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WO2003068791A3 - Macrolides actifs contre staphylococcus aureus resistant a la methicilline - Google Patents

Macrolides actifs contre staphylococcus aureus resistant a la methicilline Download PDF

Info

Publication number
WO2003068791A3
WO2003068791A3 PCT/US2003/004130 US0304130W WO03068791A3 WO 2003068791 A3 WO2003068791 A3 WO 2003068791A3 US 0304130 W US0304130 W US 0304130W WO 03068791 A3 WO03068791 A3 WO 03068791A3
Authority
WO
WIPO (PCT)
Prior art keywords
staphylococcus aureus
activity against
resistant staphylococcus
compounds
macrolides
Prior art date
Application number
PCT/US2003/004130
Other languages
English (en)
Other versions
WO2003068791A2 (fr
Inventor
Zhenkun Ma
Robert Keyes
Stevan Djuric
Hong Yong
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US10/075,012 external-priority patent/US20030162729A1/en
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of WO2003068791A2 publication Critical patent/WO2003068791A2/fr
Publication of WO2003068791A3 publication Critical patent/WO2003068791A3/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Biotechnology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention concerne des composés actifs contre des staphylocoques dorés résistants à la méthicilline (MRSA), ces composés étant représentés par la formule (I). Elle concerne aussi des sels, des promédicaments de ces composés, des procédés de fabrication de ces composés et des intermédiaires utilisés dans les procédés, des compositions contenant ces composés, et des méthodes de prophylaxie et de traitement d'infections dues aux staphylocoques dorés résistants à la méthicilline, au moyen de ces composés.
PCT/US2003/004130 2002-02-13 2003-02-11 Macrolides actifs contre staphylococcus aureus resistant a la methicilline WO2003068791A2 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US10/075,012 US20030162729A1 (en) 2002-02-13 2002-02-13 Macrolides with activity against methicillin-resistant staphylococcus aureus
US10/075,012 2002-02-13
US36147103A 2003-02-10 2003-02-10
US10/361,471 2003-02-10

Publications (2)

Publication Number Publication Date
WO2003068791A2 WO2003068791A2 (fr) 2003-08-21
WO2003068791A3 true WO2003068791A3 (fr) 2004-01-22

Family

ID=27736826

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2003/004130 WO2003068791A2 (fr) 2002-02-13 2003-02-11 Macrolides actifs contre staphylococcus aureus resistant a la methicilline

Country Status (1)

Country Link
WO (1) WO2003068791A2 (fr)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000055168A1 (fr) * 1999-03-15 2000-09-21 Abbott Laboratories Macrolides substitues en 6-o a activite antibacterienne

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000055168A1 (fr) * 1999-03-15 2000-09-21 Abbott Laboratories Macrolides substitues en 6-o a activite antibacterienne

Also Published As

Publication number Publication date
WO2003068791A2 (fr) 2003-08-21

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