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WO2010072398A3 - Formulations vétérinaires - Google Patents

Formulations vétérinaires Download PDF

Info

Publication number
WO2010072398A3
WO2010072398A3 PCT/EP2009/009196 EP2009009196W WO2010072398A3 WO 2010072398 A3 WO2010072398 A3 WO 2010072398A3 EP 2009009196 W EP2009009196 W EP 2009009196W WO 2010072398 A3 WO2010072398 A3 WO 2010072398A3
Authority
WO
WIPO (PCT)
Prior art keywords
alcohol
buprenorphine
pharmaceutical formulations
pharmaceutically acceptable
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/EP2009/009196
Other languages
English (en)
Other versions
WO2010072398A2 (fr
Inventor
Philip Watson
Claire Fowler
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Ltd
Original Assignee
Boehringer Ingelheim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Ltd filed Critical Boehringer Ingelheim Ltd
Publication of WO2010072398A2 publication Critical patent/WO2010072398A2/fr
Publication of WO2010072398A3 publication Critical patent/WO2010072398A3/fr
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La présente invention concerne une formulation pharmaceutique comprenant de la buprénorphine ou l'un de ses sels pharmaceutiquement acceptables et un alcool, ladite formulation contenant une concentration ≤ 1 % p/v de buprénorphine ou de son sel ; et une formulation pharmaceutique comprenant de la buprénorphine ou l'un de ses sels pharmaceutiquement acceptables et un alcool, ladite formulation contenant une concentration ≤ 3 % p/v d'alcool. L'invention concerne également l'utilisation desdites préparations en tant qu'antalgiques ou sédatifs. L'invention concerne en outre un produit comprenant un récipient doté d'une ouverture refermable contenant de 5 à 50 ml, de préférence de 10 à 20 ml, d'une formulation pharmaceutique comprenant de la buprénorphine ou l'un de ses sels acceptables pharmaceutiquement et un alcool, de préférence l'alcool benzylique.
PCT/EP2009/009196 2008-12-22 2009-12-21 Formulations vétérinaires Ceased WO2010072398A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08254107 2008-12-22
EP08254107.9 2008-12-22

Publications (2)

Publication Number Publication Date
WO2010072398A2 WO2010072398A2 (fr) 2010-07-01
WO2010072398A3 true WO2010072398A3 (fr) 2010-11-25

Family

ID=40655918

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2009/009196 Ceased WO2010072398A2 (fr) 2008-12-22 2009-12-21 Formulations vétérinaires

Country Status (1)

Country Link
WO (1) WO2010072398A2 (fr)

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0069600A2 (fr) * 1981-07-10 1983-01-12 Reckitt And Colman Products Limited Compositions pharmaceutiques
WO2003080022A2 (fr) * 2002-03-19 2003-10-02 Ionix Pharmaceuticals Limited Analgesiques
US20070117828A1 (en) * 2005-11-21 2007-05-24 Schering-Plough Animal Health Corp. Pharmaceutical compositions
WO2008047163A1 (fr) * 2006-10-18 2008-04-24 Pharmasol Limited Composition de pulvérisation sans pressurisation contenant de la buprénorphine pour administration par voie transmuqueuse
WO2008106571A2 (fr) * 2007-02-28 2008-09-04 Abbott Laboratories Formulations parentérales de buprénorphine à libération prolongée

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0069600A2 (fr) * 1981-07-10 1983-01-12 Reckitt And Colman Products Limited Compositions pharmaceutiques
WO2003080022A2 (fr) * 2002-03-19 2003-10-02 Ionix Pharmaceuticals Limited Analgesiques
US20070117828A1 (en) * 2005-11-21 2007-05-24 Schering-Plough Animal Health Corp. Pharmaceutical compositions
WO2008047163A1 (fr) * 2006-10-18 2008-04-24 Pharmasol Limited Composition de pulvérisation sans pressurisation contenant de la buprénorphine pour administration par voie transmuqueuse
WO2008106571A2 (fr) * 2007-02-28 2008-09-04 Abbott Laboratories Formulations parentérales de buprénorphine à libération prolongée

Also Published As

Publication number Publication date
WO2010072398A2 (fr) 2010-07-01

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