WO2011143772A9 - Inhibitors of hiv replication - Google Patents
Inhibitors of hiv replication Download PDFInfo
- Publication number
- WO2011143772A9 WO2011143772A9 PCT/CA2011/050308 CA2011050308W WO2011143772A9 WO 2011143772 A9 WO2011143772 A9 WO 2011143772A9 CA 2011050308 W CA2011050308 W CA 2011050308W WO 2011143772 A9 WO2011143772 A9 WO 2011143772A9
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- inhibitors
- hiv replication
- hiv
- replication
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- AIDS & HIV (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Compounds of formula (I) wherein R1, R2, n and R3 are defined herein, are useful as inhibitors of HIV replication.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US34714110P | 2010-05-21 | 2010-05-21 | |
| US61/347,141 | 2010-05-21 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO2011143772A1 WO2011143772A1 (en) | 2011-11-24 |
| WO2011143772A9 true WO2011143772A9 (en) | 2012-12-20 |
Family
ID=44991137
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/CA2011/050308 Ceased WO2011143772A1 (en) | 2010-05-21 | 2011-05-17 | Inhibitors of hiv replication |
Country Status (1)
| Country | Link |
|---|---|
| WO (1) | WO2011143772A1 (en) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT2729448E (en) | 2011-07-06 | 2015-12-02 | Gilead Sciences Inc | Compounds for the treatment of hiv |
| TWI694071B (en) | 2013-03-01 | 2020-05-21 | 美商基利科學股份有限公司 | Therapeutic compounds for the treatment of retroviridae virus infections |
| TWI652014B (en) * | 2013-09-13 | 2019-03-01 | 美商艾佛艾姆希公司 | Heterocyclic substituted bicycloazole insecticide |
| US10202353B2 (en) | 2014-02-28 | 2019-02-12 | Gilead Sciences, Inc. | Therapeutic compounds |
| JP6716785B2 (en) | 2016-08-19 | 2020-07-01 | ギリアード サイエンシーズ， インコーポレイテッド | Therapeutic compounds useful for prophylactic or therapeutic treatment of HIV viral infections |
| TWI687415B (en) | 2017-08-17 | 2020-03-11 | 美商基利科學股份有限公司 | Solid forms of an hiv capsid inhibitor |
| AR112412A1 (en) | 2017-08-17 | 2019-10-23 | Gilead Sciences Inc | CHOLINE SALT FORMS OF AN HIV CAPSID INHIBITOR |
| ES2958828T3 (en) | 2018-02-15 | 2024-02-15 | Gilead Sciences Inc | Pyridine derivatives and their use to treat HIV infection |
| PL3752496T3 (en) | 2018-02-16 | 2023-11-27 | Gilead Sciences, Inc. | Methods and intermediates for preparing a therapeutic compound useful in the treatment of retroviridae viral infection |
| CN120078775A (en) | 2018-07-16 | 2025-06-03 | 吉利德科学公司 | Capsid inhibitors for HIV treatment |
| AU2020391466B2 (en) | 2019-11-26 | 2024-05-23 | Gilead Sciences, Inc. | Capsid inhibitors for the prevention of HIV |
| CA3181690A1 (en) | 2020-06-25 | 2021-12-30 | Chienhung CHOU | Capsid inhibitors for the treatment of hiv |
| PL4445900T3 (en) | 2021-12-03 | 2025-09-22 | Gilead Sciences, Inc. | THERAPEUTIC COMPOUNDS AGAINST HIV INFECTION |
| WO2023102529A1 (en) | 2021-12-03 | 2023-06-08 | Gilead Sciences, Inc. | Therapeutic compounds for hiv virus infection |
| WO2023102523A1 (en) | 2021-12-03 | 2023-06-08 | Gilead Sciences, Inc. | Therapeutic compounds for hiv virus infection |
-
2011
- 2011-05-17 WO PCT/CA2011/050308 patent/WO2011143772A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011143772A1 (en) | 2011-11-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 121 | Ep: the epo has been informed by wipo that ep was designated in this application |
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| NENP | Non-entry into the national phase in: |
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| 122 | Ep: pct application non-entry in european phase |
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