UY33514A - GUANOSINE DERIVATIVE PHOSPHORAMIDATE NECLEOSID COMPOUNDS FOR TREATMENT OF VIRAL INFECTION - Google Patents
GUANOSINE DERIVATIVE PHOSPHORAMIDATE NECLEOSID COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONInfo
- Publication number
- UY33514A UY33514A UY0001033514A UY33514A UY33514A UY 33514 A UY33514 A UY 33514A UY 0001033514 A UY0001033514 A UY 0001033514A UY 33514 A UY33514 A UY 33514A UY 33514 A UY33514 A UY 33514A
- Authority
- UY
- Uruguay
- Prior art keywords
- compounds
- phosphoramidate
- treatment
- necleosid
- viral infection
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 208000036142 Viral infection Diseases 0.000 title abstract 3
- 230000009385 viral infection Effects 0.000 title abstract 3
- NYHBQMYGNKIUIF-UUOKFMHZSA-N Guanosine Chemical class C1=NC=2C(=O)NC(N)=NC=2N1[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O NYHBQMYGNKIUIF-UUOKFMHZSA-N 0.000 title 1
- PTMHPRAIXMAOOB-UHFFFAOYSA-L phosphoramidate Chemical compound NP([O-])([O-])=O PTMHPRAIXMAOOB-UHFFFAOYSA-L 0.000 title 1
- UYTPUPDQBNUYGX-UHFFFAOYSA-N guanine Chemical compound O=C1NC(N)=NC2=C1N=CN2 UYTPUPDQBNUYGX-UHFFFAOYSA-N 0.000 abstract 2
- 241000711549 Hepacivirus C Species 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000008298 phosphoramidates Chemical class 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Los compuestos de Fosforamidato derivados de bases guanina con una mayor potencia terapéutica se proporcionan, y estos compuestos, en particular, tienen mayor potencia con respecto al tratamiento de las infecciones virales, como el virus de la hepatitis C. Composiciones farmacéuticas, los métodos de preparación de los compuestos, y métodos de uso de los compuestos y composiciones para tratar infe cciones virales también se proporcionan.Phosphoramidate compounds derived from guanine bases with greater therapeutic potency are provided, and these compounds, in particular, have greater potency with respect to the treatment of viral infections, such as hepatitis C virus. Pharmaceutical compositions, preparation methods of the compounds, and methods of using the compounds and compositions to treat viral infections are also provided.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UY0001033514A UY33514A (en) | 2011-07-13 | 2011-07-13 | GUANOSINE DERIVATIVE PHOSPHORAMIDATE NECLEOSID COMPOUNDS FOR TREATMENT OF VIRAL INFECTION |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UY0001033514A UY33514A (en) | 2011-07-13 | 2011-07-13 | GUANOSINE DERIVATIVE PHOSPHORAMIDATE NECLEOSID COMPOUNDS FOR TREATMENT OF VIRAL INFECTION |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY33514A true UY33514A (en) | 2013-02-28 |
Family
ID=47846604
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY0001033514A UY33514A (en) | 2011-07-13 | 2011-07-13 | GUANOSINE DERIVATIVE PHOSPHORAMIDATE NECLEOSID COMPOUNDS FOR TREATMENT OF VIRAL INFECTION |
Country Status (1)
| Country | Link |
|---|---|
| UY (1) | UY33514A (en) |
-
2011
- 2011-07-13 UY UY0001033514A patent/UY33514A/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20200813 |