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WO2000020399A3 - Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for the production thereof and agents containing the same - Google Patents

Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for the production thereof and agents containing the same Download PDF

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Publication number
WO2000020399A3
WO2000020399A3 PCT/EP1999/007125 EP9907125W WO0020399A3 WO 2000020399 A3 WO2000020399 A3 WO 2000020399A3 EP 9907125 W EP9907125 W EP 9907125W WO 0020399 A3 WO0020399 A3 WO 0020399A3
Authority
WO
WIPO (PCT)
Prior art keywords
halide
alkyl
hydroxypyrazoles
alkynyl
alkenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/EP1999/007125
Other languages
German (de)
French (fr)
Other versions
WO2000020399A2 (en
Inventor
Andreas Gypser
Reinhard Kirstgen
Hubert Sauter
Herbert Bayer
Oliver Cullmann
Markus Gewehr
Wassilios Grammenos
Bernd Mueller
Arne Ptock
I Blasco Jordi Tormo
Eberhard Ammermann
Thomas Grote
Gisela Lorenz
Siegfried Strathmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Priority to EP99948860A priority Critical patent/EP1117650A2/en
Priority to AU61965/99A priority patent/AU6196599A/en
Priority to JP2000574516A priority patent/JP2002526536A/en
Publication of WO2000020399A2 publication Critical patent/WO2000020399A2/en
Publication of WO2000020399A3 publication Critical patent/WO2000020399A3/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D231/08—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with oxygen or sulfur atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

The invention relates to the use of substituted 5-hydroxypyrazoles of formula (I) in which the substituents have the following meanings: B represents aryl or heteroaryl; A represents C=O, C=S or SO2; R1 represents alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, cycloalkyl, C¿3?-C10-cycloalkenyl, cycloalkynyl, or aryl, heterocyclyl or heteroaryl; R?2¿ represents hydrogen; R3 represents hydrogen, nitro, cyano, N(R')¿2?, alkyl, alkyl halide, alkoxy, alkoxy halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, whereby R', independent of one another, represents hydrogen or alkyl; or R?2 and R3¿, together, represent a group =O, =S or =N-O-R5, whereby R5 represents hydrogen, alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide; R4 represents hydrogen, halogen, nitro, cyano N(R')¿2?, alkyl, alkyl halide, COOR', heteroaryl or heterocyclyl. The invention also relates to the use of said compounds for combating harmful fungi, to agents containing the compounds, to novel 5-hydroxypyrazoles and to methods for the production thereof.
PCT/EP1999/007125 1998-10-02 1999-09-24 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for the production thereof and agents containing the same Ceased WO2000020399A2 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
EP99948860A EP1117650A2 (en) 1998-10-02 1999-09-24 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for the production thereof and agents containing the same
AU61965/99A AU6196599A (en) 1998-10-02 1999-09-24 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for theproduction thereof and agents containing the same
JP2000574516A JP2002526536A (en) 1998-10-02 1999-09-24 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, processes for their preparation and compositions containing them

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19845509 1998-10-02
DE19845509.7 1998-10-02

Publications (2)

Publication Number Publication Date
WO2000020399A2 WO2000020399A2 (en) 2000-04-13
WO2000020399A3 true WO2000020399A3 (en) 2000-07-27

Family

ID=7883246

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP1999/007125 Ceased WO2000020399A2 (en) 1998-10-02 1999-09-24 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for the production thereof and agents containing the same

Country Status (4)

Country Link
EP (1) EP1117650A2 (en)
JP (1) JP2002526536A (en)
AU (1) AU6196599A (en)
WO (1) WO2000020399A2 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006128815A1 (en) * 2005-05-31 2006-12-07 Basf Aktiengesellschaft Bicyclic 5-hydroxypyrazolines, method for producing the same and agents comprising the same
EP1891015A1 (en) * 2005-05-31 2008-02-27 Basf Aktiengesellschaft Fungicidal 5-hydroxypyrazolines, method for the production thereof, and agents containing the same
WO2006128817A1 (en) * 2005-05-31 2006-12-07 Basf Aktiengesellschaft Fungicidal 5-hydroxypyrazolines, method for producing the same and agents comprising the same
BRPI0610576A2 (en) * 2005-05-31 2016-11-16 Basf Ag compounds, process for preparing same, fungicidal agent, seed, process for combating phytopathogenic harmful fungi, and use of compounds

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0556396A1 (en) * 1990-11-09 1993-08-25 Nissan Chemical Industries, Limited Substituted pyrazole derivative and agrohorticultural bactericide

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0556396A1 (en) * 1990-11-09 1993-08-25 Nissan Chemical Industries, Limited Substituted pyrazole derivative and agrohorticultural bactericide

Non-Patent Citations (12)

* Cited by examiner, † Cited by third party
Title
ANAL. CHIM. ACTA (1985), 170(2), 319-24 *
CHEMICAL ABSTRACTS, vol. 100, no. 3, 16 January 1984, Columbus, Ohio, US; abstract no. 22225, YAKIMOVICH, S.I. ET AL.: "Tautomerism of thiobenzoylhydrazones of aroylacetones and aroylacetaldehydes" XP002133646 *
CHEMICAL ABSTRACTS, vol. 103, no. 20, 18 November 1985, Columbus, Ohio, US; abstract no. 171065, UHLEMANN, E. ET AL: "Complex formation and liquid-liquid extraction of tin with potentially tridentate dianionic ligands" XP002133643 *
CHEMICAL ABSTRACTS, vol. 117, no. 24, 14 December 1992, Columbus, Ohio, US; abstract no. 244557, TOSHEV, M.T. ET AL.: "Structures of condensation products of .beta.-diketones with thiobenzoylhydrazine and their nickel(II) complexes" XP002133644 *
CHEMICAL ABSTRACTS, vol. 131, Columbus, Ohio, US; abstract no. 271830, KALLURAYA, BALAKRISHNA ET AL: "Reactions of aryl/aryloxyacet hydrazides with acetylenic ketones" XP002133647 *
CHEMICAL ABSTRACTS, vol. 96, no. 11, 15 March 1982, Columbus, Ohio, US; abstract no. 85477, KHRUSTALEV, V.A. ET AL.: "Ring-ring tautomerism in 1-thioacyl-5-hydroxy-2-pyrazoline 5-(2-oxoalkyl)-.Delta.21,3,4-thiadiazoline" XP002133645 *
D.M. EVANS ET AL.: "Thiadiazoles and Dihydrothiadiazoles. Part 5. Synthesis of 2,3-Dithydro-1,3,4-thiadiazoles by Reaction of Aldehydes or Ketones with Thioaroylhydrazines", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 1, no. 8, 1986, LETCHWORTH GB, pages 1499 - 1505, XP002133641 *
INDIAN J. HETEROCYCL. CHEM. (1999), 8(4), 309-314 *
YAKIMOVICH, S. I. ET AL: "Tautomerism in a series of products of condensation of fluorinated 1,3-diketones with aroylhydrazines", RUSS. J. ORG. CHEM. (1997), 33(3), 370-374, XP002133642 *
ZH. NEORG. KHIM., vol. 37, no. 5, 1992, pages 1052 - 1061 *
ZH. ORG. KHIM., vol. 17, no. 11, 1981, pages 2451 - 2452 *
ZH. ORG. KHIM., vol. 19, no. 9, 1983, pages 1875 - 1881 *

Also Published As

Publication number Publication date
JP2002526536A (en) 2002-08-20
AU6196599A (en) 2000-04-26
EP1117650A2 (en) 2001-07-25
WO2000020399A2 (en) 2000-04-13

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