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WO2012060790A3 - Formulations de cefpodoxime proxétil dispersibles dans l'eau - Google Patents

Formulations de cefpodoxime proxétil dispersibles dans l'eau Download PDF

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Publication number
WO2012060790A3
WO2012060790A3 PCT/TR2011/000255 TR2011000255W WO2012060790A3 WO 2012060790 A3 WO2012060790 A3 WO 2012060790A3 TR 2011000255 W TR2011000255 W TR 2011000255W WO 2012060790 A3 WO2012060790 A3 WO 2012060790A3
Authority
WO
WIPO (PCT)
Prior art keywords
formulations
water dispersible
cefpodoxime proxetil
proxetil
cefpodoxime
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/TR2011/000255
Other languages
English (en)
Other versions
WO2012060790A2 (fr
Inventor
Mahmut Bilgic
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of WO2012060790A2 publication Critical patent/WO2012060790A2/fr
Publication of WO2012060790A3 publication Critical patent/WO2012060790A3/fr
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne des formulations pharmaceutiques comprenant du cefpodoxime proxétil.
PCT/TR2011/000255 2010-11-05 2011-11-03 Formulations de cefpodoxime proxétil dispersibles dans l'eau Ceased WO2012060790A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
TR2010/09168 2010-11-05
TR2010/09168A TR201009168A2 (tr) 2010-11-05 2010-11-05 Suda dağılan sefpodoksim proksetil formülasyonları.

Publications (2)

Publication Number Publication Date
WO2012060790A2 WO2012060790A2 (fr) 2012-05-10
WO2012060790A3 true WO2012060790A3 (fr) 2012-09-20

Family

ID=45446166

Family Applications (2)

Application Number Title Priority Date Filing Date
PCT/TR2011/000251 Ceased WO2012060786A2 (fr) 2010-11-05 2011-11-03 Formulations de proxétil cefpodoxime comprenant un agent de viscosité
PCT/TR2011/000255 Ceased WO2012060790A2 (fr) 2010-11-05 2011-11-03 Formulations de cefpodoxime proxétil dispersibles dans l'eau

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PCT/TR2011/000251 Ceased WO2012060786A2 (fr) 2010-11-05 2011-11-03 Formulations de proxétil cefpodoxime comprenant un agent de viscosité

Country Status (2)

Country Link
TR (1) TR201009168A2 (fr)
WO (2) WO2012060786A2 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2833872A1 (fr) * 2012-04-04 2015-02-11 Mahmut Bilgic Formulations en comprimés comprenant du cefpodoxime proxétil et de l'acide clavulanique
CN103142506B (zh) * 2013-04-03 2015-02-25 天津医药集团津康制药有限公司 一种头孢泊肟酯颗粒剂及其制备方法
CN103230367B (zh) * 2013-05-07 2014-11-12 山东罗欣药业集团股份有限公司 一种头孢泊肟酯组合物干混悬剂及其制备方法
MX2017007287A (es) * 2014-12-01 2017-08-25 Sun Pharmaceutical Ind Ltd Composicion de cefpodoxima proxetil de liberacion prolongada.

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002067943A1 (fr) * 2001-02-27 2002-09-06 Ranbaxy Laboratories Limited Composition pharmaceutique orale de cefpodoxime-proxetil
WO2004004737A1 (fr) * 2002-07-08 2004-01-15 Sankyo Company, Limited Preparation de cephalosporine a administration orale
WO2004006917A1 (fr) * 2002-07-16 2004-01-22 Ranbaxy Laboratories Limited Comprimes dispersibles pour administration par voie orale
WO2007017895A2 (fr) * 2005-05-05 2007-02-15 Lupin Limited Compositions pharmaceutiques stabilisees de cephalosporines
WO2011129792A1 (fr) * 2010-04-13 2011-10-20 Mahmut Bilgic Formulations dispersibles dans l'eau comprenant le cefpodoxime proxétil

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4486425A (en) 1980-09-30 1984-12-04 Sankyo Company Limited 7-[2-(2-Aminothiazol-4-yl)-2-(syn)-methoxyiminoacetamido]-3-methoxymethyl-3-cephem-4-carboxylates
JP4526247B2 (ja) * 2002-07-08 2010-08-18 第一三共株式会社 経口用セファロスポリン製剤

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002067943A1 (fr) * 2001-02-27 2002-09-06 Ranbaxy Laboratories Limited Composition pharmaceutique orale de cefpodoxime-proxetil
WO2004004737A1 (fr) * 2002-07-08 2004-01-15 Sankyo Company, Limited Preparation de cephalosporine a administration orale
WO2004006917A1 (fr) * 2002-07-16 2004-01-22 Ranbaxy Laboratories Limited Comprimes dispersibles pour administration par voie orale
WO2007017895A2 (fr) * 2005-05-05 2007-02-15 Lupin Limited Compositions pharmaceutiques stabilisees de cephalosporines
WO2011129792A1 (fr) * 2010-04-13 2011-10-20 Mahmut Bilgic Formulations dispersibles dans l'eau comprenant le cefpodoxime proxétil

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
DATABASE WPI Week 200416, Derwent World Patents Index; AN 2004-169094, XP002676813 *

Also Published As

Publication number Publication date
WO2012060790A2 (fr) 2012-05-10
WO2012060786A3 (fr) 2012-07-26
WO2012060786A2 (fr) 2012-05-10
TR201009168A2 (tr) 2012-05-21

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