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WO2009051162A1 - Procédé de production d'un composé cyclique bicyclo - Google Patents

Procédé de production d'un composé cyclique bicyclo Download PDF

Info

Publication number
WO2009051162A1
WO2009051162A1 PCT/JP2008/068716 JP2008068716W WO2009051162A1 WO 2009051162 A1 WO2009051162 A1 WO 2009051162A1 JP 2008068716 W JP2008068716 W JP 2008068716W WO 2009051162 A1 WO2009051162 A1 WO 2009051162A1
Authority
WO
WIPO (PCT)
Prior art keywords
bicyclo
ring compound
bicyclo ring
dihaloamine
enables
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/JP2008/068716
Other languages
English (en)
Japanese (ja)
Inventor
Takafumi Yoshimura
Shoji Hara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hokkaido University NUC
Mitsubishi Gas Chemical Co Inc
Original Assignee
Hokkaido University NUC
Mitsubishi Gas Chemical Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hokkaido University NUC, Mitsubishi Gas Chemical Co Inc filed Critical Hokkaido University NUC
Priority to JP2009538126A priority Critical patent/JPWO2009051162A1/ja
Publication of WO2009051162A1 publication Critical patent/WO2009051162A1/fr
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/08—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

L'invention concerne un procédé industriellement avantageux qui permet de produire rapidement un composé cyclique bicyclo qui est utile en tant que matière première pour des produits très fonctionnels comme les produits pharmaceutiques, les produits agrochimiques et les cristaux liquides, dans des conditions modérées autour de la température ambiante. L'invention concerne en particulier un procédé de production d'un composé cyclique bicyclo, ledit composé qui comporte trois atomes d'hydrogène actifs dérivés d'un groupe hydroxy et/ou d'un groupe amine étant amené à réagir avec une α,α-dihaloamine. Ce procédé permet de simplifier et de produire avec un bon rendement un bicyclo-orthoester, un bicyclo-acétal d'amide ou une bicyclo-trisaminométhane en faisant réagir un triol, un aminodiol ou une triamine avec une α,α-dihaloamine.
PCT/JP2008/068716 2007-10-17 2008-10-16 Procédé de production d'un composé cyclique bicyclo Ceased WO2009051162A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2009538126A JPWO2009051162A1 (ja) 2007-10-17 2008-10-16 ビシクロ環化合物の製造方法

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007-269791 2007-10-17
JP2007269791 2007-10-17

Publications (1)

Publication Number Publication Date
WO2009051162A1 true WO2009051162A1 (fr) 2009-04-23

Family

ID=40567424

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2008/068716 Ceased WO2009051162A1 (fr) 2007-10-17 2008-10-16 Procédé de production d'un composé cyclique bicyclo

Country Status (2)

Country Link
JP (1) JPWO2009051162A1 (fr)
WO (1) WO2009051162A1 (fr)

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3143251A1 (de) * 1981-10-31 1983-05-11 Bayer Ag, 5090 Leverkusen Bicyclische orthoesteramide
EP0279698A2 (fr) * 1987-02-20 1988-08-24 The Wellcome Foundation Limited Composés pesticides
EP0285342A2 (fr) * 1987-03-26 1988-10-05 The Wellcome Foundation Limited Pepticides
WO2003020685A1 (fr) * 2001-08-28 2003-03-13 Mitsubishi Gas Chemical Company, Inc. Compose fluore et agent de fluoration contenant ce compose
WO2004050676A1 (fr) * 2002-12-04 2004-06-17 Mitsubishi Gas Chemical Company, Inc. Procede de fluoration

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3143251A1 (de) * 1981-10-31 1983-05-11 Bayer Ag, 5090 Leverkusen Bicyclische orthoesteramide
EP0279698A2 (fr) * 1987-02-20 1988-08-24 The Wellcome Foundation Limited Composés pesticides
EP0285342A2 (fr) * 1987-03-26 1988-10-05 The Wellcome Foundation Limited Pepticides
WO2003020685A1 (fr) * 2001-08-28 2003-03-13 Mitsubishi Gas Chemical Company, Inc. Compose fluore et agent de fluoration contenant ce compose
WO2004050676A1 (fr) * 2002-12-04 2004-06-17 Mitsubishi Gas Chemical Company, Inc. Procede de fluoration

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
FUKUYAMA T. ET AL.: "A Facile Synthesis of Oxazolines, Thiazolines, and Imidazolines Using a, a-Difluoroalkylamines", SYNTHESIS, vol. 10, 16 May 2007 (2007-05-16), pages 1528 - 1534 *

Also Published As

Publication number Publication date
JPWO2009051162A1 (ja) 2011-03-03

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