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WO2025035020A3 - Diluted carfilzomib for use in treating multiple myeloma - Google Patents

Diluted carfilzomib for use in treating multiple myeloma Download PDF

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Publication number
WO2025035020A3
WO2025035020A3 PCT/US2024/041550 US2024041550W WO2025035020A3 WO 2025035020 A3 WO2025035020 A3 WO 2025035020A3 US 2024041550 W US2024041550 W US 2024041550W WO 2025035020 A3 WO2025035020 A3 WO 2025035020A3
Authority
WO
WIPO (PCT)
Prior art keywords
carfilzomib
patient
multiple myeloma
treating multiple
diluted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
PCT/US2024/041550
Other languages
French (fr)
Other versions
WO2025035020A2 (en
Inventor
Jeanine BUSSIERE
William J. CALLAHAN III
Rahul Rajan KAUSHIK
Alona TERAN
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Amgen Inc
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of WO2025035020A2 publication Critical patent/WO2025035020A2/en
Publication of WO2025035020A3 publication Critical patent/WO2025035020A3/en
Pending legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/07Tetrapeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Provided herein are methods for treating a disease or condition selected from the group consisting of cancer, autoimmune disease, graft or transplant-related condition, neurodegenerative disease, fibrotic-associated condition, ischemic-related conditions, infection (viral, parasitic or prokaryotic) and diseases associated with bone loss, the method comprising administering to a patient a therapeutically effective amount of carfilzomib or a pharmaceutically acceptable salt thereof at a dose volume of 10 mL/kg or higher. Also provided herein are methods for treating multiple myeloma in a patient, comprising administering to the patient a pharmaceutical composition comprising carfilzomib or a pharmaceutically acceptable salt thereof and an aqueous carrier, wherein the carfilzomib is administered at a dose volume of 2.5 mL/kg or higher and/or at a concentration of less than 2 mg/mL.
PCT/US2024/041550 2023-08-09 2024-08-08 Methods of using carfilzomib Pending WO2025035020A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US202363518343P 2023-08-09 2023-08-09
US63/518,343 2023-08-09

Publications (2)

Publication Number Publication Date
WO2025035020A2 WO2025035020A2 (en) 2025-02-13
WO2025035020A3 true WO2025035020A3 (en) 2025-03-20

Family

ID=92582818

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2024/041550 Pending WO2025035020A2 (en) 2023-08-09 2024-08-08 Methods of using carfilzomib

Country Status (1)

Country Link
WO (1) WO2025035020A2 (en)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017205392A1 (en) * 2016-05-24 2017-11-30 Amgen Inc. Pegylated carfilzomib compounds
WO2018138556A1 (en) * 2017-01-24 2018-08-02 Orbicular Pharmaceutical Technologies Pvt. Ltd. Non-aqueous carfilzomib compositions

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7232818B2 (en) 2004-04-15 2007-06-19 Proteolix, Inc. Compounds for enzyme inhibition
ES2408216T3 (en) 2004-12-07 2013-06-19 Onyx Therapeutics, Inc. Composition for proteasome inhibition
MX2010003732A (en) 2007-10-04 2010-08-09 Onyx Therapeutics Inc Crystalline peptide epoxy ketone protease inhibitors and the synthesis of amino acid keto-epoxides.
PE20120059A1 (en) 2008-10-21 2012-02-27 Onyx Therapeutics Inc PHARMACEUTICAL COMBINATIONS WITH PEPTIDIC EPOXYCETONES
BR112012028726B1 (en) 2012-05-08 2021-07-13 Onyx Therapeutics, Inc. METHOD FOR PREPARING A LOW CHLORIDE PHARMACEUTICAL COMPOSITION
US9309283B2 (en) 2012-07-09 2016-04-12 Onyx Therapeutics, Inc. Prodrugs of peptide epoxy ketone protease inhibitors
US10022326B2 (en) 2012-07-18 2018-07-17 Onyx Therapeutics, Inc. Liposomal compositions of epoxyketone-based proteasome inhibitors
DE102013104003B3 (en) 2013-04-19 2014-03-13 Glatt Systemtechnik Gmbh Device for introducing a defined amount of a second powder into a process container

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017205392A1 (en) * 2016-05-24 2017-11-30 Amgen Inc. Pegylated carfilzomib compounds
WO2018138556A1 (en) * 2017-01-24 2018-08-02 Orbicular Pharmaceutical Technologies Pvt. Ltd. Non-aqueous carfilzomib compositions

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
BRINGHEN SARA ET AL: "Once-weekly versus twice-weekly carfilzomib in patients with newly diagnosed multiple myeloma: a pooled analysis of two phase I/II studies", HAEMATOLOGICA, vol. 104, no. 8, 1 August 2019 (2019-08-01), pages 1640 - 1647, XP093222355, ISSN: 0390-6078, Retrieved from the Internet <URL:https://pmc.ncbi.nlm.nih.gov/articles/PMC6669142/pdf/1041640.pdf> DOI: 10.3324/haematol.2018.208272 *

Also Published As

Publication number Publication date
WO2025035020A2 (en) 2025-02-13

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