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UY26547A1 - AMIDE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES, AND THEIR METHOD OF USE - Google Patents

AMIDE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES, AND THEIR METHOD OF USE

Info

Publication number
UY26547A1
UY26547A1 UY26547A UY26547A UY26547A1 UY 26547 A1 UY26547 A1 UY 26547A1 UY 26547 A UY26547 A UY 26547A UY 26547 A UY26547 A UY 26547A UY 26547 A1 UY26547 A1 UY 26547A1
Authority
UY
Uruguay
Prior art keywords
pharmaceutical compositions
compounds
amide compounds
proteinkinases
inhibiting
Prior art date
Application number
UY26547A
Other languages
Spanish (es)
Inventor
Steven Lee Bender
Stephan James Cripps
Cynthia Louise Palmer
Michael David Varney
Dilip Bhumralkar
Michael Raymond Collins
Judith Gail Deal
Lei Jia
Michell David Nambu
Zhengwei Peng
Original Assignee
Agouron Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agouron Pharma filed Critical Agouron Pharma
Priority to UY26547A priority Critical patent/UY26547A1/en
Publication of UY26547A1 publication Critical patent/UY26547A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se describen los compuestos de las amidas que modulan y/o inhiben la actividad de ciertas proteínas cinasa. Estos compuestos y las composiciones farmacéuticas que los contienen son capaces de actuar como mediador de la senal de transducción de la tirosina cinasa con el fin de modular y/o inhibir la proliferación celular indeseada. La invención también va dirigida al uso terapéutico o profiláctico de las composiciones farmacéuticas que contienen dichos compuetos, y a los métodos para el tratamiento del cáncer y de otras enfermedades asociadas a la angiogénesis y/o proliferación celular indeseada, tal como lo son la retinopatía diabética, neovascularización del glaucoma, artritis reumatoide, y soriasis, mediante la administración de cantidades eficaces de dichos compuestos.The amide compounds that modulate and / or inhibit the activity of certain protein kinases are described. These compounds and the pharmaceutical compositions containing them are capable of acting as a mediator of the tyrosine kinase transduction signal in order to modulate and / or inhibit unwanted cell proliferation. The invention is also directed to the therapeutic or prophylactic use of pharmaceutical compositions containing said compounds, and to methods for the treatment of cancer and other diseases associated with angiogenesis and / or unwanted cell proliferation, such as diabetic retinopathy, neovascularization of glaucoma, rheumatoid arthritis, and psoriasis, by administering effective amounts of these compounds.

UY26547A 2001-01-19 2001-01-19 AMIDE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES, AND THEIR METHOD OF USE UY26547A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UY26547A UY26547A1 (en) 2001-01-19 2001-01-19 AMIDE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES, AND THEIR METHOD OF USE

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
UY26547A UY26547A1 (en) 2001-01-19 2001-01-19 AMIDE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES, AND THEIR METHOD OF USE

Publications (1)

Publication Number Publication Date
UY26547A1 true UY26547A1 (en) 2001-09-28

Family

ID=38812320

Family Applications (1)

Application Number Title Priority Date Filing Date
UY26547A UY26547A1 (en) 2001-01-19 2001-01-19 AMIDE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES, AND THEIR METHOD OF USE

Country Status (1)

Country Link
UY (1) UY26547A1 (en)

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20120814