WO2007067757A3 - Certains types d'entites chimiques, compositions et methode de modulation de trpv1 - Google Patents
Certains types d'entites chimiques, compositions et methode de modulation de trpv1 Download PDFInfo
- Publication number
- WO2007067757A3 WO2007067757A3 PCT/US2006/047003 US2006047003W WO2007067757A3 WO 2007067757 A3 WO2007067757 A3 WO 2007067757A3 US 2006047003 W US2006047003 W US 2006047003W WO 2007067757 A3 WO2007067757 A3 WO 2007067757A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- chemical entities
- compositions
- methods
- certain chemical
- trpv1
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'invention porte sur des entités chimiques choisies parmi des composés de formule (I) et sur des sels acceptables d'un point de vue pharmaceutique ou cosmétique, des solvates, des chélates, des complexes non covalents, des promédicaments et des mélanges de ceux-ci. Les entités chimiques modulent TRPV1 et sont utiles dans le traitement d'au moins une maladie ou trouble modulé par l'activité de TRPV1.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74935105P | 2005-12-08 | 2005-12-08 | |
| US60/749,351 | 2005-12-08 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO2007067757A2 WO2007067757A2 (fr) | 2007-06-14 |
| WO2007067757A3 true WO2007067757A3 (fr) | 2008-01-31 |
Family
ID=38123536
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/US2006/047003 Ceased WO2007067757A2 (fr) | 2005-12-08 | 2006-12-05 | Certains types d'entites chimiques, compositions et methode de modulation de trpv1 |
Country Status (1)
| Country | Link |
|---|---|
| WO (1) | WO2007067757A2 (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5643112B2 (ja) | 2008-01-28 | 2014-12-17 | アモーレパシフィック コーポレイションAmorepacific Corporation | バニロイド受容体としての新規化合物、その異性体または薬剤学的に許容し得る塩、及びこれを含有する医薬組成物 |
| US8362012B2 (en) | 2008-04-18 | 2013-01-29 | Daewoong Pharmaceutical Co., Ltd. | Benzoxazine benzimidazole derivative, a pharmaceutical composition comprising the same, and a use thereof |
| KR101621444B1 (ko) | 2008-07-02 | 2016-05-19 | (주)아모레퍼시픽 | 바닐로이드 수용체 길항제로 작용하는 신규 화합물, 이의 이성질체 또는 이의 약제학적으로 허용 가능한 염, 및 이를 포함하는 약학 조성물 |
| KR101293384B1 (ko) | 2010-10-13 | 2013-08-05 | 주식회사 대웅제약 | 신규 피리딜 벤조옥사진 유도체, 이를 포함하는 약학 조성물 및 이의 용도 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004096784A1 (fr) * | 2003-04-28 | 2004-11-11 | Astrazeneca Ab | Nouveaux amides heterocycliques |
-
2006
- 2006-12-05 WO PCT/US2006/047003 patent/WO2007067757A2/fr not_active Ceased
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004096784A1 (fr) * | 2003-04-28 | 2004-11-11 | Astrazeneca Ab | Nouveaux amides heterocycliques |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007067757A2 (fr) | 2007-06-14 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| WO2007067711A3 (fr) | Certains types d'entites chimiques, compositions et methode de modulation de trpv1 | |
| WO2005005378A3 (fr) | Hydrazides d'indolinone utilises en tant qu'inhibiteurs du recepteur c-met | |
| WO2005086661A3 (fr) | Composes, compositions pharmaceutiques et procedes d'utilisation dans le traitement de troubles metaboliques | |
| WO2007024717A3 (fr) | Agents permettant de prevenir et de traiter des troubles entrainant la modulation des recepteurs ryr | |
| WO2005040116A3 (fr) | Derives d'indolinone et utilisations de ceux-ci pour traiter des etats pathologiques tels que le cancer | |
| WO2008062276A3 (fr) | Dérivés d'acétylène comme inhibiteurs de la stéaroyl coa désaturase | |
| WO2004080377A3 (fr) | Nouveaux composes modulant le canal kcnq et leur utilisation | |
| ATE540024T1 (de) | Allosterische modulatoren von metabotropen glutamatrezeptoren | |
| TW200602036A (en) | Diphenylazetidone derivates | |
| NO20082145L (no) | Prolinamidderivater som natriumkanalmodulatorer | |
| WO2005061452A8 (fr) | Derives diphenylazetidinone a activite inhibitrice de l'absorption du cholesterol | |
| CY1112727T1 (el) | Παραγωγα κυκλοβουτυλ αμινης βενζοθειαζολης και η χρηση αυτων ως προσδετες των υποδοχεων ισταμινης-3 | |
| DE602005017895D1 (de) | Pyrazolamid-derivate, diese verbindungen enthaltende zusammensetzungen und anwendungsverfahren | |
| WO2007062999A3 (fr) | Derives de indole-2-yl amide substitues en 1,5 | |
| BR0316723A (pt) | Derivados de anilinopirazol úteis para o tratamento de diabetes | |
| WO2005086656A3 (fr) | Derives d'heteroarylaminopyrazole utilises pour traiter le diabete | |
| ATE472529T1 (de) | Prolinamidderivate als natriumkanalmodulatoren | |
| WO2009037542A3 (fr) | Composés spirocycliques en tant qu'inhibiteurs de stéaroyle coa désaturase | |
| MY148538A (en) | Novel 2-azetidinone derivatives as cholesterol absorption inhibitors for the treatment of hyperlipidaemic conditions | |
| ATE380816T1 (de) | Substituierte imidazopyrimidine zur prävention und behandlung von krebs | |
| NO20054787L (no) | Indenderivater som farmasotiske midler | |
| WO2007131907A3 (fr) | Dérivés de 1h-indol-5-yl-pipérazin-1-yl-méthanone | |
| MY138466A (en) | Aminoalkoxyndoles as 5-ht6-receptor ligands for the treatment of cns-disorders | |
| WO2007067757A3 (fr) | Certains types d'entites chimiques, compositions et methode de modulation de trpv1 | |
| WO2007067756A3 (fr) | Certains types d'entites chimiques, compositions et methode de modulation de trpv1 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 121 | Ep: the epo has been informed by wipo that ep was designated in this application | ||
| NENP | Non-entry into the national phase |
Ref country code: DE |
|
| 122 | Ep: pct application non-entry in european phase |
Ref document number: 06845092 Country of ref document: EP Kind code of ref document: A2 |