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WO2013190569A3 - Novel salts of sunitinib and preparation thereof - Google Patents

Novel salts of sunitinib and preparation thereof Download PDF

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Publication number
WO2013190569A3
WO2013190569A3 PCT/IN2013/000374 IN2013000374W WO2013190569A3 WO 2013190569 A3 WO2013190569 A3 WO 2013190569A3 IN 2013000374 W IN2013000374 W IN 2013000374W WO 2013190569 A3 WO2013190569 A3 WO 2013190569A3
Authority
WO
WIPO (PCT)
Prior art keywords
sunitinib
preparation
novel salts
salts
novel
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/IN2013/000374
Other languages
French (fr)
Other versions
WO2013190569A2 (en
Inventor
Rampalli SRIRAM
Upalla LAVKUMAR
Seshagiri VIJAYA MURALI MOHANRAO
Akshaykant CHATURVEDI
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shilpa Medicare Ltd
Original Assignee
Shilpa Medicare Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shilpa Medicare Ltd filed Critical Shilpa Medicare Ltd
Publication of WO2013190569A2 publication Critical patent/WO2013190569A2/en
Publication of WO2013190569A3 publication Critical patent/WO2013190569A3/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Substituted aryl acrylic acid addition salts of Sunitinib (I), hydrate thereof, solvate thereof, processes thereof, and pharmaceutical composition thereof are provided. [Formula should be inserted here]
PCT/IN2013/000374 2012-06-22 2013-06-17 Novel salts of sunitinib and their preparation Ceased WO2013190569A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN2471/CHE/2012 2012-06-22
IN2471CH2012 2012-06-22

Publications (2)

Publication Number Publication Date
WO2013190569A2 WO2013190569A2 (en) 2013-12-27
WO2013190569A3 true WO2013190569A3 (en) 2014-02-13

Family

ID=49769635

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IN2013/000374 Ceased WO2013190569A2 (en) 2012-06-22 2013-06-17 Novel salts of sunitinib and their preparation

Country Status (1)

Country Link
WO (1) WO2013190569A2 (en)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101333215A (en) * 2008-07-29 2008-12-31 南京工业大学 A kind of synthetic method of sunitinib base
WO2010049449A2 (en) * 2008-10-28 2010-05-06 Lek Pharmaceuticals D.D. Novel salts of sunitinib
WO2011104555A2 (en) * 2010-02-25 2011-09-01 Generics [Uk] Limited Novel process

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101333215A (en) * 2008-07-29 2008-12-31 南京工业大学 A kind of synthetic method of sunitinib base
WO2010049449A2 (en) * 2008-10-28 2010-05-06 Lek Pharmaceuticals D.D. Novel salts of sunitinib
WO2011104555A2 (en) * 2010-02-25 2011-09-01 Generics [Uk] Limited Novel process

Also Published As

Publication number Publication date
WO2013190569A2 (en) 2013-12-27

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