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WO2011062437A3 - 고나도트로핀 방출 호르몬 수용체 길항제, 이의 제조방법 및 이를 함유하는 약제학적 조성물 - Google Patents

고나도트로핀 방출 호르몬 수용체 길항제, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Download PDF

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Publication number
WO2011062437A3
WO2011062437A3 PCT/KR2010/008194 KR2010008194W WO2011062437A3 WO 2011062437 A3 WO2011062437 A3 WO 2011062437A3 KR 2010008194 W KR2010008194 W KR 2010008194W WO 2011062437 A3 WO2011062437 A3 WO 2011062437A3
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WO
WIPO (PCT)
Prior art keywords
releasing hormone
receptor antagonists
manufacturing
pharmaceutical composition
composition containing
Prior art date
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Ceased
Application number
PCT/KR2010/008194
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English (en)
French (fr)
Other versions
WO2011062437A2 (ko
Inventor
김선미
이민희
김재선
정회철
이소영
이수민
김은정
박의선
박성훈
이봉용
엄기안
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SK Chemicals Co Ltd
Original Assignee
SK Chemicals Co Ltd
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Publication date
Application filed by SK Chemicals Co Ltd filed Critical SK Chemicals Co Ltd
Priority to US13/511,065 priority Critical patent/US9034850B2/en
Priority to EP10831804.9A priority patent/EP2390250B1/en
Priority to ES10831804T priority patent/ES2549502T3/es
Priority to JP2012539815A priority patent/JP5757956B2/ja
Publication of WO2011062437A2 publication Critical patent/WO2011062437A2/ko
Publication of WO2011062437A3 publication Critical patent/WO2011062437A3/ko
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D239/52—Two oxygen atoms
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

본 발명은 고나도트로핀 방출 호르몬("GnRH")(황체형성 호르몬 방출 호르몬으로서도 공지됨) 수용체 길항제에 관한 것이다.
PCT/KR2010/008194 2009-11-20 2010-11-19 고나도트로핀 방출 호르몬 수용체 길항제, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Ceased WO2011062437A2 (ko)

Priority Applications (4)

Application Number Priority Date Filing Date Title
US13/511,065 US9034850B2 (en) 2009-11-20 2010-11-19 Gonadotropin releasing hormone receptor antagonist, preparation method thereof and pharmaceutical composition comprising the same
EP10831804.9A EP2390250B1 (en) 2009-11-20 2010-11-19 Gonadotropin releasing hormone receptor antagonists, manufacturing method thereof, and pharmaceutical composition containing same
ES10831804T ES2549502T3 (es) 2009-11-20 2010-11-19 Antagonistas de receptores de gonadoliberina, método de fabricación de los mismos, y composición farmacéutica que los contienen
JP2012539815A JP5757956B2 (ja) 2009-11-20 2010-11-19 ゴナドトロピン放出ホルモン受容体拮抗剤、その製造方法及びそれを含む医薬組成物

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
KR10-2009-0112896 2009-11-20
KR20090112896 2009-11-20
KR10-2010-0115345 2010-11-19
KR1020100115345A KR101122606B1 (ko) 2009-11-20 2010-11-19 고나도트로핀 방출 호르몬 수용체 길항제, 이의 제조방법 및 이를 함유하는 약제학적 조성물

Publications (2)

Publication Number Publication Date
WO2011062437A2 WO2011062437A2 (ko) 2011-05-26
WO2011062437A3 true WO2011062437A3 (ko) 2011-11-03

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PCT/KR2010/008194 Ceased WO2011062437A2 (ko) 2009-11-20 2010-11-19 고나도트로핀 방출 호르몬 수용체 길항제, 이의 제조방법 및 이를 함유하는 약제학적 조성물

Country Status (6)

Country Link
US (1) US9034850B2 (ko)
EP (1) EP2390250B1 (ko)
JP (1) JP5757956B2 (ko)
KR (2) KR101122606B1 (ko)
ES (1) ES2549502T3 (ko)
WO (1) WO2011062437A2 (ko)

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