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WO2004018481A3 - Gossypol derivatives, production methods thereof and uses of same - Google Patents

Gossypol derivatives, production methods thereof and uses of same Download PDF

Info

Publication number
WO2004018481A3
WO2004018481A3 PCT/FR2003/002542 FR0302542W WO2004018481A3 WO 2004018481 A3 WO2004018481 A3 WO 2004018481A3 FR 0302542 W FR0302542 W FR 0302542W WO 2004018481 A3 WO2004018481 A3 WO 2004018481A3
Authority
WO
WIPO (PCT)
Prior art keywords
same
gossypol
production methods
derivatives
gossypol derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/FR2003/002542
Other languages
French (fr)
Other versions
WO2004018481A2 (en
Inventor
Vi-Thuy Dao
Christiane Gaspard
Robert Michelot
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Centre National de la Recherche Scientifique CNRS
Original Assignee
Centre National de la Recherche Scientifique CNRS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Centre National de la Recherche Scientifique CNRS filed Critical Centre National de la Recherche Scientifique CNRS
Priority to AU2003290604A priority Critical patent/AU2003290604A1/en
Publication of WO2004018481A2 publication Critical patent/WO2004018481A2/en
Publication of WO2004018481A3 publication Critical patent/WO2004018481A3/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D339/00Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
    • C07D339/08Six-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D339/00Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
    • C07D339/02Five-membered rings
    • C07D339/06Five-membered rings having the hetero atoms in positions 1 and 3, e.g. cyclic dithiocarbonates

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

The invention relates to derivatives of gossypol and, more specifically, thioderivatives, such as 1,3-dithiolane and 1,3-dithiane, of gossypol, gossypolone and methyl ethers of gossypol. The invention also relates to the methods of producing said derivatives and to the uses of same, e.g. in pharmaceutical compositions for the treatment of cancers.
PCT/FR2003/002542 2002-08-20 2003-08-19 Gossypol derivatives, production methods thereof and uses of same Ceased WO2004018481A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2003290604A AU2003290604A1 (en) 2002-08-20 2003-08-19 Gossypol derivatives, production methods thereof and uses of same

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0210407A FR2843751B1 (en) 2002-08-20 2002-08-20 GOSSYPOL DERIVATIVES, PROCESSES FOR OBTAINING SAME, AND USES THEREOF
FR02/10407 2002-08-20

Publications (2)

Publication Number Publication Date
WO2004018481A2 WO2004018481A2 (en) 2004-03-04
WO2004018481A3 true WO2004018481A3 (en) 2004-04-08

Family

ID=31198223

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/FR2003/002542 Ceased WO2004018481A2 (en) 2002-08-20 2003-08-19 Gossypol derivatives, production methods thereof and uses of same

Country Status (3)

Country Link
AU (1) AU2003290604A1 (en)
FR (1) FR2843751B1 (en)
WO (1) WO2004018481A2 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060144723A1 (en) * 2004-11-02 2006-07-06 Mary Fuller Device for securing valuables

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5385936A (en) * 1990-07-12 1995-01-31 The United States Of America As Represented By The Secretary Of The Department Of The Health And Human Services Gossypol acetic acid for the treatment of cancer

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5385936A (en) * 1990-07-12 1995-01-31 The United States Of America As Represented By The Secretary Of The Department Of The Health And Human Services Gossypol acetic acid for the treatment of cancer

Also Published As

Publication number Publication date
FR2843751B1 (en) 2004-09-24
WO2004018481A2 (en) 2004-03-04
FR2843751A1 (en) 2004-02-27
AU2003290604A1 (en) 2004-03-11

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