UA89617C2 - Succinate and malonate salt of trans 4-(1r,3s)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and use thereof as a medicament - Google Patents
Succinate and malonate salt of trans 4-(1r,3s)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and use thereof as a medicamentInfo
- Publication number
- UA89617C2 UA89617C2 UAA200602709A UAA200602709A UA89617C2 UA 89617 C2 UA89617 C2 UA 89617C2 UA A200602709 A UAA200602709 A UA A200602709A UA A200602709 A UAA200602709 A UA A200602709A UA 89617 C2 UA89617 C2 UA 89617C2
- Authority
- UA
- Ukraine
- Prior art keywords
- phenylindan
- trimethylpiperazine
- chloro
- succinate
- trans
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
4-((1R,3S)-6-Chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine hydrogen succinate or hydrogen malonat, pharmaceutical compositions containing these salts and the medical use thereof, including for the treatment of schizophrenia and other psychotic disorders. Also described are methods for the preparation of 4-((1R,3S)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and medical uses thereof.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200301180 | 2003-08-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA89617C2 true UA89617C2 (en) | 2010-02-25 |
Family
ID=36701685
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200909651A UA108342C2 (en) | 2003-08-18 | 2004-08-18 | METHOD OF PREPARATION OF 4 - ((1R, 3S) -6-CHLORO-3-PHENYLINDAN-1-IL) -1,2,2-TRIMETHYLPIPERASINE OR ITS SALT (OPTIONS), CIS- (1S, 3S) -6-CHLORINE 3-PHENYLINDAN-1-OL, CIS- (1S, 3S) -3-REPLACED-5-CHLORINE-1-PHENYLINDAN AND TRANS-1 - ((1R, 3S) -6-CHLORINE-3-PHENYLINDAN-1-IL ) -3,3-DIMETHYLPIPERASINE |
| UAA200602709A UA89617C2 (en) | 2003-08-18 | 2004-08-18 | Succinate and malonate salt of trans 4-(1r,3s)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and use thereof as a medicament |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200909651A UA108342C2 (en) | 2003-08-18 | 2004-08-18 | METHOD OF PREPARATION OF 4 - ((1R, 3S) -6-CHLORO-3-PHENYLINDAN-1-IL) -1,2,2-TRIMETHYLPIPERASINE OR ITS SALT (OPTIONS), CIS- (1S, 3S) -6-CHLORINE 3-PHENYLINDAN-1-OL, CIS- (1S, 3S) -3-REPLACED-5-CHLORINE-1-PHENYLINDAN AND TRANS-1 - ((1R, 3S) -6-CHLORINE-3-PHENYLINDAN-1-IL ) -3,3-DIMETHYLPIPERASINE |
Country Status (4)
| Country | Link |
|---|---|
| CN (2) | CN1835938A (en) |
| ME (1) | ME00154B (en) |
| UA (2) | UA108342C2 (en) |
| ZA (2) | ZA200601421B (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102365265A (en) * | 2009-04-09 | 2012-02-29 | 欧加农股份有限公司 | Indane derivatives |
| CN103209949B (en) * | 2010-11-09 | 2016-08-10 | 株式会社钟化 | Halogenated indanones and method for producing optically active indanones or optically active indanols using the same |
| CN103429577A (en) * | 2011-01-07 | 2013-12-04 | H.隆德贝克有限公司 | Method for resolution of 4-((1R,3S)-6-chloro-3-phenyl-indan-1-yl)-1,2,2-trimethyl-piperazine and 1-((1R,3S)-6-chloro-3-phenyl-indan, 1-yl)-3,3-dimethyl-piperazine |
| CN112359078A (en) * | 2021-01-12 | 2021-02-12 | 凯莱英生命科学技术(天津)有限公司 | Chiral resolution method of isobutyrate compound |
-
2004
- 2004-08-18 CN CNA2004800236381A patent/CN1835938A/en active Pending
- 2004-08-18 UA UAA200909651A patent/UA108342C2/en unknown
- 2004-08-18 ME MEP-2008-26A patent/ME00154B/en unknown
- 2004-08-18 UA UAA200602709A patent/UA89617C2/en unknown
- 2004-08-18 ZA ZA200601421A patent/ZA200601421B/en unknown
- 2004-08-18 CN CN2004800237257A patent/CN1839124B/en not_active Expired - Fee Related
- 2004-08-18 ZA ZA200601173A patent/ZA200601173B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MEP2608A (en) | 2010-06-10 |
| UA108342C2 (en) | 2015-04-27 |
| ZA200601421B (en) | 2007-05-30 |
| CN1839124B (en) | 2010-06-16 |
| ME00154B (en) | 2010-10-10 |
| ZA200601173B (en) | 2007-04-25 |
| CN1835938A (en) | 2006-09-20 |
| CN1839124A (en) | 2006-09-27 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MXPA06001838A (en) | Succinate and malonate salt of trans-4-(ir, 3s)-6 -chloro- 3-phenylindan- 1-yl)-1, 2, 2- trimethylpiperazine and the use as a medicament. | |
| TW200503674A (en) | Therapeutic agents | |
| MY145590A (en) | Phenylacetamides and their use as glucokinase modulators | |
| DE50311898D1 (en) | FREDERICAMYCIN DERIVATIVES AS A MEDICAMENT FOR TUMOR TREATMENT | |
| CO5271691A1 (en) | NEW COMPOUNDS | |
| GEP20053673B (en) | Aryl or Heteroaryl Fused Imidazole Compounds as Anti-Inflammatory and Analgesic Agents | |
| TW200621762A (en) | Novel compounds | |
| IL164974A0 (en) | Novel compounds and their use | |
| WO2005037798A3 (en) | Amide or thiomide derivatives and their use in the treatment of pain | |
| DE602004011966D1 (en) | Heterocyclylverbindungen | |
| WO2003087049A3 (en) | Pharmaceutical combinations containing heterocyclic compounds and a novel anticholinergic agent | |
| NO20073176L (en) | New drugs for the treatment of respiratory diseases | |
| WO2004041802A8 (en) | 4(phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain or gastrointestinal disorders | |
| MXPA03000439A (en) | Novel form of (r)-n-[5- methyl-8-(4- methylpiperazin-1-yl) -1, 2, 3, 4-tetrahydro -2-naphthyl] -4-morpholinobenzamide. | |
| SE0300105D0 (en) | Diarylmethylidene piperdine derivatives, preparations thereof and uses thereof | |
| AU2001246999A1 (en) | New neurokinin antagonists for use as medicaments | |
| UA89617C2 (en) | Succinate and malonate salt of trans 4-(1r,3s)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and use thereof as a medicament | |
| MY139613A (en) | Novel piperazinyl-pyrazinone derivatives for the treatment of 5-ht2a receptor-related disorders | |
| TW200519098A (en) | Succinate and malonate salt of trans-4-((1R, 3S)-6-chloro-3-phenylindan-1-yl)-1, 2, 2-trimethylpiperazine and the use as a medicament | |
| MY148683A (en) | Crystalline base of trans-1-((1r,3s)-6-chloro-3-phenylindan-1-yl)-3,3-dimethylpiperazine | |
| AU2001244999A1 (en) | Naphthamide neurokinin antagonists for use as medicaments | |
| AU2003294952A1 (en) | 3,3-dimethyl-8-oxoisoquinolines for medical purposes, methods for the production thereof, medicaments containing said compounds and the use of the same | |
| SE0301442D0 (en) | Diarylmethylidene piperidine derivatives, preparations therof and uses thereof | |
| SE0403117D0 (en) | New compounds 1 | |
| TW200509915A (en) | Novel oxazoles, their manufacture and use as pharmaceutical agents |