBGB9807382.8A GB9807382D0 (en) | 1998-04-06 | 1998-04-06 | Vitronectin receptor antagonists |
| US8320998P | 1998-04-27 | 1998-04-27 | |
| GBGB9811295.6A GB9811295D0 (en) | 1998-05-26 | 1998-05-26 | Vitronectin receptor antagonists |
| US9262298P | 1998-07-13 | 1998-07-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| YU38200A true YU38200A (sh) | 2003-12-31 |
Family
ID=45477327
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU38200A YU38200A (sh) | 1997-12-17 | 1998-12-14 | Antagonisti integrinskog receptora |
Country Status (1)
| Country | Link |
|---|---|
| YU (1) | YU38200A (sh) |
-
1998
- 1998-12-14 YU YU38200A patent/YU38200A/sh unknown
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