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UY33238A - "Compuestos en calidad de antagonistas de bradiquinina-b1" - Google Patents

"Compuestos en calidad de antagonistas de bradiquinina-b1"

Info

Publication number
UY33238A
UY33238A UY0001033238A UY33238A UY33238A UY 33238 A UY33238 A UY 33238A UY 0001033238 A UY0001033238 A UY 0001033238A UY 33238 A UY33238 A UY 33238A UY 33238 A UY33238 A UY 33238A
Authority
UY
Uruguay
Prior art keywords
compounds
pain
antagonists
bradykinin
well
Prior art date
Application number
UY0001033238A
Other languages
English (en)
Inventor
Hauel Norbert
Ceci Angelo
Doods Henri
Konetzki Ingo
Mack Juergen
Priepke Henning
Annette Schuler-Metz
Walter Rainer
Wiedenmayer Dieter
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of UY33238A publication Critical patent/UY33238A/es

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    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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Abstract

La presente invención se refiere a compuestos de 3-oxo-piridazina de fórmula I y a su uso como antagonistas del receptor B1, a composiciones farmacéuticas que contienen estos compuestos así como a métodos para emplear los mismos para la prevención o tratamiento de dolores agudos, dolores viscerales, dolores neuropáticos, dolores inflamatorios y mediados por el receptor del dolor, dolores tumorales así como dolores de cabeza.
UY0001033238A 2009-02-26 2011-02-22 "Compuestos en calidad de antagonistas de bradiquinina-b1" UY33238A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09153778 2009-02-26
PCT/EP2010/052232 WO2010097372A1 (de) 2009-02-26 2010-02-23 Verbindungen als bradykinin-b1-antagonisten

Publications (1)

Publication Number Publication Date
UY33238A true UY33238A (es) 2011-09-30

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MX2011008553A (es) 2011-09-09
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US20100240669A1 (en) 2010-09-23
JP2012518672A (ja) 2012-08-16
EA201101209A1 (ru) 2012-04-30
US8372838B2 (en) 2013-02-12
CA2759126A1 (en) 2010-09-02
PH12012501678A1 (en) 2019-07-10
UA108373C2 (xx) 2015-04-27
PT2401256E (pt) 2013-05-13
TN2012000417A1 (en) 2014-01-30
BRPI1008779A2 (pt) 2020-12-22
ME01526B (me) 2014-04-20
RS53710B1 (sr) 2015-04-30
JP5629274B2 (ja) 2014-11-19
IL214129A0 (en) 2011-08-31
GEP20135933B (en) 2013-10-10
AR075599A1 (es) 2011-04-20
MA33238B1 (fr) 2012-05-02
SG173698A1 (en) 2011-09-29
AU2010217606A1 (en) 2011-09-08
DK2401256T3 (da) 2013-06-03
UA105923C2 (uk) 2014-07-10
EP2401256A1 (de) 2012-01-04
UY32463A (es) 2010-09-30
EA023437B1 (ru) 2016-06-30
IL214129A (en) 2015-08-31
HRP20130666T1 (en) 2013-10-11
WO2010097372A1 (de) 2010-09-02
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ECSP11011304A (es) 2011-10-31
RS52801B (sr) 2013-10-31
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CO6430425A2 (es) 2012-04-30
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