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UY30956A1 - Imidazo- y triazolopirimidinas sustituidas - Google Patents

Imidazo- y triazolopirimidinas sustituidas

Info

Publication number
UY30956A1
UY30956A1 UY30956A UY30956A UY30956A1 UY 30956 A1 UY30956 A1 UY 30956A1 UY 30956 A UY30956 A UY 30956A UY 30956 A UY30956 A UY 30956A UY 30956 A1 UY30956 A1 UY 30956A1
Authority
UY
Uruguay
Prior art keywords
imidazo
substituted
triazolopirimidines
preparation
triazolopyrimidines
Prior art date
Application number
UY30956A
Other languages
English (en)
Inventor
Sperzel Michael
Strayle Jochen
Zubov Dmitry
Rester Ulrich
Heitmeier Stefan
Gnoth Mark Jean
Svenstrup Niels
Rihrig Susanne
Wilmen Andreas
Siegel Stephan
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of UY30956A1 publication Critical patent/UY30956A1/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Virology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Communicable Diseases (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Molecular Biology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)

Abstract

La invencion se refiere a imidazo-y triazolopirimidinas sustituidas, a procedimientos para su preparacion y a su uso para la preparacion de medicamentos para el tratamiento y/o profilaxis de enfermedades, en particular de trastornos hematologicos, preferiblemente de leucopenias y neutropenias.
UY30956A 2007-03-16 2008-03-11 Imidazo- y triazolopirimidinas sustituidas UY30956A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102007012645A DE102007012645A1 (de) 2007-03-16 2007-03-16 Substituierte Imidazo- und Triazolopyrimidine

Publications (1)

Publication Number Publication Date
UY30956A1 true UY30956A1 (es) 2008-10-31

Family

ID=39688187

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30956A UY30956A1 (es) 2007-03-16 2008-03-11 Imidazo- y triazolopirimidinas sustituidas

Country Status (13)

Country Link
US (2) US8273752B2 (es)
EP (1) EP2137188B1 (es)
JP (1) JP5400626B2 (es)
AR (1) AR065719A1 (es)
CA (1) CA2680697C (es)
CL (1) CL2008000703A1 (es)
DE (1) DE102007012645A1 (es)
ES (1) ES2387223T3 (es)
PA (1) PA8772101A1 (es)
PE (1) PE20081806A1 (es)
TW (1) TW200904819A (es)
UY (1) UY30956A1 (es)
WO (1) WO2008113469A2 (es)

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DE102007012645A1 (de) 2007-03-16 2008-09-18 Bayer Healthcare Ag Substituierte Imidazo- und Triazolopyrimidine
DE102008023801A1 (de) * 2008-05-15 2009-11-19 Bayer Schering Pharma Aktiengesellschaft Substituierte Imidazo- und Triazolopyrimidine, Imidazo- und Pyrazolopyrazine und Imidazotriazine
DE102008035552A1 (de) * 2008-07-30 2010-02-04 Bayer Schering Pharma Aktiengesellschaft Substituierte Pyridine und ihre Verwendung
ES2435804T3 (es) * 2009-02-13 2013-12-23 Bayer Intellectual Property Gmbh Pirimidinas condensadas como inhibidores de Akt
JP5503930B2 (ja) * 2009-09-18 2014-05-28 住友化学株式会社 ３−アミノ−１−ｔｅｒｔ−ブトキシカルボニルピペリジンの精製方法およびそのクエン酸塩
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NZ599323A (en) 2009-10-15 2014-06-27 Univ Monash Affinity ligands and methods for protein purification
EP2526102B1 (en) 2010-01-22 2017-03-08 Fundación Centro Nacional de Investigaciones Oncológicas Carlos III Inhibitors of PI3 kinase
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CN102791692B (zh) * 2010-03-12 2015-05-27 日本曹达株式会社 叔丁氧基羰基胺化合物的制造方法
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EP2582709B1 (de) 2010-06-18 2018-01-24 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
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TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
AU2011338339A1 (en) 2010-12-08 2013-06-27 Vanderbilt University Bicyclic pyrazole compounds as allosteric modulators of mGluR5 receptors
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
CN103987713A (zh) * 2011-10-12 2014-08-13 阵列生物制药公司 5,7-取代的咪唑并[1,2-c]嘧啶
PT3105218T (pt) 2014-02-13 2019-12-05 Incyte Corp Ciclopropilaminas como inibidores de lsd1
DK3105226T3 (da) 2014-02-13 2019-10-14 Incyte Corp Cyclopropylaminer som lsd1-inhibitorer
EP3105219B9 (en) 2014-02-13 2018-10-03 Incyte Corporation Cyclopropylamines as lsd1 inhibitors
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MX2016011784A (es) 2014-03-19 2016-12-02 Boehringer Ingelheim Int Nuevos heteroarilos y su uso como medicamentos.
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