WO2008087736A1 - アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族アミンの製法 - Google Patents
アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族アミンの製法 Download PDFInfo
- Publication number
- WO2008087736A1 WO2008087736A1 PCT/JP2007/050782 JP2007050782W WO2008087736A1 WO 2008087736 A1 WO2008087736 A1 WO 2008087736A1 JP 2007050782 W JP2007050782 W JP 2007050782W WO 2008087736 A1 WO2008087736 A1 WO 2008087736A1
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- group
- aralkyloxy
- aromatic amine
- aromatic
- heteroaralkyloxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/02—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyridine Compounds (AREA)
Abstract
温和な条件下、簡便な方法によって、アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族ニトロ化合物と水素とを反応させ、脱アラルキル化又は脱ヘテロアラルキル化をさせることなく、またアリール基又はヘテロアリール基上の他の置換基を反応に関与させずに安定に保持しながら、ニトロ基のみを選択的に還元することにより、アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族アミン化合物を製造する方法を提供する。
本発明は、金属触媒の存在下、一般式(1)
(式中、Arは、置換基を有していても良いアリール基又はヘテロアリール基、Zは、置換基を有していても良い二価の芳香族基を示す。)
で示される芳香族ニトロ化合物と水素とを反応させることを特徴とする、一般式(2)
(式中、Ar及びZは、前記と同義である。)
で示される芳香族アミン化合物の製法に関する。
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2008553937A JPWO2008087736A1 (ja) | 2007-01-19 | 2007-01-19 | アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族アミンの製法 |
| EP07707070.4A EP2123627B1 (en) | 2007-01-19 | 2007-01-19 | Process for producing aromatic amine having aralkyloxy or heteroaralkyloxy group |
| PCT/JP2007/050782 WO2008087736A1 (ja) | 2007-01-19 | 2007-01-19 | アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族アミンの製法 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/JP2007/050782 WO2008087736A1 (ja) | 2007-01-19 | 2007-01-19 | アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族アミンの製法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| WO2008087736A1 true WO2008087736A1 (ja) | 2008-07-24 |
Family
ID=39635745
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/JP2007/050782 Ceased WO2008087736A1 (ja) | 2007-01-19 | 2007-01-19 | アラルキルオキシ又はヘテロアラルキルオキシ基を有する芳香族アミンの製法 |
Country Status (3)
| Country | Link |
|---|---|
| EP (1) | EP2123627B1 (ja) |
| JP (1) | JPWO2008087736A1 (ja) |
| WO (1) | WO2008087736A1 (ja) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10599094B2 (en) | 2015-05-29 | 2020-03-24 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102285891B (zh) * | 2011-06-30 | 2014-06-11 | 浙江工业大学 | 一种由芳香硝基化合物催化加氢制备芳胺的方法 |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5143731A (ja) * | 1974-10-08 | 1976-04-14 | Mitsubishi Chem Ind | |
| JP2001503772A (ja) * | 1996-11-11 | 2001-03-21 | セプラクール,インコーポレイテッド | フォルモテロールの光学的に純粋な異性体の製造方法 |
| JP2003286263A (ja) * | 1999-01-22 | 2003-10-10 | Kirin Brewery Co Ltd | キノリン誘導体およびキナゾリン誘導体 |
| WO2004105765A1 (en) * | 2003-05-27 | 2004-12-09 | Janssen Pharmaceutica N.V. | Macrocyclic quinazoline derivatives as antiproliferative agents |
| JP2006519232A (ja) * | 2003-02-26 | 2006-08-24 | スージェン・インコーポレーテッド | プロテインキナーゼ阻害剤としてのアミノヘテロアリール化合物 |
| JP2007051128A (ja) * | 2005-07-22 | 2007-03-01 | Ube Ind Ltd | アラルキルオキシ又はヘテロアラルキルオキシ基を有するアニリンの製法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003029199A1 (en) * | 2001-09-28 | 2003-04-10 | Takeda Chemical Industries, Ltd. | Benzene derivatives, process for preparing the same and use thereof |
| CN100418954C (zh) * | 2002-12-13 | 2008-09-17 | 弗·哈夫曼-拉罗切有限公司 | 3h-喹唑啉-4-酮衍生物 |
| DE602004023876D1 (de) * | 2003-12-18 | 2009-12-10 | Janssen Pharmaceutica Nv | 3-cyano-chinolin-derivate mit antiproliferativer wirkung |
| US7220742B2 (en) * | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
| AR055616A1 (es) * | 2005-09-06 | 2007-08-29 | Smithkline Beecham Corp | Compuestos de tiofeno bencimidazol |
-
2007
- 2007-01-19 EP EP07707070.4A patent/EP2123627B1/en not_active Not-in-force
- 2007-01-19 WO PCT/JP2007/050782 patent/WO2008087736A1/ja not_active Ceased
- 2007-01-19 JP JP2008553937A patent/JPWO2008087736A1/ja active Pending
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5143731A (ja) * | 1974-10-08 | 1976-04-14 | Mitsubishi Chem Ind | |
| JP2001503772A (ja) * | 1996-11-11 | 2001-03-21 | セプラクール,インコーポレイテッド | フォルモテロールの光学的に純粋な異性体の製造方法 |
| JP2003286263A (ja) * | 1999-01-22 | 2003-10-10 | Kirin Brewery Co Ltd | キノリン誘導体およびキナゾリン誘導体 |
| JP2006519232A (ja) * | 2003-02-26 | 2006-08-24 | スージェン・インコーポレーテッド | プロテインキナーゼ阻害剤としてのアミノヘテロアリール化合物 |
| WO2004105765A1 (en) * | 2003-05-27 | 2004-12-09 | Janssen Pharmaceutica N.V. | Macrocyclic quinazoline derivatives as antiproliferative agents |
| JP2007051128A (ja) * | 2005-07-22 | 2007-03-01 | Ube Ind Ltd | アラルキルオキシ又はヘテロアラルキルオキシ基を有するアニリンの製法 |
Non-Patent Citations (4)
| Title |
|---|
| J. MED. CHEM., vol. 45, no. 17, 2002, pages 3772 |
| J. ORG. CHEM., vol. 66, no. 8, 2001, pages 2881 |
| See also references of EP2123627A4 * |
| TETRAHEDRON, vol. 51, no. 19, 1995, pages 5617 |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10599094B2 (en) | 2015-05-29 | 2020-03-24 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
| US11156953B2 (en) | 2015-05-29 | 2021-10-26 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
| US11281156B2 (en) | 2015-05-29 | 2022-03-22 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
| US11314198B2 (en) | 2015-05-29 | 2022-04-26 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
| US11789403B2 (en) | 2015-05-29 | 2023-10-17 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
| US11982972B2 (en) | 2015-05-29 | 2024-05-14 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
| US12321129B2 (en) | 2015-05-29 | 2025-06-03 | Canon Kabushiki Kaisha | Photosensitive member cartridge and process cartridge |
Also Published As
| Publication number | Publication date |
|---|---|
| JPWO2008087736A1 (ja) | 2010-05-06 |
| EP2123627A1 (en) | 2009-11-25 |
| EP2123627A4 (en) | 2010-07-21 |
| EP2123627B1 (en) | 2013-11-20 |
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