WO2003045909A3 - Procedes et produits intermediaires pour la synthese d'azepines - Google Patents
Procedes et produits intermediaires pour la synthese d'azepines Download PDFInfo
- Publication number
- WO2003045909A3 WO2003045909A3 PCT/US2002/037423 US0237423W WO03045909A3 WO 2003045909 A3 WO2003045909 A3 WO 2003045909A3 US 0237423 W US0237423 W US 0237423W WO 03045909 A3 WO03045909 A3 WO 03045909A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- azepines
- intermediates
- methods
- synthesis
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C215/04—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
- C07C215/06—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
- C07C215/08—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic with only one hydroxy group and one amino group bound to the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C223/00—Compounds containing amino and —CHO groups bound to the same carbon skeleton
- C07C223/02—Compounds containing amino and —CHO groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D223/08—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D223/12—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
L'invention concerne des procédés et des produits intermédiaires permettant de préparer des azépines représentées par la formule (I).
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2002360409A AU2002360409A1 (en) | 2001-11-21 | 2002-11-20 | Methods and intermediates for the synthesis of azepines |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33194901P | 2001-11-21 | 2001-11-21 | |
| US60/331,949 | 2001-11-21 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO2003045909A2 WO2003045909A2 (fr) | 2003-06-05 |
| WO2003045909A3 true WO2003045909A3 (fr) | 2003-12-11 |
Family
ID=23296044
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/US2002/037423 Ceased WO2003045909A2 (fr) | 2001-11-21 | 2002-11-20 | Procedes et produits intermediaires pour la synthese d'azepines |
Country Status (2)
| Country | Link |
|---|---|
| AU (1) | AU2002360409A1 (fr) |
| WO (1) | WO2003045909A2 (fr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CZ20023168A3 (cs) | 2000-03-21 | 2003-02-12 | Smithkline Beecham Corporation | Inhibitory proteázy |
| JP2007520491A (ja) * | 2004-01-23 | 2007-07-26 | スミスクライン・ビーチャム・コーポレイション | ベンゾフラン−２−カルボン酸｛（ｓ）−３−メチル−１−［（４ｓ，７ｒ）−７−メチル−３−オキソ−１−（ピリジン−２−スルホニル）−アゼパン−４−イルカルバモイル］−ブチル｝−アミドの製造方法 |
| CN119504587A (zh) * | 2024-11-26 | 2025-02-25 | 贵州民族大学 | 一种茚并氮杂䓬化合物、其制备方法及医药用途 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001070232A1 (fr) * | 2000-03-21 | 2001-09-27 | Smithkline Beecham Corporation | Inhibiteur de proteinase |
-
2002
- 2002-11-20 WO PCT/US2002/037423 patent/WO2003045909A2/fr not_active Ceased
- 2002-11-20 AU AU2002360409A patent/AU2002360409A1/en not_active Abandoned
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001070232A1 (fr) * | 2000-03-21 | 2001-09-27 | Smithkline Beecham Corporation | Inhibiteur de proteinase |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003045909A2 (fr) | 2003-06-05 |
| AU2002360409A1 (en) | 2003-06-10 |
| AU2002360409A8 (en) | 2003-06-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AK | Designated states |
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| 121 | Ep: the epo has been informed by wipo that ep was designated in this application | ||
| 122 | Ep: pct application non-entry in european phase | ||
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