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UY29875A1 - Compuestos quimicos - Google Patents

Compuestos quimicos

Info

Publication number
UY29875A1
UY29875A1 UY29875A UY29875A UY29875A1 UY 29875 A1 UY29875 A1 UY 29875A1 UY 29875 A UY29875 A UY 29875A UY 29875 A UY29875 A UY 29875A UY 29875 A1 UY29875 A1 UY 29875A1
Authority
UY
Uruguay
Prior art keywords
chemical compounds
compounds
warm
compositions
preparing
Prior art date
Application number
UY29875A
Other languages
English (en)
Inventor
Stinabritt Nilsson
Thomas G Hansson
Jan Dahmen
Lepisto Matti
Henriksson Krister
Hakan Bladh
Original Assignee
Astrazeneca Ab
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab, Schering Ag filed Critical Astrazeneca Ab
Publication of UY29875A1 publication Critical patent/UY29875A1/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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    • C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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Abstract

Compuestos de fórmula (I): o una sal farmacéuticamente aceptable del mismo; composiciones que los comprenden, procesos para prepararlos y su uso en terapia médica (por ejemplo modulando el receptor de glucocorticoides en un animal de sangre caliente)
UY29875A 2005-10-20 2006-10-19 Compuestos quimicos UY29875A1 (es)

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EP (1) EP1940800A4 (es)
JP (1) JP2009512687A (es)
AR (1) AR056877A1 (es)
CA (1) CA2628577A1 (es)
CL (1) CL2006002831A1 (es)
PE (1) PE20070712A1 (es)
TW (1) TW200815361A (es)
UY (1) UY29875A1 (es)
WO (1) WO2007046747A1 (es)

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DE10238722A1 (de) 2002-08-23 2004-03-11 Bayer Ag Selektive Phosphodiesterase 9A-Inhibitoren als Arzneimittel zur Verbesserung kognitiver Prozesse
GB0620385D0 (en) 2006-10-13 2006-11-22 Glaxo Group Ltd Novel compounds
EP2099767A1 (en) 2006-11-01 2009-09-16 Brystol-Myers Squibb Company Modulators of glucocorticoid receptor, ap-1, and/or nf- b activity and use thereof
TW200829578A (en) * 2006-11-23 2008-07-16 Astrazeneca Ab Chemical compounds 537
JO2754B1 (en) 2006-12-21 2014-03-15 استرازينكا ايه بي Amylendazoleil derivatives for the treatment of glucocorticoid-mediated disorders
GB0704407D0 (en) * 2007-03-07 2007-04-18 Glaxo Group Ltd Compounds
WO2008124665A1 (en) * 2007-04-10 2008-10-16 Boehringer Ingelheim International Gmbh Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
GB0720549D0 (en) * 2007-10-19 2007-11-28 Glaxo Group Ltd Novel compounds
GB0720557D0 (en) * 2007-10-19 2007-11-28 Glaxo Group Ltd Novel compounds
GB0720556D0 (en) * 2007-10-19 2007-11-28 Glaxo Group Ltd Novel compounds
PE20091211A1 (es) 2007-11-30 2009-09-14 Boehringer Ingelheim Int Derivados de pirazolopirimidina como moduladores de pde9a
GB0724254D0 (en) * 2007-12-12 2008-01-23 Glaxo Group Ltd Novel compounds
AU2009220458A1 (en) * 2008-03-06 2009-09-11 Merck Sharp & Dohme Corp. Hexahydrocyclopentyl[f]findazole sulfonamides and derivates thereof as selective glucocorticoid receptor modulators
CA2719018A1 (en) * 2008-03-20 2009-09-24 Abbott Laboratories Methods for making central nervous system agents that are trpv1 antagonists
UA105362C2 (en) 2008-04-02 2014-05-12 Бьорингер Ингельхайм Интернациональ Гмбх 1-heterocyclyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their use as pde9a modulators
WO2009142568A1 (en) * 2008-05-20 2009-11-26 Astrazeneca Ab Combination of (a) glucocorticoid receptor modulator and (b) a b2-agonist
TW200951114A (en) * 2008-05-20 2009-12-16 Astrazeneca Ab Phenyl or pyridinyl substituted indazoles derivatives
WO2009142588A1 (en) * 2008-05-20 2009-11-26 Astrazeneca Ab Combination of (a) a chemokine receptor 1 (ccr1) antagonist and (b) glucocorticoid receptor modulator
WO2009142589A1 (en) * 2008-05-20 2009-11-26 Astrazeneca Ab Combination of (a) glucocorticoid receptor modulator and (b) a muscarinic antagonist
CA2736304A1 (en) 2008-09-08 2010-03-11 Boehringer Ingelheim International Gmbh Pyrazolopyrimidines and their use for the treatment of cns disorders
GEP20146098B (en) 2009-03-31 2014-05-27 Boehringer Ingelheim Int 1-heterocyclyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their usage as pde9a modulators
MX344770B (es) 2010-08-12 2017-01-06 Boehringer Ingelheim Int Gmbh * Derivados de 6-cicloalquil-1,5-dihidro-pirazolo (3,4-d) pirimidin-4-onas y su uso como inhibidores de pde9a.
US8809345B2 (en) 2011-02-15 2014-08-19 Boehringer Ingelheim International Gmbh 6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders
US9149346B1 (en) * 2014-10-17 2015-10-06 Kelly Walter Lee Caldiero Method for synthetic polymer tooth replacement
KR102412146B1 (ko) 2015-02-11 2022-06-22 주식회사 아이엔테라퓨틱스 소디움 채널 차단제
WO2017161518A1 (en) 2016-03-23 2017-09-28 Astrazeneca Ab New physical form
WO2020144375A1 (en) 2019-01-11 2020-07-16 Grünenthal GmbH Substituted pyrrolidine amides iii

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US3992441A (en) * 1972-12-26 1976-11-16 Pfizer Inc. Sulfamylbenzoic acids
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PE20070712A1 (es) 2007-09-21
EP1940800A1 (en) 2008-07-09
CL2006002831A1 (es) 2008-02-22
AR056877A1 (es) 2007-10-31
CA2628577A1 (en) 2007-04-26
EP1940800A4 (en) 2009-12-30
TW200815361A (en) 2008-04-01
US20090124607A1 (en) 2009-05-14
WO2007046747A1 (en) 2007-04-26
JP2009512687A (ja) 2009-03-26

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