WO2003068791A3 - Macrolides actifs contre staphylococcus aureus resistant a la methicilline - Google Patents
Macrolides actifs contre staphylococcus aureus resistant a la methicilline Download PDFInfo
- Publication number
- WO2003068791A3 WO2003068791A3 PCT/US2003/004130 US0304130W WO03068791A3 WO 2003068791 A3 WO2003068791 A3 WO 2003068791A3 US 0304130 W US0304130 W US 0304130W WO 03068791 A3 WO03068791 A3 WO 03068791A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- staphylococcus aureus
- activity against
- resistant staphylococcus
- compounds
- macrolides
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Biotechnology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
L'invention concerne des composés actifs contre des staphylocoques dorés résistants à la méthicilline (MRSA), ces composés étant représentés par la formule (I). Elle concerne aussi des sels, des promédicaments de ces composés, des procédés de fabrication de ces composés et des intermédiaires utilisés dans les procédés, des compositions contenant ces composés, et des méthodes de prophylaxie et de traitement d'infections dues aux staphylocoques dorés résistants à la méthicilline, au moyen de ces composés.
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/075,012 US20030162729A1 (en) | 2002-02-13 | 2002-02-13 | Macrolides with activity against methicillin-resistant staphylococcus aureus |
| US10/075,012 | 2002-02-13 | ||
| US36147103A | 2003-02-10 | 2003-02-10 | |
| US10/361,471 | 2003-02-10 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO2003068791A2 WO2003068791A2 (fr) | 2003-08-21 |
| WO2003068791A3 true WO2003068791A3 (fr) | 2004-01-22 |
Family
ID=27736826
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/US2003/004130 WO2003068791A2 (fr) | 2002-02-13 | 2003-02-11 | Macrolides actifs contre staphylococcus aureus resistant a la methicilline |
Country Status (1)
| Country | Link |
|---|---|
| WO (1) | WO2003068791A2 (fr) |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2000055168A1 (fr) * | 1999-03-15 | 2000-09-21 | Abbott Laboratories | Macrolides substitues en 6-o a activite antibacterienne |
-
2003
- 2003-02-11 WO PCT/US2003/004130 patent/WO2003068791A2/fr active Search and Examination
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2000055168A1 (fr) * | 1999-03-15 | 2000-09-21 | Abbott Laboratories | Macrolides substitues en 6-o a activite antibacterienne |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003068791A2 (fr) | 2003-08-21 |
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