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WO2009069312A1 - （１ｈ－１，２，４－トリアゾール－１－イル）アリール化合物及びその製造方法 - Google Patents

（１ｈ－１，２，４－トリアゾール－１－イル）アリール化合物及びその製造方法 Download PDF

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Publication number
WO2009069312A1
WO2009069312A1 PCT/JP2008/003520 JP2008003520W WO2009069312A1 WO 2009069312 A1 WO2009069312 A1 WO 2009069312A1 JP 2008003520 W JP2008003520 W JP 2008003520W WO 2009069312 A1 WO2009069312 A1 WO 2009069312A1
Authority
WO
WIPO (PCT)
Prior art keywords
compound
triazol
group
aryl
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/JP2008/003520
Other languages
English (en)
French (fr)
Inventor
Kentaro Kawazoe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ihara Chemical Industry Co Ltd
Original Assignee
Ihara Chemical Industry Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ihara Chemical Industry Co Ltd filed Critical Ihara Chemical Industry Co Ltd
Priority to US12/743,730 priority Critical patent/US8440838B2/en
Priority to CN2008801237500A priority patent/CN101910140A/zh
Priority to JP2009543675A priority patent/JP5507257B2/ja
Priority to EP08854741.9A priority patent/EP2226317B1/en
Publication of WO2009069312A1 publication Critical patent/WO2009069312A1/ja
Anticipated expiration legal-status Critical
Priority to US13/624,107 priority patent/US8648207B2/en
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/14—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

【課題】本発明は、殺虫剤等として有用な３－（１Ｈ－１，２，４－トリアゾール－１－イル）フェニルスルフィド化合物を簡便に効率よく製造するために有用な、（１Ｈ－１，２，４－トリアゾール－１－イル）アリール化合物並びにその製造方法を提供する。 【解決手段】一般式（１） （式中、ＲはＣ１～Ｃ６アルキル基又は環状Ｃ１～Ｃ６アルキル基を示し、Ａ１は水素原子、アミノ基、モノ（Ｃ１～Ｃ６アルキル）アミノ基又はジ（Ｃ１～Ｃ６アルキル）アミノ基を示し、Ａ２はハロゲン原子、Ｃ１～Ｃ６アルキル基又は環状Ｃ１～Ｃ６アルキル基を示し、Ｚは水素原子、ハロスルホニル基又はメルカプト基を示す。）で表される（１Ｈ－１，２，４－トリアゾール－１－イル）アリール化合物並びにその製造方法。
PCT/JP2008/003520 2007-11-30 2008-11-28 （１ｈ－１，２，４－トリアゾール－１－イル）アリール化合物及びその製造方法 Ceased WO2009069312A1 (ja)

Priority Applications (5)

Application Number Priority Date Filing Date Title
US12/743,730 US8440838B2 (en) 2007-11-30 2008-11-28 Aryl (1H-1,2,4-triazol-1-yl) compound and process for production thereof
CN2008801237500A CN101910140A (zh) 2007-11-30 2008-11-28 (1h-1,2,4-三唑-1-基)芳基化合物及其制备方法
JP2009543675A JP5507257B2 (ja) 2007-11-30 2008-11-28 （１ｈ−１，２，４−トリアゾール−１−イル）アリール化合物及びその製造方法
EP08854741.9A EP2226317B1 (en) 2007-11-30 2008-11-28 Aryl (1h-1,2,4-triazol-1-yl) compound, and process for production thereof
US13/624,107 US8648207B2 (en) 2007-11-30 2012-09-21 Aryl (1H-1,2,4-triazol-1-yl) compound, and process for production thereof

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007-310537 2007-11-30
JP2007310537 2007-11-30

Related Child Applications (2)

Application Number Title Priority Date Filing Date
US12/743,730 A-371-Of-International US8440838B2 (en) 2007-11-30 2008-11-28 Aryl (1H-1,2,4-triazol-1-yl) compound and process for production thereof
US13/624,107 Division US8648207B2 (en) 2007-11-30 2012-09-21 Aryl (1H-1,2,4-triazol-1-yl) compound, and process for production thereof

Publications (1)

Publication Number Publication Date
WO2009069312A1 true WO2009069312A1 (ja) 2009-06-04

Family

ID=40678224

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2008/003520 Ceased WO2009069312A1 (ja) 2007-11-30 2008-11-28 （１ｈ－１，２，４－トリアゾール－１－イル）アリール化合物及びその製造方法

Country Status (6)

Country Link
US (2) US8440838B2 (ja)
EP (1) EP2226317B1 (ja)
JP (1) JP5507257B2 (ja)
KR (1) KR101574655B1 (ja)
CN (2) CN101910140A (ja)
WO (1) WO2009069312A1 (ja)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2274982A1 (de) * 2009-07-16 2011-01-19 Bayer CropScience AG Verwendung von Phenyltriazolen zur Bekämpfung von Insekten und Spinnmilben durch Angiessen, Tröpfchen- oder Tauchapplikation oder durch Behandlung von Saatgut
CN102471290A (zh) * 2009-07-16 2012-05-23 拜尔农作物科学股份公司 手性3-三唑基亚砜衍生物的制备方法
JP2013502387A (ja) * 2009-08-20 2013-01-24 バイエル・クロップサイエンス・アーゲー 殺ダニ剤および殺虫剤としての３−トリアゾリルフェニル置換スルフィド誘導体
JP2013502386A (ja) * 2009-08-20 2013-01-24 バイエル・クロップサイエンス・アーゲー 殺ダニ剤及び殺虫剤として使用するための３−［１−（３−ハロアルキル）−トリアゾリル］−フェニル−スルフィド誘導体
EP3002279A1 (de) 2014-10-02 2016-04-06 Bayer CropScience AG Verfahren zur Herstellung von 3-(5-Aminotriazolyl)-Sulfid-Derivaten

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT5937B (lt) 2011-09-01 2013-05-27 Uab "Precizika - Met Sc" Puslaidininkinis elementas, turintis legiruotas p/n struktūras, ir būdas jas izoliuoti naudojant ultratrumpus ultravioletinius lazerio impulsus
CN111825585B (zh) 2019-09-23 2021-12-14 山东康乔生物科技有限公司 一种含苄胺结构的芳基硫化物及其合成方法和应用

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2000198768A (ja) * 1998-04-27 2000-07-18 Kumiai Chem Ind Co Ltd ３―アリ―ルフェニルスルフィド誘導体及び殺虫、殺ダニ剤
WO2006043635A1 (ja) 2004-10-20 2006-04-27 Kumiai Chemical Industry Co., Ltd. ３－トリアゾリルフェニルスルフィド誘導体及びそれを有効成分として含有する殺虫・殺ダニ・殺線虫剤
JP2007284356A (ja) * 2006-04-12 2007-11-01 Kumiai Chem Ind Co Ltd ３−トリアゾリルフェニルスルフィド誘導体及びそれを有効成分として含有する農園芸用殺虫・殺ダニ・殺線虫剤

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3869167D1 (de) * 1987-03-27 1992-04-23 Kumiai Chemical Industry Co Phenyltriazol-derivate und insectizid.
JP2729810B2 (ja) * 1988-09-27 1998-03-18 クミアイ化学工業株式会社 フェニルトリアゾール誘導体及び殺虫剤
TW226993B (ja) * 1992-05-29 1994-07-21 Kumiai Chemical Industry Co
JP3682075B2 (ja) * 1993-04-16 2005-08-10 クミアイ化学工業株式会社 トリアゾール誘導体及び殺虫、殺ダニ剤
JPH07258227A (ja) * 1994-03-25 1995-10-09 Kumiai Chem Ind Co Ltd フェニルトリアゾール誘導体及び殺虫剤
DE19548415A1 (de) * 1995-12-22 1997-06-26 Bayer Ag 1-Aryl-3-halogenalkyl-5-arylaminotriazole
WO1999055668A1 (en) * 1998-04-27 1999-11-04 Kumiai Chemical Industry Co., Ltd. 3-arylphenyl sulfide derivatives and insecticides and miticides
JP2000239262A (ja) * 1999-02-17 2000-09-05 Sumitomo Chem Co Ltd トリアゾール化合物およびその用途
WO2007114532A1 (en) * 2006-04-03 2007-10-11 Industry-Academic Cooperation Foundation Gyeongsang National University Novel chalcone derivatives, pharmaceutically acceptable salt, method for preparation and uses thereof
WO2008129288A2 (en) * 2007-04-19 2008-10-30 Boehringer Ingelheim International Gmbh Disulfonamides useful in the treatment of inflammation

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2000198768A (ja) * 1998-04-27 2000-07-18 Kumiai Chem Ind Co Ltd ３―アリ―ルフェニルスルフィド誘導体及び殺虫、殺ダニ剤
WO2006043635A1 (ja) 2004-10-20 2006-04-27 Kumiai Chemical Industry Co., Ltd. ３－トリアゾリルフェニルスルフィド誘導体及びそれを有効成分として含有する殺虫・殺ダニ・殺線虫剤
JP2007284356A (ja) * 2006-04-12 2007-11-01 Kumiai Chem Ind Co Ltd ３−トリアゾリルフェニルスルフィド誘導体及びそれを有効成分として含有する農園芸用殺虫・殺ダニ・殺線虫剤

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
See also references of EP2226317A4 *

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2274982A1 (de) * 2009-07-16 2011-01-19 Bayer CropScience AG Verwendung von Phenyltriazolen zur Bekämpfung von Insekten und Spinnmilben durch Angiessen, Tröpfchen- oder Tauchapplikation oder durch Behandlung von Saatgut
WO2011006605A1 (de) * 2009-07-16 2011-01-20 Bayer Cropscience Aktiengesellschaft Verwendung von phenyltriazolen zur bekämpfung von insekten und spinnmilben durch angiessen, tröpfchen- oder tauchapplikation oder durch behandlung von saatgut
CN102469787A (zh) * 2009-07-16 2012-05-23 拜尔农作物科学股份公司 苯基三唑通过浇水、弥雾或浸渍或者通过处理种子而用于防治昆虫和叶螨的用途
CN102471290A (zh) * 2009-07-16 2012-05-23 拜尔农作物科学股份公司 手性3-三唑基亚砜衍生物的制备方法
AU2010272874B2 (en) * 2009-07-16 2015-01-15 Bayer Intellectual Property Gmbh Use of phenyl triazoles for controlling insects and spider mites by splashing, misting or immersion or by treatment of seeds
CN102471290B (zh) * 2009-07-16 2016-02-03 拜耳知识产权有限责任公司 手性3-三唑基亚砜衍生物的制备方法
JP2013502387A (ja) * 2009-08-20 2013-01-24 バイエル・クロップサイエンス・アーゲー 殺ダニ剤および殺虫剤としての３−トリアゾリルフェニル置換スルフィド誘導体
JP2013502386A (ja) * 2009-08-20 2013-01-24 バイエル・クロップサイエンス・アーゲー 殺ダニ剤及び殺虫剤として使用するための３−［１−（３−ハロアルキル）−トリアゾリル］−フェニル−スルフィド誘導体
EP3002279A1 (de) 2014-10-02 2016-04-06 Bayer CropScience AG Verfahren zur Herstellung von 3-(5-Aminotriazolyl)-Sulfid-Derivaten

Also Published As

Publication number Publication date
KR20100087025A (ko) 2010-08-02
US8440838B2 (en) 2013-05-14
CN103664811B (zh) 2015-09-16
EP2226317A1 (en) 2010-09-08
CN103664811A (zh) 2014-03-26
EP2226317B1 (en) 2015-08-12
US20130023666A1 (en) 2013-01-24
US20100256386A1 (en) 2010-10-07
EP2226317A4 (en) 2012-03-21
CN101910140A (zh) 2010-12-08
US8648207B2 (en) 2014-02-11
JPWO2009069312A1 (ja) 2011-04-07
JP5507257B2 (ja) 2014-05-28
KR101574655B1 (ko) 2015-12-04

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