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WO2002062805A1 - 6-substituted alkylamino-3-pyridylboric acid derivative or salt thereof and processes for producing these - Google Patents

6-substituted alkylamino-3-pyridylboric acid derivative or salt thereof and processes for producing these Download PDF

Info

Publication number
WO2002062805A1
WO2002062805A1 PCT/JP2002/000972 JP0200972W WO02062805A1 WO 2002062805 A1 WO2002062805 A1 WO 2002062805A1 JP 0200972 W JP0200972 W JP 0200972W WO 02062805 A1 WO02062805 A1 WO 02062805A1
Authority
WO
WIPO (PCT)
Prior art keywords
salt
acid derivative
processes
substituted alkylamino
producing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/JP2002/000972
Other languages
French (fr)
Japanese (ja)
Inventor
Hiroshi Kuroda
Kazuya Hayashi
Keisuke Tohdo
Junichi Yokotani
Tamotsu Takamatsu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Toyama Chemical Co Ltd
Original Assignee
Toyama Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Toyama Chemical Co Ltd filed Critical Toyama Chemical Co Ltd
Priority to JP2002563157A priority Critical patent/JP4061194B2/en
Publication of WO2002062805A1 publication Critical patent/WO2002062805A1/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

A 6-substituted alkylamino-3-pyridylboric acid derivative or a salt thereof; and processes for producing these. The processes are shown by the following reaction scheme: [I] wherein each symbol is the same as defined in the description. The processes are useful for the industrial production of intermediates for a quinolonecarboxylic acid derivative or salt thereof useful as an antiinfective remedy. The 6-substituted alkylamino-3-pyridylboric acid derivative or salt thereof is represented by the general formula [1d]: [1d] wherein each symbol is the same as defined in the description. These compounds are useful as intermediates for a quinolonecarboxylic acid derivative or salt thereof useful as an antiinfective remedy.
PCT/JP2002/000972 2001-02-08 2002-02-06 6-substituted alkylamino-3-pyridylboric acid derivative or salt thereof and processes for producing these Ceased WO2002062805A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2002563157A JP4061194B2 (en) 2001-02-08 2002-02-06 6-Substituted alkylamino-3-pyridylboric acid derivatives or salts thereof and methods for producing them

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2001031760 2001-02-08
JP2001-31760 2001-02-08
JP2001111170 2001-04-10
JP2001-111170 2001-04-10

Publications (1)

Publication Number Publication Date
WO2002062805A1 true WO2002062805A1 (en) 2002-08-15

Family

ID=26609099

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2002/000972 Ceased WO2002062805A1 (en) 2001-02-08 2002-02-06 6-substituted alkylamino-3-pyridylboric acid derivative or salt thereof and processes for producing these

Country Status (2)

Country Link
JP (1) JP4061194B2 (en)
WO (1) WO2002062805A1 (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009005015A1 (en) 2007-06-29 2009-01-08 Nissan Chemical Industries, Ltd. Substituted isoxazoline or enone oxime compound, and pest control agent
JP2016502510A (en) * 2012-10-23 2016-01-28 ノバルティス アーゲー Improved process for preparing 5- (2,6-di-4-morpholinyl-4-pyrimidinyl) -4-trifluoromethylpyridin-2-amine
CN107304198A (en) * 2016-04-19 2017-10-31 北京桦冠医药科技有限公司 A kind of new synthesis process of quinolone antibiotic intermediates
CN110563643A (en) * 2019-10-14 2019-12-13 常州齐晖药业有限公司 synthesis method of (5-bromo-3-methyl-pyridin-2-yl) -methylamine

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2018186146A1 (en) * 2017-04-07 2020-02-13 株式会社カネカ Method for producing hydrogenated product and method for removing borane
CN108299480A (en) * 2017-12-27 2018-07-20 山东百诺医药股份有限公司 A kind of preparation method of Ao Zesha stars and its intermediate
CN111675692A (en) * 2020-06-08 2020-09-18 浙江科技学院 A kind of synthetic method of Ao Zesha star

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1070713A1 (en) * 1998-04-06 2001-01-24 Toyama Chemical Co., Ltd. Quinolonecarboxylic acid derivatives or salts thereof

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1070713A1 (en) * 1998-04-06 2001-01-24 Toyama Chemical Co., Ltd. Quinolonecarboxylic acid derivatives or salts thereof

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009005015A1 (en) 2007-06-29 2009-01-08 Nissan Chemical Industries, Ltd. Substituted isoxazoline or enone oxime compound, and pest control agent
US8053452B2 (en) 2007-06-29 2011-11-08 Nissan Chemical Industries, Ltd. Substituted isoxazoline or enone oxime compound, and pest control agent
JP2016502510A (en) * 2012-10-23 2016-01-28 ノバルティス アーゲー Improved process for preparing 5- (2,6-di-4-morpholinyl-4-pyrimidinyl) -4-trifluoromethylpyridin-2-amine
CN107304198A (en) * 2016-04-19 2017-10-31 北京桦冠医药科技有限公司 A kind of new synthesis process of quinolone antibiotic intermediates
CN107304198B (en) * 2016-04-19 2021-02-05 北京桦冠生物技术有限公司 Novel synthesis process of quinolone antibiotic intermediate
CN110563643A (en) * 2019-10-14 2019-12-13 常州齐晖药业有限公司 synthesis method of (5-bromo-3-methyl-pyridin-2-yl) -methylamine

Also Published As

Publication number Publication date
JPWO2002062805A1 (en) 2004-06-10
JP4061194B2 (en) 2008-03-12

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