[go: up one dir, main page]

WO2000066573A3 - Oxa combinatorial library, production and use thereof - Google Patents

Oxa combinatorial library, production and use thereof Download PDF

Info

Publication number
WO2000066573A3
WO2000066573A3 PCT/FR2000/001138 FR0001138W WO0066573A3 WO 2000066573 A3 WO2000066573 A3 WO 2000066573A3 FR 0001138 W FR0001138 W FR 0001138W WO 0066573 A3 WO0066573 A3 WO 0066573A3
Authority
WO
WIPO (PCT)
Prior art keywords
combinatorial library
oxa
production
compounds
relates
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/FR2000/001138
Other languages
French (fr)
Other versions
WO2000066573A2 (en
Inventor
Xavier Williard
Juliana Pop-Botez
Benoit Deprez
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Cerep SA
Original Assignee
Cerep SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cerep SA filed Critical Cerep SA
Priority to AU43063/00A priority Critical patent/AU4306300A/en
Publication of WO2000066573A2 publication Critical patent/WO2000066573A2/en
Publication of WO2000066573A3 publication Critical patent/WO2000066573A3/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/113—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

The invention relates to a combinatorial library of compounds, characterized in that it comprises substituted derivatives of oxadiazolinone and/or oxadiazolinthione. The invention also relates to novel synthesis paths, such as automated synthesis, for said libraries and compounds. The invention also relates to the use of said libraries in the identification or optimization of compounds which can be used in chemistry, pharmacy or in the agro-food industry.
PCT/FR2000/001138 1999-04-30 2000-04-28 Oxa combinatorial library, production and use thereof Ceased WO2000066573A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU43063/00A AU4306300A (en) 1999-04-30 2000-04-28 Oxa combinatorial library, production and use thereof

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR99/05553 1999-04-30
FR9905553A FR2792936A1 (en) 1999-04-30 1999-04-30 OXA COMBINATORIAL BANKS, PREPARATION AND UTILIZATION.

Publications (2)

Publication Number Publication Date
WO2000066573A2 WO2000066573A2 (en) 2000-11-09
WO2000066573A3 true WO2000066573A3 (en) 2001-03-29

Family

ID=9545115

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/FR2000/001138 Ceased WO2000066573A2 (en) 1999-04-30 2000-04-28 Oxa combinatorial library, production and use thereof

Country Status (3)

Country Link
AU (1) AU4306300A (en)
FR (1) FR2792936A1 (en)
WO (1) WO2000066573A2 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10601074B2 (en) 2011-06-29 2020-03-24 Space Charge, LLC Rugged, gel-free, lithium-free, high energy density solid-state electrochemical energy storage devices
US9853325B2 (en) 2011-06-29 2017-12-26 Space Charge, LLC Rugged, gel-free, lithium-free, high energy density solid-state electrochemical energy storage devices
US10658705B2 (en) 2018-03-07 2020-05-19 Space Charge, LLC Thin-film solid-state energy storage devices
US11996517B2 (en) 2011-06-29 2024-05-28 Space Charge, LLC Electrochemical energy storage devices
US11527774B2 (en) 2011-06-29 2022-12-13 Space Charge, LLC Electrochemical energy storage devices

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0435616A2 (en) * 1989-12-25 1991-07-03 Sumitomo Chemical Company, Limited An oxadiazolinone derivative and its production and use
WO1999009977A1 (en) * 1997-08-22 1999-03-04 Wichita State University 1,2,5-thiadiazolidin-3-one 1,1-dioxide derivatives

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0435616A2 (en) * 1989-12-25 1991-07-03 Sumitomo Chemical Company, Limited An oxadiazolinone derivative and its production and use
WO1999009977A1 (en) * 1997-08-22 1999-03-04 Wichita State University 1,2,5-thiadiazolidin-3-one 1,1-dioxide derivatives

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
BOSCHELLI D H ET AL: "1,3,4-OXADIAZOLE, 1,3,4-THIADIAZOLE, AND 1,2,4-TRIAZOLE ANALOGS OF THE FENAMATES: IN VITRO INHIBITION OF CYCLOOXYGENASE AND 5-LIPOXYGENASE ACTIVITIES", JOURNAL OF MEDICINAL CHEMISTRY,US,AMERICAN CHEMICAL SOCIETY. WASHINGTON, vol. 36, no. 13, pages 1802-1810, XP002049115, ISSN: 0022-2623 *
BRANDSTETTER T W ET AL: "A Galactopyranose Analogue of Hydantocidin", TETRAHEDRON: ASYMMETRY,NL,ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, vol. 7, no. 1, pages 157-170, XP002128624, ISSN: 0957-4166 *
DAVIDSON, JOHN S.: "Some 1-aroyl-4,4-dialkylsemicarbazides and their cyclization to afford 5-aryl-1,3,4-oxadiazol-2(3H)-ones", MONATSH. CHEM. (1988), 119(8-9), 1027-9, XP002128623 *

Also Published As

Publication number Publication date
FR2792936A1 (en) 2000-11-03
WO2000066573A2 (en) 2000-11-09
AU4306300A (en) 2000-11-17

Similar Documents

Publication Publication Date Title
WO2003081261A3 (en) Microdevices having a preferential axis of magnetization and uses thereof
ZA200200179B (en) Process for upgrading of Fischer-Tropsch products.
GB0008392D0 (en) Process for the production of a deodorant or antiperspirant product
ZA200805207B (en) Process for producing condensed-phase product from one or more gas-phase reactants
IS7239A (en) Process for the production of acitalopram
EP1422522A4 (en) Column packing and process for production thereof
WO2000066573A3 (en) Oxa combinatorial library, production and use thereof
ZA200309472B (en) Process for the production of detergent granules.
MXPA03006821A (en) Process and plant for the heterogeneous synthesis of chemical compounds.
IL135804A0 (en) Process for the production of compressed granulates of fertilizers
AU2003279281A1 (en) Automated processes for the production of garments
NO20040566L (en) Improved process for encapsulating a product
IS7834A (en) Process for the synthesis of a benzimidol-sulfur compound
AU2003281818A1 (en) A continuous process for the production of combinatorial libraries of modified materials
SI1403264T1 (en) Process for the industrial synthesis of 5-amino-3-carboxymethyl-4-cyano-2-thiophenecarboxydimethylester
WO1997008190A3 (en) Compounds
EG23204A (en) Process for the production of quinazolines.
AU2002236908A1 (en) Systems, methods, and computer program products for determining the parameters for chemical synthesis and for supplying the reagents, equipment and/or chemicals synthesized thereby
NO20041224L (en) Process for the production of hydrocarbons
AU2002364378A1 (en) Multifunctional reagent for the synthesis of thiol modified oligomers
NO20026112L (en) Process for the preparation of mineral fertilizers
NO20026113L (en) Process for the preparation of mineral fertilizers
NO20010738D0 (en) Luke as well as the process for making it
NO20034839D0 (en) Process for glossing mechanical pulp
NO20022664D0 (en) Process for the preparation of a reaction vessel for vehicles

Legal Events

Date Code Title Description
AK Designated states

Kind code of ref document: A2

Designated state(s): AE AG AL AM AT AU AZ BA BB BG BR BY CA CH CN CR CU CZ DE DK DM DZ EE ES FI GB GD GE GH GM HR HU ID IL IN IS JP KE KG KP KR KZ LC LK LR LS LT LU LV MA MD MG MK MN MW MX NO NZ PL PT RO RU SD SE SG SI SK SL TJ TM TR TT TZ UA UG US UZ VN YU ZA ZW

AL Designated countries for regional patents

Kind code of ref document: A2

Designated state(s): GH GM KE LS MW SD SL SZ TZ UG ZW AM AZ BY KG KZ MD RU TJ TM AT BE CH CY DE DK ES FI FR GB GR IE IT LU MC NL PT SE BF BJ CF CG CI CM GA GN GW ML MR NE SN TD TG

121 Ep: the epo has been informed by wipo that ep was designated in this application
DFPE Request for preliminary examination filed prior to expiration of 19th month from priority date (pct application filed before 20040101)
AK Designated states

Kind code of ref document: A3

Designated state(s): AE AG AL AM AT AU AZ BA BB BG BR BY CA CH CN CR CU CZ DE DK DM DZ EE ES FI GB GD GE GH GM HR HU ID IL IN IS JP KE KG KP KR KZ LC LK LR LS LT LU LV MA MD MG MK MN MW MX NO NZ PL PT RO RU SD SE SG SI SK SL TJ TM TR TT TZ UA UG US UZ VN YU ZA ZW

AL Designated countries for regional patents

Kind code of ref document: A3

Designated state(s): GH GM KE LS MW SD SL SZ TZ UG ZW AM AZ BY KG KZ MD RU TJ TM AT BE CH CY DE DK ES FI FR GB GR IE IT LU MC NL PT SE BF BJ CF CG CI CM GA GN GW ML MR NE SN TD TG

REG Reference to national code

Ref country code: DE

Ref legal event code: 8642

122 Ep: pct application non-entry in european phase
NENP Non-entry into the national phase

Ref country code: JP